公开(公告)号：US20060293346A1

公开(公告)日：2006-12-28

申请号：US10573288

申请日：2004-09-30

申请人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N43/42

CPC分类号： A01N43/42 ,  A01N43/90 ,  A01N2300/00

摘要： Fungicidal mixtures comprising, as active components, 1) the triazolopyrimidine derivative of the formula I 2) quinoxyfen of the formula II in a synergistically effective amount, methods for controlling harmful fungi from the class of the Oomycetes using mixtures of the compound I with the compound II, the use of the compound I with the compound II for preparing such mixtures and compositions comprising these mixtures are described.

摘要翻译： 包含作为活性组分的1）式I的三氮代嘧啶衍生物2）协同有效量的式II的喹喔啉的方法，使用化合物I与化合物的混合物来控制来自卵菌纲的有害真菌的方法 II，描述了化合物I与化合物II用于制备这种混合物的使用和包含这些混合物的组合物。

公开(公告)号：US20070149551A1

公开(公告)日：2007-06-28

申请号：US11677862

申请日：2007-02-22

申请人： Andreas GYPSER ,  Thomas Grote ,  Anja Schwogler ,  Joachim Rheiheimer ,  Frank Schieweck ,  Jordi Blasco ,  Ingo Rose ,  Peter Schafer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Eberhard Ammernann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas GYPSER ,  Thomas Grote ,  Anja Schwogler ,  Joachim Rheiheimer ,  Frank Schieweck ,  Jordi Blasco ,  Ingo Rose ,  Peter Schafer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Eberhard Ammernann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A61K31/506 ,  C07D403/02

CPC分类号： C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D403/12

摘要： 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRNaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC (═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC (═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C (═O)NRaRb or —C(═O) Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

公开(公告)号：US20060217400A1

公开(公告)日：2006-09-28

申请号：US10539559

申请日：2003-12-17

申请人： Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of the formula I in which the index n and the substituents R1, R2 and R3 are as defined in the description, and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 其中指数n和取代基R 1，R 2和R 3的式I的三唑并嘧啶如说明书中所定义，以及 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20060079537A1

公开(公告)日：2006-04-13

申请号：US10531898

申请日：2003-11-14

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, —C(═O)-A or S(═O)pA′; A and A′ are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R1 and/or R2 may be substituted as defined in the description; and R3 is cyano, hydroxyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, NR1R2 or S(O)nR31, where n and R31 are as defined in the description; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基，-C（ - O） - 取代的取代基如下： -A或S（-O） A'; A和A'如说明书所定义; p为0,1或2; m为0,1,2,3,4或5; X是氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 - 至十元饱和的，部分不饱和的或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1和R 2连同 它们所连接的氮原子也可以形成可被来自O，N和S的原子间隔的五元或六元环，其中R 1和/或 R 2可以如说明书中定义的取代; 和R 3是氰基，羟基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，NR 1 R 2或S（O）n 其中n和R 31如在说明书中所定义的; 描述了制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060074093A1

公开(公告)日：2006-04-06

申请号：US10532770

申请日：2003-11-14

申请人： Jordi Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/40 ,  A01N43/90

CPC分类号： A01N43/90 ,  A01N43/40 ,  A01N2300/00

摘要： Fungicidal mixtures, comprising A) the triazolopyrimidine of the formula I and B) amide compounds of the formula II where X1 and X2 are halogen, nitro, cyano, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxy, haloalkoxy, haloalkylthio, alkylsulfinyl or alkylsulfonyl; x is 1, 2, 3 or 4; and y is 1, 2, 3, 4 or 5; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II, compositions comprising these compounds and the use of the compounds I and II for preparing such mixtures are described.

摘要翻译： 杀真菌混合物，其包含A）式I的三唑并嘧啶和B）式II的酰胺化合物，其中X 1和X 2是卤素，硝基，氰基，烷基， 烯基，炔基，卤代烷基，卤代烯基，卤代炔基，烷氧基，卤代烷氧基，卤代烷硫基，烷基亚磺酰基或烷基磺酰基; x为1,2,3或4; y为1,2,3,4或5; 在协同有效量下，描述了使用化合物I和II的混合物来控制有害真菌的方法，包含这些化合物的组合物以及化合物I和II用于制备这种混合物的用途。

公开(公告)号：US20060111320A1

公开(公告)日：2006-05-25

申请号：US10532755

申请日：2003-11-14

申请人： Jordi Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/64 ,  A01N55/00 ,  A01N43/90 ,  A01N43/54 ,  A01N43/50

CPC分类号： A01N43/90 ,  A01N55/00 ,  A01N47/38 ,  A01N43/653 ,  A01N2300/00

摘要： Disclosed are fungicidal mixtures containing A) a triazolopyrimidine derivative of formula (1), and B) an azole derivative or the salts or addition compound thereof selected among bromuconazole, difenoconazole, diniconazole, fenbuconazole, fluquinconazole, flusilazole, hexaconazole, prochloraz, tetraconazole, triflumizole, flutriafol, myclobutanil, penconazole, simeconazole, ipconazole, triticonazole, and prothioconazole as active components in a synergistically effective quantity, methods for controlling plant-pathogenic fungi by means of mixtures of compounds I and II-XVIII, substances containing said mixtures, and the use of compounds I and II-XVIII for producing such mixtures.

