公开(公告)号：US06222035B1

公开(公告)日：2001-04-24

申请号：US09401984

申请日：1999-09-23

申请人： Hiroshi Tsumuki ,  Junichi Shimada ,  Hironori Imma ,  Akiko Nakamura ,  Hiromi Nonaka ,  Shizuo Shiozaki ,  Shunji Ichikawa ,  Tomoyuki Kanda ,  Yoshihisa Kuwana ,  Michio Ichimura ,  Fumio Suzuki

发明人： Hiroshi Tsumuki ,  Junichi Shimada ,  Hironori Imma ,  Akiko Nakamura ,  Hiromi Nonaka ,  Shizuo Shiozaki ,  Shunji Ichikawa ,  Tomoyuki Kanda ,  Yoshihisa Kuwana ,  Michio Ichimura ,  Fumio Suzuki

IPC分类号： C07D48700

CPC分类号： C07D487/04

摘要： [1,2,4]Triazolo[1,5-c]pyrimidine derivatives represented by formula (I) or pharmaceutically acceptable salts thereof are provided, which have adenosine A2A receptor antagonism and are useful for the treatment or prevention of various diseases induced by hyperactivity of adenosine A2A receptors (for example, Parkinson's disease or senile dementia): wherein R1 represents substituted or unsubstituted aryl, or the like; R2 represents hydrogen, halogen, lower alkyl, substituted or unsubstituted aryl, or the like; R3 represents hydrogen, halogen, XR10 (wherein X represents O or S; and R10 represents substituted or unsubstituted aryl, a substituted or unsubstituted aromatic heterocyclic ring, substituted or unsubstituted aralkyl, lower alkyl, or hydroxy lower alkyl), or the like; and Q represents hydrogen or 3,4-dimethoxybenzyl.

摘要翻译： [1,2,4]具有式（I）表示的三唑并[1,5-c]嘧啶衍生物或其药学上可接受的盐，其具有腺苷A2A受体拮抗作用，可用于治疗或预防由 腺苷A2A受体（例如帕金森病或老年性痴呆）的多动症：其中R1表示取代或未取代的芳基等; R 2表示氢，卤素，低级烷基，取代或未取代的芳基等; R3表示氢，卤素，XR10（其中X表示O或S; R10表示取代或未取代的芳基，取代或未取代的芳族杂环，取代或未取代的芳烷基，低级烷基或羟基低级烷基）等; Q表示氢或3,4-二甲氧基苄基。

公开(公告)号：US06182508B2

公开(公告)日：2001-02-06

申请号：US08992008

申请日：1997-12-17

申请人： Yoshinobu Takeuchi ,  Satoshi Hayashi ,  Takehiro Watarai ,  Shinro Oda ,  Junji Moriwaki ,  Tomoyuki Kanda ,  Katuhide Akimoto

发明人： Yoshinobu Takeuchi ,  Satoshi Hayashi ,  Takehiro Watarai ,  Shinro Oda ,  Junji Moriwaki ,  Tomoyuki Kanda ,  Katuhide Akimoto

IPC分类号： G01P102

CPC分类号： G01C19/5607

摘要： An angular rate sensor is provided which measures the angular rate of a moving object such as an automotive vehicle. The angular rate sensor includes an installation base and an oscillator. The oscillator is excited to oscillate in a preselected direction perpendicular to an axis of rotation of the moving object and provides a signal indicative thereof. The installation base is used for installation of the sensor on the moving object and has an improved orientation structure for orienting the oscillator relative to the installation base during installation of the oscillator on the installation base so that the oscillator may oscillate in the preselected direction. The angular rate sensor is disposed within a casing through improved vibration isolators for absorbing unwanted vibrations impinging upon an operation of the sensor.

