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    2-(Pyridin-2-yl)-pyrimidines and Their Use for Controlling Harmful Fungi
    1.
    发明申请
    2-(Pyridin-2-yl)-pyrimidines and Their Use for Controlling Harmful Fungi 审中-公开
    2-（吡啶-2-基） - 嘧啶及其用于控制​​有害真菌的用途

    公开(公告)号：US20100286175A1

    公开(公告)日：2010-11-11

    申请号：US12840392

    申请日：2010-07-21

    Applicant: Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

    Inventor： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

    IPC: A01N43/54 ,  C07D401/04 ,  A01P3/00

    CPC classification number: C07D401/04

    Abstract: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

    Abstract translation: 本发明涉及通式（I）的2-（吡啶-2-基） - 嘧啶化合物及其用于控制​​致病真菌的用途，作为作为活性成分的植物保护产品含有这种化合物：通式 （I）中，k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素，OH，CN，NO 2，C 1 -C 4烷基，C 1 -C 4烷基卤，C 1 -C 4烷氧基，C 1 -C 4烷氧基卤化物，C 2 -C 4烯基，C 2 -C 4炔基， C8环烷基，C1-C4烷氧基-C1-C4烷基，氨基，苯氧基，其任选被卤素或C 1 -C 4烷基取代，NHR，NR 2，C（R a）= N-OR b，S（= O）p A1或C （ΟO）A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-，其中Alk表示直链或支链C 1 -C 4亚烷基，和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤，C1-C4烷氧基，C1-C4烷氧基卤化物，羟基，卤素，CN或NO2; 其中当满足以下三个条件中的至少一个时，R2还可以表示氢或C1-C4烷基：n表示3,4或5; k表示1,2或3; 如果m不等于0，则基团R1中的至少一个表示与卤素，C 1 -C 4烷基，C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团， R3表示C1-C4烷基。

    (Hetero)Cyclyl(Thio) Carboxylic Acid Anilides For Controlling Pathogenic Fungi
    6.
    发明申请
    (Hetero)Cyclyl(Thio) Carboxylic Acid Anilides For Controlling Pathogenic Fungi 审中-公开
    （异构）环状（硫代）羧酸酰苯胺用于控制致病真菌

    公开(公告)号：US20070299115A1

    公开(公告)日：2007-12-27

    申请号：US11661679

    申请日：2005-09-05

    Applicant: Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Shwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

    Inventor： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Shwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

    IPC: A01N37/48 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01P3/00 ,  C07C233/00 ,  C07D213/82 ,  C07D231/14 ,  C07D277/56

    CPC classification number: C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07D231/14 ,  C07D277/56

    Abstract: The invention relates to (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I) and to salts of said anilides that can be used for agricultural purposes for controlling pathogenic fungi. In said formula, the variables are defined as follows: A represents a phenyl or at least a monounsaturated 5- or 6-membered heterocycle comprising 1, 2 or 3 heteroatoms, selected from N, O, S, S(═O) and S(═O)2 as ring members, whereby phenyl and the monounsaturated 5- or 6-membered heterocycle can be unsubstituted or can be substituted according to the description; B represents a group of general formula (II), in which the variables R3, R4, R5 and the index m are defined as cited in the claims and the description; Y represents oxygen or sulphur, R1 represents H, OH, alkyl, cycloalkyl, alkoxy, haloalkyl, halocycloalkyl or haloalkoxy; R2 represents halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, haloalkyl, halocycloalkyl, haloalkenyl, haloalkynyl or haloalkoxy; and n represents 0, 1, 2, 3 or 4; and salts that can be used for agricultural purposes. The invention also relates to the use of the (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I), to a method for controlling pathogenic fungi and to a crop protection agent containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound.

