公开(公告)号：US20080274883A1

公开(公告)日：2008-11-06

申请号：US11793796

申请日：2005-12-21

Applicant: Markus Gewehr ,  Reinhard Stierl ,  Matthias Niedenbruck ,  Udo Hunger

Inventor： Markus Gewehr ,  Reinhard Stierl ,  Matthias Niedenbruck ,  Udo Hunger

IPC: A01N43/84 ,  A01N25/00 ,  A01P3/00

CPC classification number: A01N37/10 ,  A01N2300/00

Abstract: Fungicidal mixtures comprising 1) enestroburin of formula I: and 2) dimethomorph of formula II: as active components in a synergistically effective amount, method of controlling harmful fungi using mixtures of compound I with compound II, use of compound I with compound II for the preparation of such mixtures, and compositions comprising these mixtures.

Abstract translation: 杀真菌混合物，其包含1）式I的地芬布林和2）式II的烯酰吗啉：以协同有效量作为活性成分，使用化合物I与化合物II的混合物来控制有害真菌的方法，将化合物I与化合物II用于 这些混合物的制备和包含这些混合物的组合物。

公开(公告)号：US20080249113A1

公开(公告)日：2008-10-09

申请号：US11659192

申请日：2005-07-28

Applicant: Carsten Blettner ,  Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Carsten Blettner ,  Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04 ,  A01N25/26 ,  A01P3/00

CPC classification number: A01N43/90 ,  A01N43/653 ,  A01N47/14 ,  A01N43/50 ,  A01N57/12 ,  A01N47/04 ,  A01N37/34 ,  A01N43/40 ,  A01N37/50 ,  A01N37/46 ,  A01N43/84 ,  A01N37/38 ,  A01N43/28 ,  A01N47/38 ,  A01N43/54 ,  A01N43/32 ,  A01N59/20 ,  A01N2300/00

Abstract: Fungicidal mixtures, comprising as active components 1) a 5-chloro-6-phenyl-7-heterocyclylaminotriazolopyrimidine of the formula I, in which D together with the nitrogen atom forms a pyrrolidine, piperidine or azepine ring, which rings are unsubstituted or substituted by one or two methyl groups or by an ethyl, propyl or butyl group; and L is methyl, fluorine or chlorine; and 2) at least one active compound II selected from the following groups: A) azoles; B) strobilurins; C) acylalanines; D) amine derivatives; E) anilinopyrimidines; F) dicarboximides; G) cinnamides and analogs; H) antibiotics; K) dithiocarbamates; L) heterocyclic compounds according to the description; M) sulfur and copper fungicides; N) nitrophenyl derivatives; O) phenylpyrroles; P) sulfenic acid derivatives; Q) other fungicides according to the description; or R) growth retardants; in a synergistically effective amount, novel triazolopyrimidines, methods for controlling harmful fungi using compounds or mixtures of a compound I with an active compound of groups A) to R) and the use of the compounds I with the active compounds of groups A) to R) for preparing such mixtures, and also compositions comprising these compounds or mixtures.

Abstract translation: 包含作为活性组分的杀真菌混合物1）式I的5-氯-6-苯基-7-杂环基氨基三唑并嘧啶，其中D与氮原子一起形成吡咯烷，哌啶或氮杂环，该环是未取代的或被 一个或两个甲基或乙基，丙基或丁基; L为甲基，氟或氯; 和2）至少一种选自以下组的活性化合物II：A）唑类; B）嗜球果伞素 C）酰基丙氨酸; D）胺衍生物; E）苯胺嘧啶嘧啶; F）二羧酰亚胺; G）肉桂酸酯类似物; H）抗生素; K）二硫代氨基甲酸盐; L）杂环化合物; M）硫和铜杀菌剂; N）硝基苯基衍生物; O）苯基吡咯; P）亚磺酸衍生物; Q）其他杀菌剂根据说明; 或R）生长阻滞剂; 协同有效量的新型三唑并嘧啶，使用化合物或化合物I与A）至R）的活性化合物的混合物来控制有害真菌的方法以及将化合物I与基团A）至R的活性化合物 ），以及包含这些化合物或混合物的组合物。

公开(公告)号：US20080221130A1

公开(公告)日：2008-09-11

申请号：US11996783

申请日：2006-07-20

Applicant: Jochen Dietz ,  Wassilios Grammenos ,  Udo Hunger ,  Jan Klaas Lohmann ,  Jens Renner ,  Joachim Rheinheimer

