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公开(公告)号:US20160256445A1
公开(公告)日:2016-09-08
申请号:US15154210
申请日:2016-05-13
Applicant: Bristol-Myers Squibb Company
Inventor: Saleem Ahmad , Lidet A. Negash
IPC: A61K31/4412 , C07D417/04 , C07D409/04 , A61K45/06 , A61K31/444 , C07D409/14 , A61K31/4439 , A61K31/4436 , C07D211/90 , C07D401/04
CPC classification number: C07D211/90 , A61K31/4412 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K45/06 , C07D211/78 , C07D211/86 , C07D401/04 , C07D409/04 , C07D409/14 , C07D417/04
Abstract: The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.
Abstract translation: 本发明提供式(I)化合物或其立体异构体或其药学上可接受的盐,其中所有变量如本文所定义。 这些化合物是可用作药物的单酰基甘油酰基转移酶2型(MGAT2)抑制剂。