    Abstract translation: 本发明涉及通式（I）的（杂）环（硫代）羧酸酰苯胺和可用于农业目的的用于控制致病真菌的所述酰苯胺的盐。 在所述式中，变量定义如下：A表示苯基或至少一个单不饱和的5-或6-元杂环，其包含1,2或3个选自N，O，S，S（-O）和S （-O）2，作为环成员，由此苯基和单不饱和的5-或6-元杂环可以是未取代的或可以根据描述被取代; B表示通式（II）的基团，其中定义了变量R 3，R 4，R 5和指数m， 如权利要求和说明书所引用的; Y表示氧或硫，R 1表示H，OH，烷基，环烷基，烷氧基，卤代烷基，卤代环烷基或卤代烷氧基; R 2表示卤素，硝基，CN，烷基，环烷基，烯基，炔基，烷氧基，卤代烷基，卤代环烷基，卤代烯基，卤代炔基或卤代烷氧基。 并且n表示0,1,2,3或4; 和可用于农业目的的盐。 本发明还涉及通式（I）的（杂）环（硫代）羧酸二酰苯胺用于控制致病真菌的方法和含有至少一种通式（I）的化合物的作物保护剂， 和/或所述化合物的农业上相容的盐。

    Mevalonate kinase as a target for fungicides
    9.
    发明申请
    Mevalonate kinase as a target for fungicides 审中-公开
    甲羟戊酸激酶作为杀真菌剂的靶标

    公开(公告)号：US20060068393A1

    公开(公告)日：2006-03-30

    申请号：US10544657

    申请日：2004-01-28

    Applicant: Thierry Lacour ,  Jan Rether ,  Annette Freund ,  Ralf-Michael Schmidt

    Inventor： Thierry Lacour ,  Jan Rether ,  Annette Freund ,  Ralf-Michael Schmidt

    IPC: C12Q1/68 ,  C07H21/04 ,  C12N9/12 ,  C12N1/18 ,  C12N15/74 ,  A01N37/18 ,  C07K14/00

    CPC classification number: C12N9/1205

    Abstract: The present invention relates to the provision of mevalonate kinase as target for fungicides, to the provision of novel nucleic acid sequences, of functional equivalents of the abovementioned nucleic acid sequences and to the use of the gene products of the abovementioned nucleic acid sequences as novel targets for fungicides. Moreover, the present invention relates to methods for identifying fungicides which inhibit a polypeptide with the biological activity of a mevalonate kinase and to the use of these compounds identified via the abovementioned method as fungicides.

    Abstract translation: 本发明涉及提供甲羟戊酸激酶作为杀真菌剂的靶，提供新的核酸序列，上述核酸序列的功能等同物以及上述核酸序列的基因产物作为新靶标的用途 用于杀菌剂。 此外，本发明涉及用于鉴定抑制具有甲羟戊酸激酶的生物活性的多肽的杀真菌剂的方法以及通过上述方法鉴定的这些化合物作为杀真菌剂的用途的方法。

    2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi
    10.
    发明授权
    2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi 失效
    2-（吡啶-2-基） - 嘧啶及其用于控制​​有害真菌的用途

    公开(公告)号：US07786043B2

    公开(公告)日：2010-08-31

    申请号：US11632342

    申请日：2005-07-22

    Applicant: Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

    Inventor： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

    IPC: C07D239/74 ,  C07D239/70 ,  C07D401/04 ,  C07D403/04 ,  A01N43/54 ,  C07D213/16 ,  C07D213/84 ,  C07D213/53 ,  C07D213/61 ,  C07D213/26

    CPC classification number: C07D401/04

    Abstract: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

    Abstract translation: 本发明涉及通式（I）的2-（吡啶-2-基） - 嘧啶化合物及其用于控制​​致病真菌的用途，作为作为活性成分的植物保护产品含有这种化合物：通式 （I）中，k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素，OH，CN，NO 2，C 1 -C 4烷基，C 1 -C 4烷基卤，C 1 -C 4烷氧基，C 1 -C 4烷氧基卤化物，C 2 -C 4烯基，C 2 -C 4炔基， C8环烷基，C1-C4烷氧基-C1-C4烷基，氨基，苯氧基，其任选被卤素或C 1 -C 4烷基取代，NHR，NR 2，C（R a）= N-OR b，S（= O）p A1或C （ΟO）A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-，其中Alk表示直链或支链C 1 -C 4亚烷基，和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤，C1-C4烷氧基，C1-C4烷氧基卤化物，羟基，卤素，CN或NO2; 其中当满足以下三个条件中的至少一个时，R2还可以表示氢或C1-C4烷基：n表示3,4或5; k表示1,2或3; 如果m不等于0，则基团R1中的至少一个表示与卤素，C 1 -C 4烷基，C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团， R3表示C1-C4烷基。

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