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12 条记录 (耗时 0.011 秒)

    Imino-benzyl-pyrazoles
    2.
    发明授权
    Imino-benzyl-pyrazoles 失效
    亚硝基 - 吡咯烷酮

    公开(公告)号：US3714182A

    公开(公告)日：1973-01-30

    申请号：US3714182D

    申请日：1970-08-19

    申请人： USV PHARMA CORP

    发明人： BANDURCO V ,  SHROFF J

    IPC分类号： C07D231/12 ,  C07D231/14 ,  C07D521/00 ,  C07D49/36

    CPC分类号： C07D231/12 ,  C07D231/14 ,  C07D233/56 ,  C07D249/08

    摘要： WHEREIN R is alkyl, cycloalkyl, phenyl, substituted phenyl or phenylalkyl, R1 is hydrogen, halogen, alkyl, trifluoromethyl, alkoxy, hydroxy or amino, R2 is alkyl, phenylalkyl or carbalkoxy, and R3 is hydrogen, alkyl, phenyl or substituted phenyl possess hypoglycemic activity.

    Compounds of the formula

    摘要翻译： 式WHEREIN R的化合物是烷基，环烷基，苯基，取代的苯基或苯基烷基，R1是氢，卤素，烷基，三氟甲基，烷氧基，羟基或氨基，R2是烷基，苯基烷基或烷氧基，R3是氢，烷基， 或取代的苯基具有降血糖活性。

    Styrene ethers of amino alcohols
    3.
    发明授权
    Styrene ethers of amino alcohols 失效
    氨基醇的苯乙烯

    公开(公告)号：US3651067A

    公开(公告)日：1972-03-21

    申请号：US3651067D

    申请日：1970-04-15

    申请人： USV PHARMA CORP

    发明人： ELPERN BILL ,  BANDURCO VICTOR T

    IPC分类号： C07D295/088 ,  C07D29/18

    CPC分类号： C07D295/088

    摘要： COMPOUNDS OF THE FORMULA

    (R"-N(-R"'')-X-O-CH2-C(=CH2)-),R,R''-BENZENE

    WHEREIN X IS A LOWER ALKYLENE HAVING FROM 2-5 CARBON ATOMS, R AND R'' ARE HYDROGEN, LOWER ALKYL, LOWER ALKOXY OR HALOGEN, R" AND R"'' ARE HYDROGEN, LOWER ALKYL OR PHENYL LOWER ALKYL, AND R" AND R"'' TAKEN TOGETHER WITH N MAY BE PIPERIDINO, MORPHOLINO, THIOMORPHOLINO, PYRROLIDINO, OR METHYLPIPERAZINO, ARE POTENT ANTICONVULSANTS, USEFUL IN THE TREATMENT OF GRAND MAL.

    Carbamoyl oximes
    5.
    发明授权
    Carbamoyl oximes 失效
    碳水化合物

    公开(公告)号：US3636111A

    公开(公告)日：1972-01-18

    申请号：US3636111D

    申请日：1969-11-18

    申请人： USV PHARMA CORP

    发明人： KARTEN MARVIN J

    IPC分类号： C07D295/125 ,  C07C131/00

    CPC分类号： C07D295/125

    摘要： COMPOUNDS OF THE FORMULA

    R1-C(-Y-X)=N-OOC-N(-R2)-R3

    WHEREIN R1 AND R2 ARE LOWER ALIPHATIC, CYCLOALKYL, OR AROMATIC (INCLUDING HETERO), R2 IS HYDROGEN, AROMATIC, LOWER ALIPHATIC, OR PHENYL-LOWER ALKYL, Y IS AN ALKYLENE GROUP HAVING FROM 1-5 CARBON ATOMS, AND X IS A SECONDARY AMINO GROUP, HAVE POTENT ANALGESIC ACTIVITY, PARTICULARLY WHEN R3IS A P-ALKOXYPHENYL (E.G.P-METHOXYPHENYL AND P-ETHOXYPHENYL). COMPOUNDS WHEREIN BOTH R1 AND R3 ARE PHENYL EXHIBIT ANTICONVULSANT ACTIVITY. COMPOUNDS WHERE R1 IS PHENYL OR 4-CHLOROPHENYL AND R3 IS CYCLOAKYL, SUCH AS CYCLOHEXYL, SHOW TOPICAL ANESTHETIC ACTIVITY. A NUMBER OF COMPOUNDS ALSO HAVE HYPOTENSIVE ACTIVITY.

