公开(公告)号：US4134974A

公开(公告)日：1979-01-16

申请号：US749031

申请日：1976-12-08

申请人： Piero Melloni ,  Nicola Mongelli ,  Francesco Lauria ,  Alessandro Rossi ,  Raffaele Tommasini

发明人： Piero Melloni ,  Nicola Mongelli ,  Francesco Lauria ,  Alessandro Rossi ,  Raffaele Tommasini

IPC分类号： A61K31/535 ,  A61K31/5383 ,  A61K31/54 ,  A61K31/542 ,  A61P25/24 ,  A61P25/26 ,  C07D207/40 ,  C07D207/404 ,  C07D265/36 ,  C07D498/04 ,  C07D498/14 ,  C07D513/04 ,  C07D513/14

CPC分类号： C07D207/404 ,  C07C205/37 ,  C07C317/00 ,  C07D265/36 ,  C07D513/04

摘要： Cyclic derivatives of 1,4-benzoxazine and 1,4-benzothiazine are disclosd, such as, for instance, 1H,2,3,3a,4-tetrahydro-2-carbamoylmethyl-imidazo[5,1-c][1,4]benzoxazin-1-one and 1H,2,3,3a,4-tetrahydro-2-carbamoylmethyl-8-chloro-imidazo[5,1-c][1,4]benzoxazin-1-one. These compounds are active on the central nervous system, and function as antidepressant agents.

摘要翻译： 公开了1,4-苯并恶嗪和1,4-苯并噻嗪的环状衍生物，例如1H，2,3,3a，4-四氢-2-氨基甲酰基甲基 - 咪唑并[5,1-c] [1,3] 4]苯并恶嗪-1-酮和1H，2,3,3a，4-四氢-2-氨基甲酰基甲基-8-氯 - 咪唑并[5,1-c] [1,4]联苯并恶嗪-1-酮。 这些化合物在中枢神经系统上是活性的，并且作为抗抑郁剂起作用。

公开(公告)号：US4078072A

公开(公告)日：1978-03-07

申请号：US738375

申请日：1976-11-02

申请人： Piero Melloni ,  Arturo Della Torre ,  Francesco Lauria ,  Norina Passerini ,  Alessandro Rossi ,  Raffaele Tommasini

发明人： Piero Melloni ,  Arturo Della Torre ,  Francesco Lauria ,  Norina Passerini ,  Alessandro Rossi ,  Raffaele Tommasini

IPC分类号： C07D205/04 ,  C07D409/04 ,  A61K31/39

CPC分类号： C07D205/04

摘要： Novel N-tricyclic derivatives of azetidine are disclosed of the general formula: ##STR1## WHERE A is a --CH.sub.2 --S-- or --S--CH.sub.2 -- group, the remaining substituents being defined in the specification. Illustrative is the compound 1-[11-(6,11-dihydro-dibenzo [b,e] thiopinyl)]-3-methylamino-azetidine. The compounds are useful for their anti-depressant, anti-convulsant and anxiolytic activities.

摘要翻译： 公开了氮杂环丁烷的新型N-三环衍生物，具有以下通式：其中A是-CH 2 -S-或-S-CH 2 - 基团，其余取代基在说明书中定义。 示例性的是化合物1- [11-（6,11-二氢 - 二苯并[b，e]硫代基）] - 3-甲基氨基 - 氮杂环丁烷。 该化合物可用于其抗抑郁，抗惊厥和抗焦虑活性。

公开(公告)号：US5504298A

公开(公告)日：1996-04-02

申请号：US72581

申请日：1993-06-04

申请人： Alessandro Rossi

发明人： Alessandro Rossi

IPC分类号： B23K11/25 ,  H01R39/32

CPC分类号： B23K11/253 ,  H01R39/32

摘要： Methods and apparatus for identifying the occurrence of fusing electrical attachment during fusing operations are provided. After a conventional fusing operation is complete, an electrical signal is applied to the fusing electrode while the fusing electrode is returned to its home position. The electrical signal is monitored to determine whether a circuit path exists from the fusing electrode through the fused conductors to the ground electrode. The presence of a path would indicate that the fusing electrode has become attached to the fused conductors. An alternate embodiment is also described in which the force required to withdraw the fusing electrode is monitored while the electrode is returned to its home position. If the measured force does not fall within predetermined limits, or if the measured force varies during electrode movement, fusing electrode attachment has occurred.