Inventor： Jochen Dietz ,  Wassilios Grammenos ,  Udo Hunger ,  Jan Klaas Lohmann ,  Jens Renner ,  Joachim Rheinheimer

IPC: A01N43/90 ,  C07D487/04 ,  A01N25/34 ,  A01P3/00

CPC classification number: C07D487/04

Abstract: 5-Methyl-6-phenylpyrazolopyrimidin-7-ylamines of the formula I in which the substituents are defined according to the description, processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

Abstract translation: 其中取代基根据描述定义的式I的5-甲基-6-苯基吡唑并嘧啶-7-基胺，制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080176744A1

公开(公告)日：2008-07-24

申请号：US11885822

申请日：2006-03-08

Applicant: Anja Schwogler ,  Joachim Rheinheimer ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Frank Schieweck

Inventor： Anja Schwogler ,  Joachim Rheinheimer ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Frank Schieweck

IPC: A01N43/54 ,  C07D239/42 ,  A01C1/06

CPC classification number: A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/84 ,  C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D401/04 ,  C07D403/04 ,  C07D405/12

Abstract: The invention relates to the use of 4-aminopyrimidines of formula (I), in which R1═H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkinyl, R2═H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, whereby the hydrocarbon chain in R1 and/or R2 can be substituted as given in the description, R1 and R2 can form, together with the carbon atom to which they are bonded, a 5-7-membered ring which can contain one to three same or different heteroatoms selected from the group O, N or S, R3═H, halogen, cyano, hydroxy, mercapto, azido, alkyl, alkenyl, alkinyl, alkylhalide, —O-D, —S(O)m-D, ON═CRaRb, CRc═NORa, NRcN═CRaRb, NRaRb, NRcNRaRb, NORa, NRcC(═NRc)NRaRb, NRcC(═O)NRaRb, NRaCN, —NRaC(═O)Rc, NRaC(═NORc)Rc′, OC(═O)Ra, C(═NORc)NRaRb, CRc(═NNRaRb), C(═O)NRaRb, C(═O)Ra, CO2Ra, C(═O)NRzRb, C(═O)—N—ORb, C(═S)—NRzRb, C(═O)NRa—NRzRb, C(═N—NRzRc)NRaRb, C(═NORb)Ra, C(═N—NRzRb)Ra, CRaRb—ORz, CRaRb—NRzRc, ON(═CRaRb), NRa(C(═O)Rb), NRa(C(═O)ORb), C(═NRa)NRzRb, C(═0)—NRzRb) NRa(C(═O)—NRzRb), NRa(C(═NRc)Rb), NRa(N═CRcRb), NRa—NRzRb, —NRz—ORa, NRa(C(═NRc)—NRzRb), NRa(C(═NORc)Rb) D=alkyl, alkenyl, alkinyl, alkylhalide, cycloalkyl, five- or six-membered saturated, partly-unsaturated or aromatic mono- or bicyclic heterocycles, containing one to four heteroatoms from the group O, N or S, one of the groups G1 or G2, whereby m, x, Ra, Rb, Rc, Rd, Re, Rz, Y, Z are as defined in the description and the aliphatic, alicyclic or aromatic groups R3, Ra, Rb, Rc, Rd or Re can be substituted as given in the description for the prevention of fungal pests, novel 4-aminopyridines, method for production of said compounds and agents comprising the same.

公开(公告)号：US20080153707A1

公开(公告)日：2008-06-26

申请号：US11883957

申请日：2006-02-15

Applicant: Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl

Inventor： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl

IPC: A01N43/56 ,  C07D231/00 ,  A01N25/26

CPC classification number: C07D231/14 ,  A01N43/56

Abstract: The present invention relates to pyrazolecarboxanilides I in which the variables are as defined below: n is zero or 2; m is 2 or 3; X1 is fluorine or chlorine; X2 is halogen; Y is CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p is zero or 1; R1 is fluorine, chlorine, bromine, C1-C4-alkyl or C1-C4-haloalkyl; R2 is hydrogen or halogen; R3 is hydrogen, methyl or ethyl; W is O or S; with the proviso that, if a) W═O, R1=methyl and R3 is hydrogen, R2 is not fluorine, or b) W═O, n=0, m=2, p=0, R2 and R3 are hydrogen, R1 is not trifluoromethyl or difluoromethyl, to processes for preparing these compounds, to compositions comprising them and to methods for using them for controlling harmful fungi.

