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1.发明授权Antibacterial mycaminosyl tylonolide derivatives and their production 失效抗菌素MYCAMINOSYL TYLONOLIDE衍生物及其生产
公开(公告)号：EP0202111B1
公开(公告)日：1989-09-13
申请号：EP86303633.1
申请日：1986-05-13
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公开(公告)号：EP0159881B1
公开(公告)日：1989-03-01
申请号：EP85302583.1
申请日：1985-04-12
发明人： Umezawa, Hamao , Umezawa, Sumio , Tsuchiya, Tsutomu , Takeuchi, Tomio , Tanaka, Akihiro , Sakamoto, Shuichi
CPC分类号： C07H17/08
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3.发明公开Tylosin derivatives, their preparation and pharmaceutical compositions containing them 失效泰乐菌素衍生物及其制备和含有它们的药物组合物
公开(公告)号：EP0132895A1
公开(公告)日：1985-02-13
申请号：EP84201085.2
申请日：1982-07-09
发明人： Umezawa, Hamao , Umezawa, Sumio , Tsuchiya, Tsutomu , Takeuchi, Tomio , Tanaka, Akihiro , Iwamoto, Hidenori , Sakamoto, Shuichi
CPC分类号： C07H17/08
摘要： A tylosin derivative represented by the general formula
wherein R. represents a hydrogen atom or a hydroxyl group and R. represents
(wherein R 9 and R 10 may be the same or different and selected from a hydrogen atom and C, to C. alkyl groups or which may together form an alkylene group having 3-7 carbon atoms) or -S-R 11 (wherein R " represents a furanyl group or a pyridyl group).摘要翻译： 由通式表示的泰乐菌素衍生物，其中R表示氢原子或羟基，并且R表示（其中R9和R10可以相同或不同并且选自氢原子和C，至C的烷基，或者 可以一起形成具有3-7个碳原子的亚烷基）或-S-R11（其中R“表示呋喃基或吡啶基）。
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公开(公告)号：EP0347158A2
公开(公告)日：1989-12-20
申请号：EP89305945.1
申请日：1989-06-13
CPC分类号： C07H17/08
摘要： 3-Deoxy mycaminosyl tylonolide derivatives represented by the following general formula and salts thereof:
wherein X represents an oxygen atom or =N-OR⁴ (wherein R⁴ represents hydrogen or lower alkyl); R¹ represents a hydrogen atom, an acyl group or an alkylsilyl group; R² represents a hydrogen atom or an acyl group; and R³ represents a hydrogen atom or a hydroxyl group. The compounds of formula (I) have excellent antibacterial activity.摘要翻译： 由下列通式表示的3-脱氧碳霉糖基太乐内酯衍生物及其盐：其中X代表氧原子或= N-OR 4（其中R 4代表氢或低级烷基）; R 1代表氢原子，酰基或烷基甲硅烷基; R 2代表氢原子或酰基; R 3代表氢原子或羟基。 式（I）化合物具有优异的抗菌活性。
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公开(公告)号：EP0347158A3
公开(公告)日：1990-04-25
申请号：EP89305945.1
申请日：1989-06-13
CPC分类号： C07H17/08
摘要： 3-Deoxy mycaminosyl tylonolide derivatives represented by the following general formula and salts thereof:
wherein X represents an oxygen atom or =N-OR⁴ (wherein R⁴ represents hydrogen or lower alkyl); R¹ represents a hydrogen atom, an acyl group or an alkylsilyl group; R² represents a hydrogen atom or an acyl group; and R³ represents a hydrogen atom or a hydroxyl group. The compounds of formula (I) have excellent antibacterial activity.-
7.发明公开
公开(公告)号：EP0202111A1
公开(公告)日：1986-11-20
申请号：EP86303633.1
申请日：1986-05-13
发明人： Umezawa, Hamao , Umezawa, Sumio , Tsuchiya, Tsutomu , Takeuchi, Tomio , Tanaka, Akihiro , Sakamoto, Shuichi
摘要： Mycaminosyl tylonolide derivatives represented by the following general formula
(wherein R 1 is a hydroxyl, lower alkanoyloxy, benzoyloxy, or azido group, or an amino group optionally substituted with lower alkyl and/or lower alkanoyl group(s); R 2 is a hydrogen atom or hydroxyl group; R 3 is a hydrogen atom or formyl group; and means a double bond or the group ), and salts thereof. These compounds have antibacterial activity.-
公开(公告)号：EP0159881A2
公开(公告)日：1985-10-30
申请号：EP85302583.1
申请日：1985-04-12
发明人： Umezawa, Hamao , Umezawa, Sumio , Tsuchiya, Tsutomu , Takeuchi, Tomio , Tanaka, Akihiro , Sakamoto, Shuichi
CPC分类号： C07H17/08
摘要： Novel 23-C-substituted mycaminosyl tylonolide of the general formula (I)
wherein R 1 represents a lower alkyl group, an aryl group, a lower alkenyl group or a lower alkinyl group, R 2 represents a hydrogen atom or a hydroxyl group.
These compounds have excellent antibacterial activities.摘要翻译： 通式（I）的新型23-C取代的碳霉糖基太乐内酯
其中R 1表示低级烷基，芳基，低级链烯基或低级炔基，R 2表示氢 原子或羟基。 这些化合物具有优良的抗菌活性。 -
9.发明公开Tylosin derivatives, their preparation and pharmaceutical compositions containing them 失效泰乐菌素的衍生物，它们的制备和含有它们的药物组合物。
公开(公告)号：EP0134054A1
公开(公告)日：1985-03-13
申请号：EP84201086.0
申请日：1982-07-09
发明人： Umezawa, Hamao , Umezawa, Sumio , Tsuchiya, Tsutomu , Takeuchi, Tomio , Tanaka, Akihiro , Iwamoto, Hidenori , Sakamoto, Shuichi
CPC分类号： C07H17/08
摘要： A tylosin derivative represented by the general formula
wherein R 4 represents a hydrogen atom or a hydroxyl group.摘要翻译： 由通式
worin R4表示的泰乐菌素衍生物darstellt氢原子或羟基。
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