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公开(公告)号：EP4143196A1
公开(公告)日：2023-03-08
申请号：EP21795690.3
申请日：2021-04-29
发明人： BOEZIO, Alessandro , DIPIETRO, Lucian V. , FRIDRICH, Cary Griffin , GUNAYDIN, Hakan , KURUKULASURIYA, Ravi , LESCARBEAU, Andre , MADER, Mary M. , MCLEAN, Thomas H. , PIERCE, Levi Charles Thomas , RAYNOR, Kevin David , SHORTSLEEVES, Kelley C. , TANG, Yong , TAYLOR, Alexander M. , WALTERS, W. Patrick , ZHANG, Hanmo , GIORDANETTO, Fabrizio , PECHERSKY, Yakov , WANG, Qi , ATIENZA, Bren-Jordan , BERTRAND-LAPERLE, Megan , BURNIE, Andrew J. , CHEN, Fei , CHITALE, Sampada , GELOZIA, Shorena , GIGUERE, Jean-Benoit , LANDAGARAY, Elodie , LARIVEE, Alexandre , LEPITRE, Thomas , MAERTENS, Gaetan , OUTIN, Johanne , PAL, Mohan , STURINO, Claudio , TANVEER, Kashif , THORAT, Rakesh , VEMULA, Naresh , KRUEGER, Elaine B. , PAN, Yue , DENINNO, Michael Paul , BOUSQUET, Yves , JOBIN-DES LAURIERS, Antoine , LEE, Jessica , MOHAMED, Tarek
IPC分类号： C07D487/04
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公开(公告)号：EP3768668A1
公开(公告)日：2021-01-27
申请号：EP19715690.4
申请日：2019-03-21
发明人： TAYLOR, Alexander, M. , LESCARBEAU, André , KELLEY, Elizabeth, H. , SHORTSLEEVES, Kelley, C. , WALTERS, W., Patrick , MURCKO, Mark, Andrew , MCLEAN, Thomas, H. , GUNAYDIN, Hakan , GIORDANETTO, Fabrizio , THERRIEN, Eric
IPC分类号： C07D401/14 , C07D405/14 , C07D221/20 , C07D401/04 , C07D401/06 , C07D401/12 , C07D241/18 , C07D417/04 , C07D417/06 , C07D471/04 , C07D487/04 , C07D487/20 , C07D491/10 , C07D491/107 , C07D491/20
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公开(公告)号：EP4247816A1
公开(公告)日：2023-09-27
申请号：EP21895864.3
申请日：2021-11-17
发明人： MOUSTAKAS, Demetri T. , DIPIETRO, Lucian V. , SCHOENHERR, Heike , TOURÉ, Bakary-Barry , WALTERS, W. Patrick , MURCKO, Mark A. , KURUKULASURIYA, Ravi , PIERCE, Levi Charles Thomas , GIORDANETTO, Fabrizio , SHAN, Yibing , SAGAWA, Shiori , KRILOV, Goran , MCROBB, Fiona , THERRIEN, Eric
IPC分类号： C07D487/04 , A61K31/519 , C07H19/14
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公开(公告)号：EP3968999A1
公开(公告)日：2022-03-23
申请号：EP20805444.5
申请日：2020-05-12
发明人： TOURÉ, Bakary-Barry , SCHOENHERR, Heike , TAYLOR, Alexander M. , GIORDANETTO, Fabrizio , MOUSTAKAS, Demetri T. , MCLEAN, Thomas H. , HUDSON, Brandi M. , MADER, Mary M. , AYAZ, Pelin , SHARON, Dina A. , KURUKULASURIYA, Ravi , BOEZIO, Alessandro
IPC分类号： A61K31/519 , C07D487/04
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公开(公告)号：EP3768680A1
公开(公告)日：2021-01-27
申请号：EP19715687.0
申请日：2019-03-21
发明人： TAYLOR, Alexander, M. , GIORDANETTO, Fabrizio , GREISMAN, Jack, Benjamin , MARAGAKIS, Paul , SCHOENHERR, Heike
IPC分类号： C07D487/04 , C07D519/00 , A61K31/4985 , A61P43/00 , A61P7/00 , A61P3/10 , A61P35/00
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公开(公告)号：EP4306529A3
公开(公告)日：2024-04-10
申请号：EP23210430.7
申请日：2020-05-12
发明人： TOURÉ, Bakary-Barry , SCHOENHERR, Heike , TAYLOR, Alexander M. , GIORDANETTO, Fabrizio , MOUSTAKAS, Demetri T. , MCLEAN, Thomas H. , HUDSON, Brandi M. , MADER, Mary M. , AYAZ, Pelin , SHARON, Dina A. , KURUKULASURIYA, Ravi , BOEZIO, Alessandro
IPC分类号： C07D519/00 , C07D471/14 , C07D487/04 , C07D491/04 , C07D498/04 , C07D498/22 , A61P35/00 , C07D471/04
摘要： The present disclosure relates to novel compounds and pharmaceutical compositions thereof, and methods for inhibiting the activity of FGFR enzymes with the compounds and compositions of the disclosure. The present disclosure further relates to, but is not limited to, methods for treating disorders associated with FGFR signaling with the compounds and compositions of the disclosure.
