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21.发明申请公开(公告)号：US20060276482A1
公开(公告)日：2006-12-07
申请号：US11447459
申请日：2006-06-06
申请人： Roland Gendron , Seok-ki Choi , Paul Fatheree , Adam Goldblum , Daniel Long , Daniel Marquess , S. Turner
发明人： Roland Gendron , Seok-ki Choi , Paul Fatheree , Adam Goldblum , Daniel Long , Daniel Marquess , S. Turner
IPC分类号： A61K31/496 , A61K31/46 , C07D451/04
CPC分类号： C07D451/04 , A61K31/46 , A61K31/496
摘要： The invention provides novel benzoimidazolone-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供了新的苯并咪唑酮 - 甲酰胺5-HT 4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT 4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：US20050197335A1
公开(公告)日：2005-09-08
申请号：US11060195
申请日：2005-02-17
申请人： Daniel Marquess , Seok-Ki Choi , Paul Fatheree , Roland Gendron , Adam Goldblum , Daniel Long , S. Derek Turner , Jyanwei Liu
发明人： Daniel Marquess , Seok-Ki Choi , Paul Fatheree , Roland Gendron , Adam Goldblum , Daniel Long , S. Derek Turner , Jyanwei Liu
IPC分类号： A61K31/46 , A61K31/496 , A61K31/541 , C07D451/04 , G01N33/50
CPC分类号： G01N33/5044 , C07D451/04 , G01N33/5008 , G01N2333/70571
摘要： The invention provides novel indazole-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供了新的吲唑 - 甲酰胺5-HT 4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT 4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：US20070042942A1
公开(公告)日：2007-02-22
申请号：US11589614
申请日：2006-10-30
申请人： Martin Linsell , Paul Fatheree , Michael Leadbetter , Yan Zhu , J. Judice
发明人： Martin Linsell , Paul Fatheree , Michael Leadbetter , Yan Zhu , J. Judice
CPC分类号： B82Y5/00 , A61K9/0014 , A61K9/0019 , A61K38/00 , A61K47/40 , A61K47/6951 , C07K9/008
摘要： Disclosed are glycopeptide derivatives substituted at the C-terminus and/or the R-terminus with a substituent that comprises one or more saccharide groups and a carboxy group; and pharmaceutical compositions containing such glycopeptide derivatives. The disclosed glycopeptide derivatives are useful as antibacterial agents.
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公开(公告)号：US20050159344A1
公开(公告)日：2005-07-21
申请号：US11080130
申请日：2005-03-15
申请人： Martin Linsell , Paul Fatheree , Michael Leadbetter , Yan Zhu , J. Judice
发明人： Martin Linsell , Paul Fatheree , Michael Leadbetter , Yan Zhu , J. Judice
CPC分类号： B82Y5/00 , A61K9/0014 , A61K9/0019 , A61K38/00 , A61K47/40 , A61K47/6951 , C07K9/008
摘要： Disclosed are glycopeptide derivatives substituted at the C-terminus and/or the R-terminus with a substituent that comprises one or more saccharide groups and a carboxy group; and pharmaceutical compositions containing such glycopeptide derivatives. The disclosed glycopeptide derivatives are useful as antibacterial agents.
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公开(公告)号：US07786136B2
公开(公告)日：2010-08-31
申请号：US12008840
申请日：2008-01-15
申请人： Paul Fatheree , Roland Gendron , Adam A Goldblum , Daniel D Long , Daniel Marquess , S. Derek Turner , Seok-Ki Choi
发明人： Paul Fatheree , Roland Gendron , Adam A Goldblum , Daniel D Long , Daniel Marquess , S. Derek Turner , Seok-Ki Choi
IPC分类号： A61K31/46
CPC分类号： C07D451/04
摘要： The invention provides novel indazole-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供了新的吲唑 - 甲酰胺5-HT4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：US07534889B2
公开(公告)日：2009-05-19
申请号：US12136891
申请日：2008-06-11
申请人： Seok-Ki Choi , Paul Fatheree , Adam A Goldblum , Lan Jiang , Daniel D Long , Daniel Marquess , S. Derek Turner
发明人： Seok-Ki Choi , Paul Fatheree , Adam A Goldblum , Lan Jiang , Daniel D Long , Daniel Marquess , S. Derek Turner
IPC分类号： C07D215/00 , A01N43/90
CPC分类号： C07D451/04
摘要： The invention provides novel quinolinone-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供新的喹啉酮 - 甲酰胺5-HT 4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：US07498442B2
公开(公告)日：2009-03-03
申请号：US12075740
申请日：2008-03-13
申请人： Seok-Ki Choi , Paul Fatheree , Roland Gendron , Adam A Goldblum , Lan Jiang , Daniel D Long , Daniel Marquess
发明人： Seok-Ki Choi , Paul Fatheree , Roland Gendron , Adam A Goldblum , Lan Jiang , Daniel D Long , Daniel Marquess
IPC分类号： C07D215/00 , C07D471/02
CPC分类号： C07D451/04
摘要： The invention provides novel quinolinone-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供新的喹啉酮 - 甲酰胺5-HT 4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：US20080255187A1
公开(公告)日：2008-10-16
申请号：US12136891
申请日：2008-06-11
申请人： Seok-Ki Choi , Paul Fatheree , Adam A. Goldblum , Lan Jiang , Daniel D. Long , Daniel Marquess , S. Derek Turner
发明人： Seok-Ki Choi , Paul Fatheree , Adam A. Goldblum , Lan Jiang , Daniel D. Long , Daniel Marquess , S. Derek Turner
IPC分类号： A61K31/439 , A61P1/00
CPC分类号： C07D451/04
摘要： The invention provides novel quinolinone-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供新颖的喹啉酮 - 甲酰胺5-HT 4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT 4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：US20060199839A1
公开(公告)日：2006-09-07
申请号：US11365320
申请日：2006-03-01
申请人： Adam Goldblum , Seok-ki Choi , Paul Fatheree , Roland Gendron , Lan Jiang , Daniel Long , Daniel Marquess , S. Turner
发明人： Adam Goldblum , Seok-ki Choi , Paul Fatheree , Roland Gendron , Lan Jiang , Daniel Long , Daniel Marquess , S. Turner
IPC分类号： A61K31/46 , C07D453/02
CPC分类号： C07D451/04 , C07D453/02
摘要： The invention provides novel quinolinone-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供新颖的喹啉酮 - 甲酰胺5-HT 4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT 4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：US20060100236A1
公开(公告)日：2006-05-11
申请号：US11266881
申请日：2005-11-04
申请人： Seok-Ki Choi , Paul Fatheree , Adam Goldblum , Lan Jiang , Daniel Long , Daniel Marquess , S. Turner
发明人： Seok-Ki Choi , Paul Fatheree , Adam Goldblum , Lan Jiang , Daniel Long , Daniel Marquess , S. Turner
IPC分类号： A61K31/4709
CPC分类号： C07D451/04
摘要： The invention provides novel quinolinone-carboxamide 5-HT4 receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with 5-HT4 receptor activity, and processes and intermediates useful for preparing such compounds.
摘要翻译： 本发明提供新颖的喹啉酮 - 甲酰胺5-HT 4受体激动剂化合物。 本发明还提供包含这些化合物的药物组合物，使用这些化合物治疗与5-HT 4受体活性有关的疾病的方法，以及可用于制备这些化合物的方法和中间体。
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