Abstract translation: 本发明涉及吡唑烷酰苯胺I，其中变量如下：n为0或2; m为2或3; X 1是氟或氯; X 2是卤素; Y是CN，NO 2，C 1 -C 4 - 烷基，C 1 -C 3 - 4 - 卤代烷基，甲氧基或甲硫基; p为零或1; R 1是氟，氯，溴，C 1 -C 4 - C 1-4烷基或C 1 -C 3 - 低级烷基; R 2是氢或卤素; R 3是氢，甲基或乙基; W为O或S; 条件是，如果a）WO，R 1 =甲基和R 3是氢，R 2不是氟，或b） WO，n = 0，m = 2，p = 0，R 2和R 3是氢，R 1不是三氟甲基或二氟甲基 ，制备这些化合物的方法，包含它们的组合物以及用于控制有害真菌的方法。

公开(公告)号：US20080125445A1

公开(公告)日：2008-05-29

申请号：US11885359

申请日：2006-03-01

Applicant: Peter Schafer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

Inventor： Peter Schafer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

IPC: A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC classification number: C07D487/04

Abstract: 5,6-Dialkyl-7-aminoazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl or alkoxyalkyl, R2 is alkyl, where R1 and/or R2 may be substituted according to the description, A is N or CH, and R3 is CH3 and, if A is CH, additionally hydrogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

Abstract translation: 其中取代基如下定义的式I的5,6-二烷基-7-氨基偶氮嘧啶：R 1是烷基或烷氧基烷基，R 2是烷基，其中R 根据描述，可以取代1和/或R 2，A是N或CH，R 3是CH 3 如果A是CH，另外是氢; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080119493A1

公开(公告)日：2008-05-22

申请号：US10590326

申请日：2005-03-08

Applicant: Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl ,  Udo Hunger

Inventor： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl ,  Udo Hunger

IPC: A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R2 represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R1 and/or R2 being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

Abstract translation: 本发明涉及式（I）的5,6-二烷基-7-氨基 - 三唑并嘧啶，其中取代基定义如下：R 1表示烷基，烷氧基烷基，烯基或炔基; R 2表示根据描述被取代的烷基，烷氧基烷基，烯基或炔基，R 1和/或R 2 2。 本发明还涉及一种生产所述化合物的方法，含有后者的药剂及其用于控制​​植物致病真菌的用途。

公开(公告)号：US20080039319A1

公开(公告)日：2008-02-14

申请号：US11596464

申请日：2005-05-11

Applicant: Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  A01N25/34 ,  A01N59/20

CPC classification number: A01N43/90 ,  A01N59/06 ,  A01N59/02 ,  A01N57/12 ,  A01N47/38 ,  A01N47/34 ,  A01N47/24 ,  A01N47/04 ,  A01N43/50 ,  A01N43/76 ,  A01N43/653 ,  A01N43/36 ,  A01N43/40 ,  A01N43/32 ,  A01N37/48 ,  A01N37/46 ,  A01N37/38 ,  A01N37/34 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R1 is alkyl, halogenalkyl, alkenyl or cyclopentyl, R2 is hydrogen or alkyl, R1 and R2 together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L1 is fluorine or chlorine, L2, L3 are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (1) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.

Abstract translation: 本发明涉及含有活性组分形式的杀真菌混合物1）式（I）的5-甲基-7-氨基 - 三唑并嘧啶，其中R 1是烷基，卤代烷基，烯基或环戊基，R R 2是氢或烷基，R 1和R 2与它们所连接的氮原子一起可以形成可被 甲基，L 1是氟或氯，L 2，L 3，3彼此独立地为氢，氟或氯，以及2）在 至少一种活性物质选自A）唑类，B）嗜球果伞素，C）酰基丙氨酸，D）胺衍生物，E）苯胺基嘧啶; F）二羧酰亚胺; G）肉桂酸酰胺及其类似物，H）抗生素，K）二硫代氨基甲酸盐，L）杂环化合物，M）硫和铜杀真菌剂，N）硝基苯基衍生物，O）苯基吡咯，P）亚磺酸衍生物，Q）其他杀真菌剂和R ）生长阻滞剂，其中所述混合物包含协同有效量的化合物。 新型三唑并嘧啶，使用化合物（1）与A）和R）基团的活性物质的混合物来控制致病真菌的方法，将化合物（I）与A）和R）基团的活性物质一起用于生产 还公开了含有所述混合物的所述混合物和试剂。