    Oximo tetracyclic indoles
    7.
    发明授权
    Oximo tetracyclic indoles 失效
    OXIMO TETRACYCLIC INDOLES

    公开(公告)号：US3838135A

    公开(公告)日：1974-09-24

    申请号：US29865872

    申请日：1972-10-18

    申请人： USV PHARMA CORP

    发明人： MAGNIEN E ,  CABILIO J

    IPC分类号： C07D471/06 ,  C07D33/50

    CPC分类号： C07D471/06

    摘要： COMPOUNDS OF THE STRUCTURE

    1,2-(-(CH2)N-),6-(R3-N(-R4)-X-O-N=),R1,R2-5,6-DIHYDRO-4H-

    PYRROLO(3,2,1-IJ)QUINOLINE

    WHEREIN N IS AN INTEGER FROM 4-6, R1 IS HYDROGEN, LOWER ALKYL, LOWER ALKOXY, OR HALOGEN, R2 IS HYDROGEN OR LOWER ALKYL, R3 AND R4 ARE LOWER ALKYL OR CYCLOALKYL OR TAKEN TOGETHER WITH THE N TO WHICH THEY ARE ATTACHED, ARE PYRROLIDINO, PIPERIDINO, MORPHOLINO, OR PIPERAZINO, HAVE HYPOTENSIVE ACTIVITY.

    O-(substituted carbamoyl)-3-pyrrolidinopropio and butyrophenone oximes
    8.
    发明授权
    O-(substituted carbamoyl)-3-pyrrolidinopropio and butyrophenone oximes 失效
    O-（取代的羰基）-3-吡咯烷酮和丁基酚氧化物

    公开(公告)号：US3823159A

    公开(公告)日：1974-07-09

    申请号：US14137471

    申请日：1971-05-07

    申请人： USV PHARMA CORP

    发明人： KARTEN M

    IPC分类号： C07D295/125 ,  C07D27/04

    CPC分类号： C07D295/125

    摘要： COMPOUNDS OF THE FORMULA

    X-Y-C(-R1)=N-O-CO-N(-R2)-R3

    WHEREIN R1 AND R3 ARE LOWER ALIPHATIC, CYCLOALKYL, OR AROMATIC (INCLUDING HETERO), R2 IS HYDROGEN, AROMATIC, LOWER ALIPHATIC, OR PHENYL-LOWER ALKYL, Y IS AN ALKYLENE GROUP HAVING FROM 1-5 CARBON ATOMS, AND X IS A HETEROCYCLIC SECONDARY AMINO GROUP, AHVING POTENT ANALGESIC ACTIVITY.

    1,4-disubstituted piperazines
    9.
    发明授权
    1,4-disubstituted piperazines 失效
    1,4-取代的哌嗪

    公开(公告)号：US3793322A

    公开(公告)日：1974-02-19

    申请号：US3793322D

    申请日：1972-12-15

    申请人： USV PHARMA CORP

    发明人： SHROFF J ,  BANDURCO V

    IPC分类号： C07D295/195 ,  C07D295/205 ,  C07D51/70

    CPC分类号： C07D295/195 ,  C07D295/205 ,  Y10S514/866

    摘要： PIPERAZINE DERIVATIVES OF THE FORMULA

    1-((R,R''-PHENYL)-C(=N-R")-),4-R"''-PIPERAZINE

    WHEREIN R AND R'' ARE HYDROGEN, HYDROXY, LOWER ALKYL, LOWER ALKOXY HALOGEN OR TRIFLUOROMETHYL, R" IS LOWER ALKYL, LOWER ALKENYL, CYCLOALKYL OR PHENYL OR R"'' IS HYDROGEN, LOWER ALKYL, LOWER ALKENYL, CARBOALKOXY, FORMYL, BENZYL, OR CINNAMYL HAVE POTENT HYPOGLYCEMIC ACTIVITY.

    N-amino-benzamidines
    10.
    发明授权
    N-amino-benzamidines 失效
    N-氨基苯甲胺

    公开(公告)号：US3715396A

    公开(公告)日：1973-02-06

    申请号：US3715396D

    申请日：1969-11-04

    申请人： USV PHARMA CORP

    发明人： BANDURCO V ,  ELPERN B ,  SHROFF J

    IPC分类号： C07C259/20 ,  C07C123/00

    CPC分类号： C07C259/20

    摘要： Compounds of the formula WHEREIN R is hydrogen, alkyl, acyl, phenyl-lower alkyl, carbamoyl, benzoyl, R1 is lower alkyl, pyridyl, naphthyl, or cycloalkyl, R2 is phenyl or substituted phenyl, and R3 and R4 are hydrogen, lower alkyl, phenyl or phenyl-lower alkyl, or taken together are alkylene, possess anti-inflammatory activity.

    摘要翻译： 式WHEREIN R的化合物是氢，烷基，酰基，苯基 - 低级烷基，氨基甲酰基，苯甲酰基，R1是低级烷基，吡啶基，萘基或环烷基，R2是苯基或取代的苯基，R3和R4是氢， ，苯基或苯基 - 低级烷基，或一起为亚烷基，具有抗炎活性。