公开(公告)号：EP1187810A2

公开(公告)日：2002-03-20

申请号：EP00937830.8

申请日：2000-05-25

申请人： SEPRACOR, INC.

发明人： CUNY, Gregory, D. ,  SHAO, Liming ,  HAUSKE, James, R. ,  HEFFERNAN, Michele, L., R. ,  AQUILA, Brian, M. ,  WU, Xinhe ,  WANG, Fengjian ,  BANNISTER, Thomas, D.

IPC分类号： C07D211/26 ,  C07D211/60 ,  C07D211/56 ,  C07D241/04 ,  C07D265/30 ,  C07D267/10 ,  C07D223/04 ,  C07D223/12 ,  C07D243/06 ,  C07D205/04 ,  C07D207/09 ,  C07D207/16 ,  C07D491/10 ,  A61K31/445 ,  A61K31/397 ,  A61K31/40 ,  A61K31/535 ,  A61K31/55 ,  A61K31/551 ,  A61K31/553 ,  A61P25/04

CPC分类号： C07D221/04 ,  C07D205/04 ,  C07D211/26 ,  C07D211/42 ,  C07D211/56 ,  C07D223/04 ,  C07D241/04 ,  C07D243/08 ,  C07D265/30 ,  C07D267/10 ,  C07D401/06 ,  C07D401/12 ,  C07D405/12 ,  C07D405/14 ,  C07D409/06 ,  C07D409/12 ,  C07D491/10

摘要： One aspect of the present invention relates to novel heterocyclic compounds. A second aspect of the present invention relates to the use of the novel heterocyclic compounds as ligands for various cellular receptors, including opiate receptors, other the G-protein coupled receptors, and ion channels. An additional aspect of the present invention relates to the use of the novel heterocyclic compounds as analgesics.