公开(公告)号：US20070249633A1

公开(公告)日：2007-10-25

申请号：US11597379

申请日：2005-06-08

Applicant: Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strahmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strahmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to triazolopyrimidines of the formula I in which the index n and the substituents R, R1, R2 and X are as defined below: X is nitro, a group —C(S)NR3R4, a group —C(═N—OR5)(NR6R7) or a group —C(═N—NR8R9)(NR10R11), R is halogen, cyano, hydroxyl, cyanato, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N or S; R1 is alkyl in which one carbon atom may be replaced by a silicon atom, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via a carbon atom and which contains one, two, three or four heteroatoms, independently of one another selected from the group consisting of O, N and S, as ring members; where R1 may be substituted as defined in the description; R2 is alkyl, alkenyl or alkynyl which may be substituted as defined in the description; R3, R4, R5, R6, R7, R8, R9, R10 and R11 are, independently of one another, selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl or alkynyl, where the 4 lastmentioned radicals may be substituted as defined in the description; or R3 and R4, R6 and R7, R8 and R9 and/or R10 and R11 together with the nitrogen atom to which they are attached form a four-, five- or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; and n is 0 or an integer 1, 2, 3 or 4; and the agriculturally acceptable salts thereof, to crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt thereof and at least one liquid or solid carrier and to a method for controlling phytopathogenic harmful fungi.

公开(公告)号：US20080188494A1

公开(公告)日：2008-08-07

申请号：US11912335

申请日：2006-04-24

Applicant: Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler

Inventor： Jochen Dietz ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler

IPC: A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The use of 5-alkyl-6-phenylalkyl-7-aminoazolopyrimidines of the formula I in which the variables are as defined below: Y is alkylene, alkenylene or alkynylene, optionally substituted by alkyl groups; R1 is halogen, cyano, nitro, hydroxyl, mercapto, alkyl, haloalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, haloalkoxy, alkenyloxy, alkynyloxy, alkylthio, NRARB, alkylcarbonyl, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S; RA, RB is hydrogen, alkyl or alkylcarbonyl; n is zero, 1, 2, 3 or 4; R2 is alkyl, alkenyl, cycloalkyl, alkoxyalkyl or alkylthioalkyl; R3 is hydrogen, halogen, cyano, NRARB, hydroxyl, mercapto, alkyl, haloalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, alkyl-S(O)m—; m is 0, 1 or 2; A is N or C—Ra; Ra is hydrogen or alkyl; where the carbon atoms in Y, R1, R2, R3 and Ra may be substituted according to the description; for controlling phytopathogenic harmful fungi; novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, processes for their preparation and compositions comprising them.

Abstract translation: 使用式I的5-烷基-6-苯基烷基-7-氨基偶氮嘧啶，其中变量如下所定义：Y是任选被烷基取代的亚烷基，亚烯基或亚炔基; R 1是卤素，氰基，硝基，羟基，巯基，烷基，卤代烷基，烯基，环烷基，环烯基，烷氧基，卤代烷氧基，烯氧基，炔氧基，烷硫基，NR 或含有一至四个由O，N和S组成的组的杂原子的五元或六元饱和的部分不饱和或芳族杂环; R A，B B是氢，烷基或烷基羰基; n为零，1,2,3或4; R 2是烷基，烯基，环烷基，烷氧基烷基或烷硫基烷基; R 3是氢，卤素，氰基，NR B，B，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基 烷氧基羰基，烷氧羰基，烷氧基羰基，苯氧基，苯硫基，苄氧基，苄硫基，烷基-S（O）m - m为0,1或2; A是N或C-R a a R a是氢或烷基; 其中Y，R 1，R 2，R 3和R a中的碳原子可以根据 描述; 用于控制植物病原性有害真菌; 新的5-烷基-6-苯基烷基-7-氨基 - 偶氮嘧啶，其制备方法和包含它们的组合物。