公开(公告)号：US20070111889A1

公开(公告)日：2007-05-17

申请号：US10580990

申请日：2004-12-17

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagne ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagne ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and may be substituted as defined in the description; L is halogen, cyano, alkyl, haloalkyl, alkoxy, alkenyloxy or alkoxycarbonyl; m is 1, 2, 3 or 4, where the groups L may be different if m is greater than 1; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi

摘要翻译： 其中取代基如下定义的式I的三唑并嘧啶：R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基， 卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1， 和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，其通过N连接并且可以含有另外的杂原子，由O ，N和S作为环成员，并且可以如说明书中所定义的取代; L是卤素，氰基，烷基，卤代烷基，烷氧基，烯氧基或烷氧基羰基; m为1,2,3或4，其中如果m大于1，则基团L可以不同; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途

公开(公告)号：US20070015770A1

公开(公告)日：2007-01-18

申请号：US10574499

申请日：2004-10-08

申请人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N37/12 ,  A01N37/44

CPC分类号： A01N43/90 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures for controlling rice pathogens. Said mixtures comprise as the active components 1) the triazolopyrimidine derivative of formula (I), and 2) metalaxyl-M of formula (II), in a synergistically effective amount. The invention also relates to a method for controlling rice pathogens using mixtures of compound (I) with the compounds (II) and to the use of compound (I) together with the compounds (II) for producing said mixtures, and to agents containing said mixtures.

摘要翻译： 本发明涉及用于防治水稻病原体的杀真菌混合物。 所述混合物以协同有效量包含作为活性组分的1）式（I）的三唑并嘧啶衍生物和2）式（II）的甲霜灵-M。 本发明还涉及使用化合物（I）与化合物（II）的混合物和化合物（I）与化合物（II）一起用于生产所述混合物的方法来控制水稻病原体的方法，以及含有所述 混合物。

公开(公告)号：US20080248952A1

公开(公告)日：2008-10-09

申请号：US11631004

申请日：2005-07-06

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90 ,  A01N25/00

CPC分类号： A01N43/90 ,  C07D487/04

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or a group R1, R1 and R2 together with the nitrogen atom, to which they are attached, may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and which may comprise one to three further heteroatoms from the groups consisting of O, N and S as ring member and/or may be substituted according to the description; L is fluorine, chlorine or methyl; X is cyano, C1-C4-alkyl, C1-C4-alkoxy or C1-C2-haloalkoxy, where X is not methyl if R1 and R2 together are n-pentylene or 3-methyl-n-pentylene and L is fluorine, or R1 and R2 together are 3-methyl-n-pentylene and L is chlorine; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义：式I的取代三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基， 包含一至四个由O，N和S组成的组的杂原子的五或六元饱和的部分不饱和或芳族杂环，R 2是氢或基团R 1， R 1，R 2和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，它们是 通过N连接并且其可以包含一个至三个由O，N和S组成的基团的另外的杂原子作为环成员和/或可以根据描述被取代; L是氟，氯或甲基; X是氰基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基或C 1 -C 4 - 如果R 1和R 2一起都是正 - 亚戊基，其中X不是甲基，其中X不是甲基 或3-甲基 - 正戊烯，L是氟，R 1和R 2一起是3-甲基 - 正戊烯，L是氯; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070249634A1

公开(公告)日：2007-10-25

申请号：US11597409

申请日：2005-06-08

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bern Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Petere Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Liliana Rapado ,  Michael Rack ,  Barbara Nave ,  Maria Schere ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bern Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Petere Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Liliana Rapado ,  Michael Rack ,  Barbara Nave ,  Maria Schere ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01P3/00

