Insecticidal compounds
    31.
    发明授权
    Insecticidal compounds 有权
    杀虫化合物

    公开(公告)号:US08410145B2

    公开(公告)日:2013-04-02

    申请号:US12808847

    申请日:2008-12-18

    IPC分类号: A61K31/44 C07D261/02

    摘要: A compound of formula (I): wherein A1, A2, A3, A4, G1, R1, R2, R3 and R4 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of Formula (I), to insecticidal, acaricidal, molluscicidal or nematicidal compositions comprising them and to methods of using them to combat and control insect, acarine, mollusc or nematode pests.

    摘要翻译: 式(I)的化合物:其中A1,A2,A3,A4,G1,R1,R2,R3和R4如权利要求1所定义; 或其盐或N-氧化物。 此外,本发明涉及制备式(I)化合物,包含它们的杀虫,杀螨,杀软体动物或杀线虫组合物的方法和中间体以及使用它们来对抗和控制昆虫,螨虫,软体动物或线虫害虫的方法。

    CHEMICAL COMPOUNDS
    35.
    发明申请
    CHEMICAL COMPOUNDS 失效
    化学化合物

    公开(公告)号:US20100305351A1

    公开(公告)日:2010-12-02

    申请号:US12841586

    申请日:2010-07-22

    IPC分类号: C07F7/10

    CPC分类号: C07F7/0812 A01N55/00

    摘要: A fungicidal compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by groups R7, R8 and R9; R1 is hydrogen, optionally substituted (C1-4alkyl, optionally substituted (C1-4alkylC(═O), optionally substituted (C1-4alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; R2, R3, R4 and R5 are each, independently, hydrogen, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4alkyl; R6 is an organic group containing three to thirteen carbon atoms and at least one silicon atom and, optionally, one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, and is optionally substituted by one to four independently selected halogen atoms; R7, R8 and R9 are each, independently, hydrogen, halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3alkoxy(C1-3)alkyl or cyano, where at least one of R7, R8 and R9 is not hydrogen; and X is O or S; or an N-oxide thereof; and when present, each optional substituent on alkyl moieties, allyl, propargyl and allenyl is, independently, selected from halogen, hydroxy, cyano, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, methylsulfonyl, ethylsulfonyl, difluoromethoxy, trifluoromethoxy and trifluorothiomethoxy.

    摘要翻译: 式(I)的杀真菌化合物:其中Het是含有一至三个杂原子的5-或6-元杂环,各自独立地选自氧,氮和硫,该环被R7,R8和R9基团取代; 任选取代的(C 1-4烷基,(C 1-4)C(= O),任选取代的(C 1-4烷基C(= O)O),任选取代的(C 1-4)烷氧基(C 1-4) 取代的烯丙基,任选取代的炔丙基或任选取代的烯丙基; R 2,R 3,R 4和R 5各自独立地为氢,卤素,任选取代的(C 1-4)烷基,任选取代的(C 1-4)烷氧基或任选取代的 4)烷氧基(C 1-4烷基; R 6是含有三至十三个碳原子和至少一个硅原子的有机基团,以及任选的一至三个杂原子,各自独立地选自氧,氮和硫,并且任选地被一个 至四个独立选择的卤素原子; R 7,R 8和R 9各自独立地为氢,卤素,C 1-3烷基,C 1-3卤代烷基,C 1-3烷氧基(C 1-3)烷基或氰基,其中R 7, R8和R9不是氢; X是O或S;或其N-氧化物;当存在时,每个任选的取代基 羟基,氰基,甲氧基羰基,乙氧基羰基,甲氧基,乙氧基,甲基磺酰基,乙基磺酰基,二氟甲氧基,三氟甲氧基和三氟硫代甲氧基,独立地选自烷基部分,烯丙基,炔丙基和烯丙基。

    Siliconated phenyl amides derivatives useful as microbiocide
    36.
    发明授权
    Siliconated phenyl amides derivatives useful as microbiocide 失效
    用作杀微生物剂的硅烷基苯基酰胺衍生物

    公开(公告)号:US07767623B2

    公开(公告)日:2010-08-03

    申请号:US10509607

    申请日:2003-03-21

    CPC分类号: C07F7/0812 A01N55/00

    摘要: A fungicidal compound of formula (1): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by groups R7, R8 and R9; R1 is hydrogen, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; R2, R3, R4and R5 are each, independently, hydrogen, halogen, optionally substituted (C1-4)alkoxy(C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R6 is an organic group containing three to thirteen carbon atoms and at least one silicon atom and, optionally, one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, and is optionally substituted by one to four independently selected halogen atoms; R7, R8 and R9are each, independently, hydrogen, halogen, C1-3alkyl, C1-3haloalkyl, C1-3alkoxy(C1-3)alkyl or cyano, where at least one of R7, R8and R9 is not hydrogen; and X is O or S; or an N-oxide thereof; and when present, each optional substituent on alkyl moieties, allyl, propargyl and allenyl is, independently, selected from halogen, hydroxy, cyano, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, methylsulfonyl, ethylsulfonyl, diflouromethoxy, trifluoromethoxy and trifluorothiomethoxy.

    摘要翻译: 式(1)的杀真菌化合物:其中Het是含有一至三个杂原子的5-或6-元杂环,各自独立地选自氧,氮和硫,该环被R7,R8和R9基团取代; 任选取代的(C 1-4)烷基C(= O)O,任选取代的(C 1-4)烷氧基(C 1-4)烷基,任选取代的烯丙基, 任选取代的炔丙基或任选取代的烯丙基; R 2,R 3,R 4和R 5各自独立地为氢,卤素,任选取代的(C 1-4)烷氧基(C 1-4)烷氧基或任选取代的(C 1-4)烷氧基(C 1-4)烷基; R6是含有3至13个碳原子和至少一个硅原子和任选的1至3个各自独立地选自氧,氮和硫的杂原子的有机基团,并且任选被一至四个独立选择的卤素原子取代; R 7,R 8和R 9各自独立地为氢,卤素,C 1-3烷基,C 1-3卤代烷基,C 1-3烷氧基(C 1-3)烷基或氰基,其中R 7,R 8和R 9中的至少一个不是氢; X为O或S; 或其N-氧化物; 当存在时,烷基部分上的每个任选的取代基,烯丙基,炔丙基和烯丙基独立地选自卤素,羟基,氰基,甲氧基羰基,乙氧基羰基,甲氧基,乙氧基,甲基磺酰基,乙基磺酰基,二氟甲氧基,三氟甲氧基和三氟硫代甲氧基。