摘要翻译： 提供了一种角速率传感器，其测量诸如机动车辆的移动物体的角速率。 角速率传感器包括安装基座和振荡器。 激励振荡器以垂直于移动物体的旋转轴的预选方向振荡并提供指示其的信号。 安装基座用于将传感器安装在移动物体上，并且在将振荡器安装在安装基座上时具有改进的定向结构，用于将振荡器相对于安装基座定向，使得振荡器可以在预选的方向上振荡。 角速率传感器通过改进的隔振器设置在壳体内，用于吸收冲击传感器操作的不想要的振动。

公开(公告)号：US6163390A

公开(公告)日：2000-12-19

申请号：US516562

申请日：2000-02-29

申请人： Tomoyuki Kanda ,  Kazutoshi Koie ,  Katsuyoshi Nishii ,  Masahiro Shiozawa ,  Katsumi Kamiya ,  Atsuo Ishizuka ,  Kenichiro Takada

发明人： Tomoyuki Kanda ,  Kazutoshi Koie ,  Katsuyoshi Nishii ,  Masahiro Shiozawa ,  Katsumi Kamiya ,  Atsuo Ishizuka ,  Kenichiro Takada

IPC分类号： G02B5/32 ,  G03H1/04 ,  G03H1/22 ,  G03H1/28 ,  H04N7/14 ,  G03H1/02

CPC分类号： G02B5/32 ,  G03H1/0256 ,  G03H1/04 ,  G03H1/0404 ,  G03H1/0486 ,  G03H1/22 ,  G03H1/265 ,  G03H1/28 ,  G03H2001/2239 ,  G03H2001/306 ,  G03H2223/14 ,  G03H2240/51 ,  G03H2240/53 ,  G03H2250/32 ,  G03H2260/10 ,  H04N7/144

摘要： A method for producing a hologram recording an interference fringe formed by an object light and a reference light on a photosensitive dry plate, and the object light either having diffusing and scattering characteristics or being passed through an optical diffusion body, mainly includes the following steps: In a first step, a ratio .eta..sub.R0 /.eta..sub.00 of a first diffraction efficiency .eta..sub.00 and a second diffraction efficiency .eta..sub.R0, is calculated. The diffraction efficiency .eta..sub.00 is dependent on two object light beams. The efficiency .eta..sub.R0 is dependent on the object light and the reference light. In a second step, the intensity E.sub.O of the object light and the intensity E.sub.R of the reference light is adjusted in such a way that the ratio .eta..sub.R0 /.eta..sub.00 is set to at least 10 and the efficiency .eta..sub.00 does not exceed 5%.A display device using the above hologram is structured by a display unit for generating a signal light; a hologram screen formed by either reflection or transmission hologram, and a projecting unit for projecting the signal light to the hologram screen.According to the present invention, it is possible to easily produce a hologram, for example, a screen hologram, having no cloudiness or cloudy state when an observer observes an image displayed on the screen, and to a display device using the above hologram screen.

摘要翻译： 一种用于产生记录由感光干板上的物体光和参考光形成的干涉条纹的全息图的方法以及具有漫射和散射特性或通过光漫射体的目标光主要包括以下步骤： 在第一步骤中，计算第一衍射效率eta 00和第二衍射效率eta R0的比率ηR0 / eta 00。 衍射效率eta 00取决于两个物体光束。 效率ηR取决于物体光和参考光。 在第二步骤中，对象光的强度EO和基准光的强度ER进行调整，使得eta R0 / eta00的比率设定为至少10，效率eta 00不超过5％ 。 使用上述全息图的显示装置由用于产生信号光的显示单元构成; 通过反射或透射全息图形成的全息屏幕和用于将信号光投影到全息屏幕的投影单元。 根据本发明，当观察者观察屏幕上显示的图像以及使用上述全息图的显示装置时，可以容易地制造全息图，例如不具有混浊状态的屏幕全息图。

公开(公告)号：US20110183992A1

公开(公告)日：2011-07-28

申请号：US13055005

申请日：2009-07-23

申请人： Junichi Ikeda ,  Shunji Ichikawa ,  Masako Kurokawa ,  Tomoyuki Kanda

发明人： Junichi Ikeda ,  Shunji Ichikawa ,  Masako Kurokawa ,  Tomoyuki Kanda

IPC分类号： A61K31/519 ,  C07D487/04 ,  C07D417/14 ,  C07D487/14 ,  C07D495/04 ,  C07D473/32 ,  C07D417/04 ,  A61K31/4439 ,  A61K31/506 ,  A61K31/52 ,  A61K31/427 ,  A61P25/06

CPC分类号： A61K31/427 ,  A61K31/519 ,  A61K31/52 ,  A61K45/06 ,  A61K2300/00

摘要： Provided are therapeutic and/or preventive agents for migraine which comprise, as an active ingredient, a compound having a selective adenosine A2A receptor antagonistic activity or a pharmaceutically acceptable salt thereof; therapeutic and/or preventive agents for migraine which comprise, as an active ingredient, a compound having a selective adenosine A2A receptor antagonistic activity, which has an affinity for the adenosine A2A receptor 10 times or higher than that for the adenosine A1 receptor, or a pharmaceutically acceptable salt thereof; and the like.