CPC分类号： A01N43/90

摘要： The invention relates to the use of triazolopyrimidines of the formula I In which: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl, C3-C6-cycloalkynyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N and S, where R1, R2 may be substituted as defined in the description or R1 and R2 together with the nitrogen atom to which they are attached may form five- to eight-membered heterocyclyl or heteroaryl which is attached via nitrogen and may contain one, two or three further heteroatoms from the group consisting of O, N and S as ring members and/or may be substituted as defined in the description; L independently of one another are halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyloxy, cyano, C(═O)A1, S(═O)mA2, NRcRd or NRc—(C═O)—Rd, where A1, A2, Rc, Rd and m are as defined in the description; L1 is halogen, alkyl or haloalkyl; L2 is nitro, a group —C(S)NR3R4, a group —C(═N—OR5)(NR6R7) or a group —C(═N—NR8R9)(NR10OR11); X is halogen, cyano, alkyl, alkoxy, haloalkyl or haloalkoxy; R3, R4, R5, R6, R7, R8, R9, R10 and R11 are independently of one another selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl and alkynyl, where the 4 last-mentioned radicals may be substituted as defined in the description; or R3 and R4, or R6 and R7, or R8 and R9 or R10 and R11 together with the nitrogen atom to which they are attached form a four, five, or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; n is 0, 1, 2 or 3; and the agriculturally acceptable salts thereof, novel triazolopyrimidines, crop protection compositions comprising at least one compound of the formula I and at least one solid or liquid carrier, and a method for controlling phytopathogenic harmful fungi.

公开(公告)号：US20070197389A1

公开(公告)日：2007-08-23

申请号：US10589496

申请日：2005-02-24

申请人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： A01N43/713 ,  C07D487/02

CPC分类号： C07D487/04

摘要： The invention relates to azolopyrimidine compounds of general formula (I), wherein A represents N or C—R6; X and Y, independent of one another, represent a chemical compound or oxygen, sulphur or a group N—R7; the variables R1, R2, R3, R4, R5, R6 and R7 have the meanings cited in the claims and the description. The invention also relates to tautomers of compounds of formula (I) and to the agriculturally compatible salts of compounds (I) and of the tautomers thereof. The invention further relates to the use of azolopyrimidine compounds of general formula (I), to the tautomers thereof and to the agriculturally compatible salts thereof which are used to combat phytopathogenic fungi, and to a method for combating phytopathogenic fungi and means for combating fungi, said means containing at least one compound of general formula (I), a tautomer of formula (I) and/or an agriculturally compatible salt thereof or the tautomer thereof and at least one liquid or solid carrier medium.

摘要翻译： 本发明涉及通式（I）的偶氮嘧啶化合物，其中A代表N或C-R 6; X和Y彼此独立地表示化合物或氧，硫或基团N-R 7; 变量R 1，R 2，R 3，R 4，R 5，...，SUP >，R 6和R 7具有权利要求书和说明书中引用的含义。 本发明还涉及式（I）化合物和化合物（I）的农业相容盐及其互变异构体的互变异构体。 本发明还涉及通式（I）的偶氮嘧啶化合物与其互变异构体及其与植物致病真菌的农业相容盐的用途，以及用于防治植物病原性真菌的方法和对抗真菌的方法， 所述方法含有至少一种通式（I）的化合物，式（I）的互变异构体和/或其农业上相容的盐或其互变异构体和至少一种液体或固体载体介质。

公开(公告)号：US20070185099A1

公开(公告)日：2007-08-09

申请号：US11628852

申请日：2005-06-24

申请人： Carsten Blettner ,  Frank Schieweck ,  Jordi i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Carsten Blettner ,  Frank Schieweck ,  Jordi i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： A01N43/90 ,  C07D487/04

摘要： The present invention relates to novel triazolopyrimidine compounds of the formula I in which: X is halogen, cyano, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C2-haloalkoxy; W is oxygen or sulfur; Y is O—R4 or a group NR5R6; A is a chemical bond or a group CR7R8; and the variables L, R1 to R7 are as defined in claim 1. The present invention furthermore provides the use of the triazolopyrimidine compounds of the formula I, their tautomers and their agriculturally acceptable salts for controlling phytopathogenic fungi (=harmful fungi) and a method for controlling phytopathogenic harmful fungi, which method comprises treating the fungi or the materials, plants, the soil or seed to be protected against fungal attack with an effective amount of a compound of the formula I, a tautomer of I and/or an agriculturally acceptable salt of I or a tautomer thereof.