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公开(公告)号：EP4399196A1
公开(公告)日：2024-07-17
申请号：EP22868344.7
申请日：2022-09-09
发明人： BOEZIO, Alessandro , TAYLOR, Alexander M. , GUNAYDIN, Hakan , ZHANG, Hanmo , RAYNOR, Kevin David , SHORTSLEEVES, Kelley C. , DIPIETRO, Lucian V. , PIERCE, Levi Charles Thomas , PABON, Nicolas , MCLEAN, Thomas H. , GIORDANETTO, Fabrizio , PECHERSKY, Yakov , WANG, Qi , LARIVEE, Alexandre , CHEN, Fei , MAERTENS, Gaetan , OUTIN, Johanne , BERTRAND-LAPERLE, Megan , PAL, Mohan , CHITALE, Sampada , DENINNO, Michael Paul
CPC分类号： A61P35/00
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公开(公告)号：EP4306529A2
公开(公告)日：2024-01-17
申请号：EP23210430.7
申请日：2020-05-12
发明人： TOURÉ, Bakary-Barry , SCHOENHERR, Heike , TAYLOR, Alexander M. , GIORDANETTO, Fabrizio , MOUSTAKAS, Demetri T. , MCLEAN, Thomas H. , HUDSON, Brandi M. , MADER, Mary M. , AYAZ, Pelin , SHARON, Dina A. , KURUKULASURIYA, Ravi , BOEZIO, Alessandro
IPC分类号： C07D519/00
摘要： The present disclosure relates to novel compounds and pharmaceutical compositions thereof, and methods for inhibiting the activity of FGFR enzymes with the compounds and compositions of the disclosure. The present disclosure further relates to, but is not limited to, methods for treating disorders associated with FGFR signaling with the compounds and compositions of the disclosure.
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公开(公告)号：EP3630770A1
公开(公告)日：2020-04-08
申请号：EP18731679.9
申请日：2018-05-25
发明人： TAYLOR, Alexander M. , LESCARBEAU, André , KELLEY, Elizabeth H. , SHORTSLEEVES, Kelley C. , DIPIETRO, Lucian V. , WALTERS, W. Patrick , MURCKO, Mark Andrew , PIERCE, Levi Charles Thomas , TANG, Yong , GIORDANETTO, Fabrizio , GREISMAN, Jack Benjamin , MARAGAKIS, Paul , BHAT, Sathesh , DAHLGEREN, Markus Kristofer , THERRIEN, Eric
IPC分类号： C07D487/04 , C07D519/00 , A61K31/4985 , A61P35/00 , A61P3/00 , A61P7/00
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公开(公告)号：EP3515916A1
公开(公告)日：2019-07-31
申请号：EP17781244.3
申请日：2017-09-22
发明人： ALBRECHT, Brian K. , GIORDANETTO, Fabrizio , GREISMAN, Jack, Benjamin , MARAGAKIS, Paul , TAYLOR, Alexander M. , WALTERS, W. Patrick
IPC分类号： C07D487/04 , A61K31/4985 , A61K31/55 , C07D498/10 , A61P9/00 , A61P35/00
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