摘要翻译： 本发明提供了作为活性成分的具有选择性腺苷A2A受体拮抗活性的化合物或其药学上可接受的盐的偏头痛治疗和/或预防剂， 或作为活性成分的具有选择性腺苷A2A受体拮抗作用的化合物，其对腺苷A2A受体的亲和力比腺苷A1受体高10倍以上，或 其药学上可接受的盐; 等等。

公开(公告)号：US20060058320A1

公开(公告)日：2006-03-16

申请号：US10528452

申请日：2003-09-24

申请人： Kyoichiro Iida ,  Takamasa Sugita ,  Shizuo Shiozaki ,  Tomoyuki Kanda ,  Yoshihisa Kuwana ,  Junichi Shimada

发明人： Kyoichiro Iida ,  Takamasa Sugita ,  Shizuo Shiozaki ,  Tomoyuki Kanda ,  Yoshihisa Kuwana ,  Junichi Shimada

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04

摘要： The present invention provides [1,2,4]triazolo[1,5-c]pyrimidine derivatives or pharmaceutically acceptable salts thereof which have adenosine A2A receptor antagonism and are useful for treating and/or preventing a disease induced by hyperactivity of an adenosine A2A receptor, the derivatives being represented by formula (I): (wherein R1 represents substituted or unsubstituted aryl or a substituted or unsubstituted aromatic heterocyclic group; R2 represents a hydrogen atom, halogen, lower alkyl, lower alkanoyl, aroyl, substituted or unsubstituted aryl, or a substituted or unsubstituted aromatic heterocyclic group; R3 represents lower alkyl, lower cycloalkyl, substituted or unsubstituted lower alkanoyl, substituted or unsubstituted aryl, or a substituted or unsubstituted aromatic heterocyclic group; and Q represents a hydrogen atom or 3,4-dimethoxybenzyl).

摘要翻译： 本发明提供具有腺苷A 2A 2受体拮抗作用的[1,2,4]三唑并[1,5-c]嘧啶衍生物或其药学上可接受的盐，可用于治疗和/或预防 由腺苷A 2A受体的多动症引起的疾病，该衍生物由式（I

公开(公告)号：US06542265B2

公开(公告)日：2003-04-01

申请号：US10079371

申请日：2002-02-20

申请人： Tomoyuki Kanda ,  Kenichiro Takada

发明人： Tomoyuki Kanda ,  Kenichiro Takada

IPC分类号： G02B532

CPC分类号： G02B5/32 ,  G03H1/0256 ,  G03H1/04 ,  G03H1/0404 ,  G03H1/0486 ,  G03H1/22 ,  G03H1/265 ,  G03H1/28 ,  G03H2001/2239 ,  G03H2001/306 ,  G03H2223/14 ,  G03H2240/51 ,  G03H2240/53 ,  G03H2250/32 ,  G03H2260/10 ,  H04N7/144

摘要： A method for producing a hologram recording an interference fringe formed by an object light and a reference light on a photosensitive dry plate, and the object light either having diffusing and scattering characteristics or being passed through an optical diffusion body, mainly includes the following steps: In a first step, a ratio &eegr;R0/&eegr;00 of a first diffraction efficiency &eegr;00 and a second diffraction efficiency &eegr;R0, is calculated. The diffraction efficiency &eegr;00 is dependent on two object light beams. The efficiency &eegr;R0 is dependent on the object light and the reference light. In a second step, the intensity E0 of the object light and the intensity ER of the reference light is adjusted in such a way that the ratio &eegr;R0/&eegr;00 is set to at least 10 and the efficiency &eegr;00 does not exceed 5%. A display device using the above hologram is structured by a display unit for generating a signal light; a hologram screen formed by either reflection or transmission hologram, and a projecting unit for projecting the signal light to the hologram screen. According to the present invention, it is possible to easily produce a hologram, for example, a screen hologram, having no cloudiness or cloudy state when an server observes an image displayed on the screen, and a display device using the above hologram screen.