摘要翻译： 提供了在定影操作期间识别熔接电附件发生的方法和装置。 在传统的定影操作完成之后，在熔断电极返回到其初始位置时，将电信号施加到定影电极。 监测电信号以确定电路路径是否存在从定影电极通过熔融导体到接地电极。 路径的存在将指示定影电极已经附着到熔融导体。 还描述了一个替代实施例，其中在电极返回到其初始位置的同时监测撤回定影电极所需的力。 如果测量的力不在预定限度内，或者如果测量的力在电极运动期间变化，则发生了熔丝电极附着。

公开(公告)号：US5486672A

公开(公告)日：1996-01-23

申请号：US166095

申请日：1993-12-13

申请人： Federico Sbalchiero ,  Alessandro Rossi

发明人： Federico Sbalchiero ,  Alessandro Rossi

IPC分类号： H01R39/32 ,  H02K15/16 ,  B23K11/11

CPC分类号： H01R39/32 ,  H02K15/165

摘要： An improved fusing machine is provided that allows commutators to be balanced during the fusing process. Commutator tangs are compressed onto coil leads to form lead connections. The fusing machine compresses the tangs to varying degrees relative to the shaft. The commutator can be balanced during fusing by compressing tangs to a common radial position or by compressing diametrically opposed tangs to the same extent.

摘要翻译： 提供了一种改进的定影机，其允许换向器在定影过程中平衡。 换向器脚被压缩到线圈引线上以形成引线连接。 定影机相对于轴不同程度地压缩柄脚。 换向器可以在熔断期间通过将柄脚压缩到公共径向位置或通过相同方向压缩直径相对的柄脚来平衡。

公开(公告)号：US5484976A

公开(公告)日：1996-01-16

申请号：US130307

申请日：1993-10-01

申请人： Federico Sbalchiero ,  Sabatino Luciani ,  Alessandro Rossi

发明人： Federico Sbalchiero ,  Sabatino Luciani ,  Alessandro Rossi

IPC分类号： B23K11/25 ,  H01R39/32 ,  H01R43/02 ,  B23K11/24

CPC分类号： B23K11/256 ,  H01R39/32 ,  H01R43/0228

摘要： In the performance of fusing operations which involve the application of force and heat to a workpiece, the heat being generated at least in part by electrical resistance heating resulting from passage of an electrical current through an electrical circuit which includes the workpiece and typically also a fusing electrode, the fusing cycle is controlled at least in part on the basis of measurements of the resistance of the above-mentioned circuit during the fusing operation. If desired, the resistance measurements may be corrected to eliminate or at least substantially reduce the contribution of electrode resistance so that the fusing operation is controlled on the basis of the resistance of the workpiece.

摘要翻译： 在涉及对工件施加力和热量的熔接操作的执行中，至少部分地由于电流通过包括工件的电路导致的电阻加热而产生的热量，并且通常也是熔化 电极，至少部分地基于在定影操作期间上述电路的电阻的测量的基础来控制定影周期。 如果需要，可以校正电阻测量以消除或至少基本上减小电极电阻的贡献，使得基于工件的电阻来控制熔化操作。

公开(公告)号：US5418346A

公开(公告)日：1995-05-23

申请号：US5644

申请日：1993-01-19

申请人： Alessandro Rossi

发明人： Alessandro Rossi

IPC分类号： B23K11/25

CPC分类号： B23K11/252

摘要： Methods and apparatus for monitoring the temperature of a workpiece during fusing operations are provided. The apparatus includes a temperature sensor which monitors the temperature of a commutator bar being fused and outputs an electrical signal corresponding to that temperature. The electric current supplied to the fusing electrode can be interrupted or modified if the temperature of the commutator bar exceeds a predetermined temperature. In this manner, fusing operations can be interrupted if the temperature of the commutator bar approaches a temperature at which other components of the workpiece, such as the core material will be adversely affected. The temperature sensor preferably contacts the workpiece to conduct heat to a sensing element.

