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公开(公告)号:US07608604B2
公开(公告)日:2009-10-27
申请号:US12028192
申请日:2008-02-08
申请人: Stuart Nicholas Comlay , Joanne Clare Hannam , William Howson , Christelle Lauret , Yogesh Anil Sabnis
发明人: Stuart Nicholas Comlay , Joanne Clare Hannam , William Howson , Christelle Lauret , Yogesh Anil Sabnis
IPC分类号: A61K31/26 , C07C255/01
CPC分类号: C07C381/00 , A01N41/12
摘要: The present invention relates to compounds of the formula (I) or a tautomer or prodrug thereof, or a pharmaceutically acceptable salt of said compound, tautomer or prodrug, wherein: R1, R2, R3, R4 and R5 are each independently selected from H, halo, CN, CF3 and CONH2; compositions containing such compounds and the uses of such compounds as antiparasitic agents.
摘要翻译: 本发明涉及式(I)化合物或其互变异构体或前药,或所述化合物,互变异构体或前药的药学上可接受的盐,其中:R 1,R 2,R 3,R 4和R 5各自独立地选自H, 卤素,CN,CF 3和CONH 2; 含有这些化合物的组合物以及这些化合物作为抗寄生虫剂的用途。
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公开(公告)号:US07544706B2
公开(公告)日:2009-06-09
申请号:US11945083
申请日:2007-11-26
申请人: Nathan Anthony Logan Chubb , Mark Roger Cox , Jerome Sebastien Dauvergne , Richard Andrew Ewin , Christelle Lauret
发明人: Nathan Anthony Logan Chubb , Mark Roger Cox , Jerome Sebastien Dauvergne , Richard Andrew Ewin , Christelle Lauret
IPC分类号: A61K31/41 , A61K31/415 , A01N43/50 , A01K29/00
CPC分类号: C07D233/56 , C07D233/54 , C07D233/64 , C07D401/12 , C07D403/10 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12 , C07D471/04
摘要: This invention relates to a range of alpha substituted 2-benzyl substituted imidazole compounds and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides.
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13.
公开(公告)号:US20080261940A1
公开(公告)日:2008-10-23
申请号:US10593133
申请日:2005-03-07
IPC分类号: A61K31/415 , C07D231/42 , A61K31/541 , C07D417/04 , A61P33/00
CPC分类号: C07D231/40 , C07D231/42 , C07D231/50 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/04 , C07D417/12
摘要: The invention relates to a sulfonamide compound of formula (I) or a pharmaceutically, veterinarily or agriculturally acceptable salt or solvate thereof, where the groups R1-R5 are described in the description, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides.
摘要翻译: 本发明涉及式(I)的磺酰胺化合物或其药学,兽药或农业上可接受的盐或溶剂化物,其中基团R 1〜5 5描述于 对包含这些化合物的组合物的描述,其合成方法及其作为杀寄生虫剂的用途。
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公开(公告)号:US20100010093A1
公开(公告)日:2010-01-14
申请号:US12559868
申请日:2009-09-15
申请人: Stuart Nicholas Comlay , Joanne Clare Hannam , William Howson , Christelle Lauret , Yogesh Anil Sabnis
发明人: Stuart Nicholas Comlay , Joanne Clare Hannam , William Howson , Christelle Lauret , Yogesh Anil Sabnis
IPC分类号: A61K31/166 , C07C255/58 , A61P33/00
CPC分类号: C07C381/00 , A01N41/12
摘要: The present invention relates to compounds of the formula (I) or a tautomer or prodrug thereof, or a pharmaceutically acceptable salt of said compound, tautomer or prodrug, wherein: R1, R2, R3, R4 and R5 are each independently selected from H, halo, CN, CF3 and CONH2; compositions containing such compounds and the uses of such compounds as antiparasitic agents.
摘要翻译: 本发明涉及式(I)化合物或其互变异构体或前药,或所述化合物,互变异构体或前药的药学上可接受的盐,其中:R 1,R 2,R 3,R 4和R 5各自独立地选自H, 卤素,CN,CF 3和CONH 2; 含有这些化合物的组合物以及这些化合物作为抗寄生虫剂的用途。
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公开(公告)号:US07547718B2
公开(公告)日:2009-06-16
申请号:US11945064
申请日:2007-11-26
申请人: Nathan Anthony Logan Chubb , Mark Roger Cox , Jerome Sebastien Dauvergne , Richard Andrew Ewin , Christelle Lauret
发明人: Nathan Anthony Logan Chubb , Mark Roger Cox , Jerome Sebastien Dauvergne , Richard Andrew Ewin , Christelle Lauret
IPC分类号: A61K31/41 , A61K31/415 , A01N43/50 , A01K29/00
CPC分类号: C07D233/56 , C07D233/54 , C07D233/64 , C07D401/12 , C07D403/10 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12 , C07D471/04
摘要: This invention relates to a range of alpha substituted 2-benzyl substituted imidazole compounds and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides.
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