摘要翻译： 一种用于产生记录由感光干板上的物体光和参考光形成的干涉条纹的全息图的方法以及具有漫射和散射特性或通过光漫射体的目标光主要包括以下步骤： 在第一步骤中，计算第一衍射效率eta00和第二衍射效率etaR0的等于etaR0 / eta00。 衍射效率eta00取决于两个物体光束。 效率etaR0取决于物体光和参考光。 在第二步骤中，调节对象光的强度E0和参考光的强度ER，使得etaR0 / eta00的比率设置为至少10，效率eta00不超过5％.A显示 使用上述全息图的装置由用于产生信号光的显示单元构成; 通过反射或透射全息图形成的全息屏幕和用于将信号光投射到全息屏幕的投影单元。根据本发明，可以容易地生成全息图，例如没有浑浊的全息图 或服务器观察屏幕上显示的图像时的混浊状态，以及使用上述全息图的显示装置。

公开(公告)号：US06392767B1

公开(公告)日：2002-05-21

申请号：US09749900

申请日：2000-12-29

申请人： Tomoyuki Kanda ,  Kenichiro Takada

发明人： Tomoyuki Kanda ,  Kenichiro Takada

IPC分类号： G02B532

摘要： A method for producing a hologram recording an interference fringe formed by an object light and a reference light on a photosensitive dry plate, and the object light either having diffusing and scattering characteristics or being passed through an optical diffusion body, mainly includes the following steps: In a first step, a ratio &eegr;RO/&eegr;OO of a first diffraction efficiency &eegr;OO and a second diffraction efficiency &eegr;RO, is calculated. The diffraction efficiency &eegr;OO is dependent on two object light beams. The efficiency &eegr;RO is dependent on the object light and the reference light. In a second step, the intensity EO of the object light and the intensity ER of the reference light is adjusted in such a way that the ratio &eegr;RO/&eegr;OO is set to at least 10 and the efficiency &eegr;OO does not exceed 5%. A display device using the above hologram is structured by a display unit for generating a signal light; a hologram screen formed by either reflection or transmission hologram, and a projecting unit for projecting the signal light to the hologram screen. According to the present invention, it is possible to easily produce a hologram, for example, a screen hologram, having no cloudiness or cloudy state when an observer observes an image displayed on the screen, and to a display device using the above hologram screen.

公开(公告)号：US06388021B1

公开(公告)日：2002-05-14

申请号：US09291192

申请日：1999-04-14

申请人： Yasuhiro Shibata ,  Tomoyuki Kanda ,  Atsuhiko Tounaka ,  Susumu Maekawa ,  Kiyotada Yasuhara

发明人： Yasuhiro Shibata ,  Tomoyuki Kanda ,  Atsuhiko Tounaka ,  Susumu Maekawa ,  Kiyotada Yasuhara

IPC分类号： C08F1600

CPC分类号： C23C22/34 ,  C09D133/066 ,  C23C22/08 ,  Y10T428/256 ,  Y10T428/31692 ,  Y10T428/31699 ,  C08L2666/54

摘要： A metal surface treatment composition is provided which improves corrosion resistance and film adhesion, and confers slip properties. This composition is an acrylic resin-containing metal surface treatment composition which is water-soluble, water-dispersible or emulsifiable, which comprises an acrylic resin, this resin comprising either or both of an amino group and an ammonium group together with a hydroxyl group and a hydrophobic group, and which further comprises a heavy metal or one of its salts.