摘要翻译： 提供了在定影操作期间监测工件的温度的方法和装置。 该装置包括温度传感器，其监测被融合的换向器条的温度，并输出对应于该温度的电信号。 如果换向器棒的温度超过预定温度，则可以中断或修改提供给定影电极的电流。 以这种方式，如果换向器条的温度接近工件的其他部件（例如芯材料）将受到不利影响的温度，则可以中断定影操作。 温度传感器优选地接触工件以将热传导到感测元件。

公开(公告)号：US5300753A

公开(公告)日：1994-04-05

申请号：US903910

申请日：1992-06-25

申请人： Alessandro Rossi

发明人： Alessandro Rossi

IPC分类号： B23K11/25 ,  B23K11/24

CPC分类号： B23K11/252

摘要： Methods and apparatus for fusing together electrical conductors to a commutator are provided. A precise, timed, and controlled delivery of electric current to the fusing electrode of the fusing machine is achieved. A generic supply signal is converted into a precise and constant input signal through the use of monitoring and feedback techniques, which compare the current status of the physical and electrical phases of the fusing operation to various predetermined fusing profiles to determine the proper application of current to the fusing electrode.

摘要翻译： 提供了将电导体融合到换向器的方法和装置。 实现了对定影机的定影电极的精确，定时和控制的电流传递。 通过使用监控和反馈技术将通用电源信号转换成精确和恒定的输入信号，监视和反馈技术将定影操作的物理和电气相位的当前状态与各种预定的熔断曲线进行比较，以确定电流的适当应用 定影电极。

公开(公告)号：US5202325A

公开(公告)日：1993-04-13

申请号：US499413

申请日：1990-07-12

申请人： Alessandro Rossi ,  Metilde Buonamici ,  Lorenzo Pegrassi ,  Enzo Brambilla

发明人： Alessandro Rossi ,  Metilde Buonamici ,  Lorenzo Pegrassi ,  Enzo Brambilla

IPC分类号： C07D457/02 ,  A61K31/48 ,  A61K31/495 ,  A61P1/08

CPC分类号： A61K31/495 ,  A61K31/48 ,  Y10S514/872

摘要： Compounds of the formula I ##STR1## wherein n is 1 or 2, R.sub.1 represents a hydrogen atom or a C.sub.1 -C.sub.4 alkyl group, R.sub.2 represents a hydrogen atom and R.sub.3 represents a hydrogen atom or a hydroxy group or R.sub.2 and R.sub.3 together represent a chemical bond, R.sub.4 represents a hydrogen atom, or a phenyl or C.sub.1 -C.sub.4 alkyl group, R.sub.5 represents a C.sub.1 -C.sub.4 alkyl group or an alkyl group and R.sub.6 represents a hydrogen or halogen atom, and the pharmaceutically acceptable salt thereof, are useful for the manufacture of a pharmaceutical composition useful in the treatment of emesis.

公开(公告)号：US5063279A

公开(公告)日：1991-11-05

申请号：US436633

申请日：1989-11-15

申请人： Alessandro Rossi

发明人： Alessandro Rossi

IPC分类号： H02K15/02 ,  B23K11/25 ,  H01R39/32

CPC分类号： H02K15/0075 ,  B23K11/255 ,  H01R39/32

摘要： Methods and apparatus for fusing armature wires to a commutator, and fusing stator lead wires and stator hooks, are provided. An electrode assembly having a screw mechanism converts the rotational motion of a motor into a translational motion of the fusing electrode. A microprocessor-based control circuit receives electrode force and displacement data from a load cell and an encoder, respectively, to control the fusing operation. The fusing operation is performed according to a predetermined force or displacement function that is stored in the control circuit.

公开(公告)号：US4847253A

公开(公告)日：1989-07-11

申请号：US273021

申请日：1988-11-18

申请人： Metilde Buonamici ,  Lorenzo Pegrassi ,  Alessandro Rossi ,  Sergio Mantegani

发明人： Metilde Buonamici ,  Lorenzo Pegrassi ,  Alessandro Rossi ,  Sergio Mantegani

IPC分类号： C07D457/02 ,  A61K31/48 ,  A61K31/495 ,  A61P25/00 ,  A61P43/00

CPC分类号： A61K31/48

摘要： Compounds of the formula I ##STR1## wherein R.sub.1 represents a hydrogen atom or a methyl group, either R.sub.2 and R.sub.3 represent hydrogen atoms or together represent a chemical bond, R.sub.4 represents a hydrogen atom or a C.sub.1 -C.sub.4 alkyl group, R.sub.5 represents a C.sub.1 -C.sub.4 alkyl group or an allyl group and R.sub.6 represents a hydrogen or halogen atom, and pharmaceutically acceptable salts thereof, are disclosed as being useful for the treatment of extrapyramidal syndromes such as Parkinson's disease.