摘要翻译： 本发明公开了含有A）式（1）的三唑并嘧啶衍生物和B）选自溴唑啉，苯醚甲环唑，二康唑，芬博康唑，氟康唑，氟西唑，己康唑，丙氯灵，四唑唑，三氟唑的盐或其加成化合物的杀真菌混合物 ，氟替卡隆，氟菌唑，康康唑，西康唑，益康唑，利唑康唑和丙硫菌唑作为协同有效量的活性组分，通过化合物I和II-XVIII的混合物控制植物致病真菌的方法，含有所述混合物的物质，以及 使用化合物I和II-XVIII制备这种混合物。

公开(公告)号：US20050107619A1

公开(公告)日：2005-05-19

申请号：US10507605

申请日：2003-03-12

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07B61/00 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34 ,  C07C233/73

CPC分类号： C07C235/34 ,  A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C233/22 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14

摘要： Z-substituted acrylamides of formula (I), where the substituents have the following meanings: X=H, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, with X in the 3- or 4-position, n=1 or 2, where X can be different if n=2, R1=alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, aziridine and oxirane and R2=H, alkyl, haloalkyl, allyl, propargyl or CH2C≡C-alkyl. Methods for production thereof, agents comprising the above and the use thereof for the treatment of plant-pathogenic fungal pests.

摘要翻译： 式（I）的Z-取代的丙烯酰胺，其中取代基具有以下含义：X = H，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，其中X为3-或4-位，n = 1或2，其中 如果n = 2，则X可以不同，R 1 =烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，氮丙啶和环氧乙烷，R 2 = H，烷基，卤代烷基，烯丙基 炔丙基或CH 2C≡C-烷基。 其制备方法，包含上述物质及其用于治疗植物致病性真菌害虫的用途。

公开(公告)号：US20060172891A1

公开(公告)日：2006-08-03

申请号：US10548840

申请日：2004-03-20

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Andreas Gypser ,  Jordi Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Frank Schieweck ,  Michael Rack ,  Ulrich Schofl ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Andreas Gypser ,  Jordi Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Frank Schieweck ,  Michael Rack ,  Ulrich Schofl ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether

IPC分类号： C07D333/22 ,  A01N43/10

CPC分类号： C07D333/38

摘要： The invention relates to novel biphenyl carboxamides of formula (I), wherein A, R, Z, X, Y, m and n have the meanings given in the description, to multiple methods for producing these substances, to their use for combating unwanted micro-organisms and to novel intermediate products and the production thereof.

公开(公告)号：US20060167017A1

公开(公告)日：2006-07-27

申请号：US10539039

申请日：2003-12-16

申请人： Bernd Muller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Bernd Muller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04

摘要： Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R1 is C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, C3-C10-cycloalkyl, C3-C10-cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R2 is C1-C4-alkyl which may be substituted by halogen, cyano, nitro or C1-C2-alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SOm—Rx, NRxRy or NRx—(C═O)—Ry; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 其中指数和取代基如下定义的式I的三唑并嘧啶：R 1是C 1 -C 10 - 烷基， C 1 -C 10亚烷基，C 2 -C 10 - 炔基，C 3 - 亚烷基 C 1 -C 10 - 环烷基，C 3 -C 10 - 环烯基，苯基，萘基或五至十元饱和的， 部分不饱和或芳族杂环，其通过碳连接到三唑并嘧啶并且包含一至四个由N，O和S组成的组的杂原子; R 2是可以被卤素，氰基，硝基或C 1 H 3取代的C 1 -C 4 - 烷基 -C 2 - 烷氧基; n为0或1至4的整数; R如说明书所定义; X是SO x，x，x，x，y，x，y，x， - （CO）-R y; m为0或1〜3的整数; 并描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20050181948A1

公开(公告)日：2005-08-18

申请号：US10509112

申请日：2003-03-27

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： C07D213/56 ,  C07D213/61 ,  C07D263/10 ,  A01N43/60 ,  A01N43/40 ,  A01N43/54

CPC分类号： C07D263/10 ,  C07D213/56 ,  C07D213/61

摘要： The present invention relates to novel phenethylacrylamides of the formula I in which the substituents R1, R2, R3 and R4 have the following meanings: R1 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C3-C8-cycloalkyl, C1-C4-haloalkoxy or C1-C4-haloalkyl; R2 is hydrogen, halogen, C1-C4-alkyl, C1-C4-alkoxy, C3-C10-cycloalkyl, C1-C4-haloalkoxy or C1-C4-haloalkyl; R3 is C1-C4-alkyl, C1-C4-haloalkyl, propargyl, C3-C4-alkenyl or a radical of the formula —H2C—C≡C—C(Ra, Ra)—Rc, wherein Ra, Rb independently of one another are hydrogen or methyl and Rc is hydrogen or C1-C4-alkyl; R4 is methyl or C1-haloalkyl; and Het is a 5- or 6-membered heteroaromatic ring, to processes for their preparation, and to the use of phenethylacrylamides of the formula I for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的新的苯乙基丙烯酰胺，其中取代基R 1，R 2，R 3和R 4 具有以下含义：R 1是氢，卤素，C 1 -C 4 - 烷基，C 1 C 1 -C 4 - 烷氧基，C 3 -C 8 - 环烷基，C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 卤代烷基; R 2是氢，卤素，C 1 -C 4 - 烷基，C 1 -C 3 - 4 - 烷氧基，C 3 -C 10 - 环烷基，C 1 -C 4 - 卤代烷氧基或C 1 -C 4 - 卤代烷基; R 3是C 1 -C 4 - 烷基，C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4 - 烷基，炔丙基，C 3 -C 4 - 烯基或式-H 2C≡CC（R 0）的基团 其中R a，R b，R b独立地为C 1 -C 4，其中R a，R b， 另一个是氢或甲基，R c是氢或C 1 -C 4 - 烷基; R 4是甲基或C 1 - 卤代烷基; 并且Het是5或6元杂芳环，用于其制备方法，以及使用式I的苯乙基丙烯酰胺来控制植物病原性有害真菌。