摘要翻译： 本发明涉及新的式I的三唑并嘧啶化合物，其中：X为卤素，氰基，C 1 -C 4 - 烷基，C 1〜 C 1 -C 4 - 低级烷基，C 1 -C 4 - 烷氧基或C 1 -C 3 > 2 - 卤代烷氧基; W是氧或硫; Y是O-R 4或NR 5或R 6基团; A是化学键或基团CR 7 R 8; 变量L，R 1至R 7如权利要求1中所定义。本发明还提供式I的三唑并嘧啶化合物，其互变异构体和 其用于控制​​植物病原真菌（=有害真菌）的农业上可接受的盐和控制植物病原性有害真菌的方法，所述方法包括用有效量的有效量处理待保护的真菌或植物，土壤或种子免受真菌侵袭 式I的化合物，I的互变异构体和/或I的农业上可接受的盐或其互变异构体。

公开(公告)号：US20070161655A1

公开(公告)日：2007-07-12

申请号：US10587915

申请日：2005-02-19

申请人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N41/12

CPC分类号： A01N43/90 ,  A01N47/04 ,  A01N2300/00

摘要： Fungicidal mixtures for controlling harmful fungi, which mixtures comprise, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) dichlofluanid of the formula II in a synergistically effective amount, methods for controlling phytopathogenic harmful fungi using mixtures of the compound I with the compound II and the use of the compound I+with the compound II for preparing such mixtures, and also compositions comprising these mixtures.

摘要翻译： 用于控制有害真菌的杀真菌混合物，其混合物包含作为活性成分的1）式I的三氮代嘧啶衍生物和2）协同有效量的式II的二氯联苯，使用化合物I的混合物控制植物病原性有害真菌的方法 化合物II和化合物I +与化合物II用于制备这种混合物的用途，以及包含这些混合物的组合物。

公开(公告)号：US20070105873A1

公开(公告)日：2007-05-10

申请号：US10564013

申请日：2004-07-15

申请人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： A01N43/54

CPC分类号： C07D239/42

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R1 to R3 and L are as defined in the description and R4 corresponds to one of the formulae in which Ra, X and Rb are as defined in the description; and also to processes for preparing these compounds, to pesticidal compositions comprising these compounds and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基R 1至R 3和L如说明书中所定义， SUP> 4 对应于其中R a，S，X和R b的定义之一如说明书中所定义; 以及制备这些化合物的方法，包括这些化合物的农药组合物及其作为农药的用途。

公开(公告)号：US20070071833A1

公开(公告)日：2007-03-29

申请号：US10574509

申请日：2004-10-08

申请人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N59/02 ,  A01N43/90

CPC分类号： A01N43/90 ,  A01N59/02 ,  A01N2300/00

摘要： Fungicidal mixtures for controlling rice pathogens, which mixtures comprise, as active components, 1) the triazolopyrimidine derivative of the formula I, and 2) sulfur (II), in a synergistically effective amount, methods for controlling rice pathogens using mix-tures of the compound I with sulfur (II), the use of the compound I with sulfur (II) for preparing such mixtures and compositions comprising these mixtures are described.

摘要翻译： 用于控制水稻病原体的杀真菌混合物，其混合物包含作为活性组分的1）式I的三氮代嘧啶衍生物和2）硫（II），协同有效量的方法，用于控制水稻病原体的混合物 化合物I与硫（II），描述了化合物I与硫（II）用于制备这些混合物的使用和包含这些混合物的组合物。

公开(公告)号：US20060293346A1

公开(公告)日：2006-12-28

申请号：US10573288

申请日：2004-09-30

申请人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N43/42

CPC分类号： A01N43/42 ,  A01N43/90 ,  A01N2300/00

摘要： Fungicidal mixtures comprising, as active components, 1) the triazolopyrimidine derivative of the formula I 2) quinoxyfen of the formula II in a synergistically effective amount, methods for controlling harmful fungi from the class of the Oomycetes using mixtures of the compound I with the compound II, the use of the compound I with the compound II for preparing such mixtures and compositions comprising these mixtures are described.

摘要翻译： 包含作为活性组分的1）式I的三氮代嘧啶衍生物2）协同有效量的式II的喹喔啉的方法，使用化合物I与化合物的混合物来控制来自卵菌纲的有害真菌的方法 II，描述了化合物I与化合物II用于制备这种混合物的使用和包含这些混合物的组合物。