摘要翻译： 提供一种金属表面处理组合物，其提高耐腐蚀性和膜粘合性，并赋予滑动性能。 该组合物是包含丙烯酸树脂的水溶性，水分散性或乳化性的含丙烯酸树脂的金属表面处理组合物，该树脂包含氨基和铵基团中的一个或两个以及羟基和羟基， 疏水基团，并且还包含重金属或其盐之一。

公开(公告)号：US06244385B1

公开(公告)日：2001-06-12

申请号：US09368350

申请日：1999-08-05

申请人： Yoshimichi Tsubata ,  Katsuyuki Narai ,  Eiji Suzuki ,  Daihei Teshima ,  Atsushi Fujikawa ,  Keiichi Hanyu ,  Masaaki Yamaguchi ,  Tomoyuki Kanda ,  Eiji Ohyama ,  Akinori Tanno

发明人： Yoshimichi Tsubata ,  Katsuyuki Narai ,  Eiji Suzuki ,  Daihei Teshima ,  Atsushi Fujikawa ,  Keiichi Hanyu ,  Masaaki Yamaguchi ,  Tomoyuki Kanda ,  Eiji Ohyama ,  Akinori Tanno

IPC分类号： F01M118

CPC分类号： F16H57/0412 ,  F16H57/0434 ,  F16H57/0489 ,  F16H59/72 ,  F16H61/0025 ,  F16H61/12 ,  F16H61/662 ,  F16H2061/0037

摘要： A lubrication pressure controller comprises a lubrication pressure regulating valve 41, which is provided in a lubrication oil passage 36 directing hydraulic oil to lubricated parts, and a cooler pressure regulating valve 42, which is provided in a discharge oil passage 51b of the lubrication pressure regulating valve 41. The lubrication pressure regulating valve 41 adjusts the pressure in the lubrication oil passage 36, and the cooler pressure regulating valve 42 adjusts the pressure supplied to an oil cooler 55. The hydraulic oil discharged from the cooler pressure regulating valve 42 is returned through a recirculation line 52 to a suction oil passage 31 of a pump. In this construction, an adequate supply of lubrication oil is maintained even if one of the valves experiences locking of a valve spool on an open side. Moreover, by providing signal pressure generating means 60, which applies a signal pressure to these two valves in correspondence with a driving condition, the lubrication pressure controller can be set to acquire a desired balance in the lubrication, cooling and recirculation for the hydraulic oil in response to a driving condition.

摘要翻译： 润滑压力控制器包括：润滑压力调节阀41，其设置在将液压油引导到润滑部件的润滑油通道36中;以及冷却器压力调节阀42，其设置在润滑压力调节用的排出油路51b中 润滑压力调节阀41调节润滑油通道36中的压力，而冷却器压力调节阀42调节供给到油冷却器55的压力。从冷却器压力调节阀42排出的液压油通过 再循环管线52连接到泵的抽吸油通道31。 在这种结构中，即使其中一个阀在开放侧经历阀芯的锁定，也能保持足够的润滑油供应。 此外，通过提供信号压力发生装置60，其对应于驱动条件向这两个阀施加信号压力，可以设置润滑压力控制器以获得润滑，冷却和再循环中所需的平衡，用于液压油的润滑，冷却和再循环 回应驾驶状况。

公开(公告)号：US06198555B1

公开(公告)日：2001-03-06

申请号：US08823484

申请日：1997-03-25

申请人： Kazumasa Kurokawa ,  Tomoyuki Kanda ,  Atsuo Ishizuka ,  Masahiro Shiozawa

发明人： Kazumasa Kurokawa ,  Tomoyuki Kanda ,  Atsuo Ishizuka ,  Masahiro Shiozawa

IPC分类号： G03H108

CPC分类号： G02B5/32 ,  G02B5/1876 ,  G03H1/04 ,  G03H2001/0417 ,  G03H2001/0439 ,  G03H2222/36

摘要： A coherent beam is converted into a light flux having an expanded width at a predetermined position closer to a photosensitive element. Part of the expanded light flux is irradiated directly on the photosensitive element as a reference beam. The remainder of the expanded light flux is diffused, and its optical direction is changed. Thus, the remainder of the expanded light flux not irradiated directly to the photosensitive element is converted into a scattered beam advancing as an object beam toward the photosensitive element. Interference fringes are formed on the photosensitive element by using the reference beam and the object beam.

摘要翻译： 相干光束被转换成在更靠近感光元件的预定位置具有扩展宽度的光束。 扩展的光束的一部分直接作为参考光束照射在感光元件上。 扩展的光束的其余部分被扩散，并且其光学方向改变。 因此，不直接照射到感光元件的扩展光束的其余部分被转换成朝向感光元件作为物体光束前进的散射光束。 通过使用参考光束和物体光束在感光元件上形成干涉条纹。