专利检索 ap:("Okinawa Institute of Science AND Technology School Corporation") AND inv:"CHOUTHAIWALE, Pandurang Vilasrao" 第 1 页

1.

发明授权
4-SUBSTITUTED PYRIDINE-2,6-DICARBOXYLIC ACID DERIVATIVES AND METHOD OF PREPARING SAME 有权

公开(公告)号：EP3191451B1

公开(公告)日：2019-06-05

申请号：EP15840917.7

申请日：2015-09-09

申请人： Okinawa Institute of Science and Technology School Corporation

发明人： CHOUTHAIWALE, Pandurang Vilasrao , TANAKA, Fujie

IPC分类号： C07D213/79 , A61K31/4418 , A61P9/10 , A61P11/00 , A61P17/06 , A61P29/00 , A61P35/00

2.

发明公开
4-SUBSTITUTED PYRIDINE-2,6-DICARBOXYLIC ACID DERIVATIVES AND METHOD OF PREPARING SAME 审中-公开
标题翻译： 4-取代的吡啶-2,6-二羧酸衍生物及其制备方法

公开(公告)号：EP3191451A1

公开(公告)日：2017-07-19

申请号：EP15840917.7

申请日：2015-09-09

申请人： Okinawa Institute of Science and Technology School Corporation

发明人： CHOUTHAIWALE, Pandurang Vilasrao , TANAKA, Fujie

IPC分类号： C07D213/79 , A61K31/4418 , A61P9/10 , A61P11/00 , A61P17/06 , A61P29/00 , A61P35/00

CPC分类号： C07D213/79 , A61P35/00 , C07D213/803 , C07D405/04

摘要： The present invention relates to novel 4-substituted pyridine-2,6-dicarboxylic acid derivatives, compounds of formula I, wherein R1 and R2 are defined herein. The compounds of formula I are useful for making pharmaceutical compositions to treat proliferative diseases. The present invention also relates to concise methods for preparing compounds of formula I that may be performed under mild reaction conditions.

摘要翻译： 本发明涉及新的4-取代的吡啶-2,6-二羧酸衍生物，式I化合物，其中R1和R2在本文中定义。式I化合物可用于制备治疗增殖性疾病的药物组合物。本发明还涉及制备可在温和反应条件下进行的式I化合物的简明方法。