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公开(公告)号:US20170247361A1
公开(公告)日:2017-08-31
申请号:US15596766
申请日:2017-05-16
IPC分类号: C07D413/12 , A01N43/80 , C07D331/04
CPC分类号: C07D413/12 , A01N43/36 , A01N43/80 , C07D331/04 , C07D409/12
摘要: The present invention relates to processes for the preparation of thietane derivatives of the formula IA and thietane derivatives of the formula IB wherein R1, R2, A1, A2, A3, A4, B, and n are as defined in the claims. The invention also relates to intermediates useful in the processes, as well as the compounds of formula IA and IB and their use as pesticides.
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公开(公告)号:US09247740B2
公开(公告)日:2016-02-02
申请号:US14240428
申请日:2012-08-24
IPC分类号: C07D413/12 , C07D331/04 , A01N43/20 , A01N43/80 , A01N43/40 , A01N43/54
CPC分类号: A01N43/20 , A01N43/40 , A01N43/54 , A01N43/80 , C07D331/04 , C07D413/12
摘要: The present invention provides compounds of formula (I), wherein G1 is oxygen; R1 is hydrogen; R2 is group P (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y1 is C—R6, CH or nitrogen; Y2 and Y3 are independently CH or nitrogen; wherein no more than two of Y1, Y2 and Y3 are nitrogen and wherein Y2 and Y3 are not both nitrogen; R5 is hydrogen, halogen, cyano, nitro, NH2, C1-C2alkyl, C1-C2haloalkyl, C3-C5cycloalkyl, C3-C5halocycloalkyl, C1-C2alkoxy, C1-C2haloalkoxy; R6 together with R5 forms a —CH═CH—CH═CH— bridge; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).
摘要翻译: 本发明提供式(I)化合物,其中G1是氧; R1是氢; R2是基团P(P)L是键,亚甲基或亚乙基; A1和A2之一是S,SO或SO2,另一个是-C(R4)R4-R3是氢或甲基; 每个R 4独立地是氢或甲基; Y1是C-R6,CH或氮; Y2和Y3独立地是CH或氮; 其中Y1,Y2和Y3中不超过两个是氮,并且其中Y 2和Y 3不都是氮; R5是氢,卤素,氰基,硝基,NH2,C1-C2烷基,C1-C2卤代烷基,C3-C5环烷基,C3-C5卤代环烷基,C1-C2烷氧基,C1-C2卤代烷氧基; R6与R5一起形成-CH = CH-CH = CH-桥; X2是C-X6或氮; X1,X3和X6独立地为氢,卤素或三卤代甲基,其中X 1,X 3和X 6中的至少两个不是氢; X4是三氟甲基,二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式(I)化合物的中间体,以及使用式(I)化合物控制昆虫,螨虫,线虫或软体动物的方法。
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公开(公告)号:US08895587B2
公开(公告)日:2014-11-25
申请号:US14118037
申请日:2012-05-15
IPC分类号: C07D307/28 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/78 , A01N43/80 , C07D207/20 , C07D261/04 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/04 , C07D413/12 , C07D417/12 , A01N43/08
CPC分类号: C07D307/28 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/78 , A01N43/80 , C07D207/20 , C07D261/04 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/04 , C07D413/12 , C07D417/12
摘要: The present invention provides compounds of formula (I) wherein R1, R2, R3, R4, G1, n, A1, A2, A3, A4, Y1, Y2, and Y3 are as defined in the claims. The invention also relates to processes and intermediates for preparing these compounds, to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising these compounds and to methods of using these compounds to control insect, acarine, nematode and mollusc pests.
摘要翻译: 本发明提供式(I)化合物,其中R1,R2,R3,R4,G1,n,A1,A2,A3,A4,Y1,Y2和Y3如权利要求中所定义。 本发明还涉及制备这些化合物的方法和中间体,包含这些化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物,以及使用这些化合物来控制昆虫,螨虫,线虫和软体动物害虫的方法。
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公开(公告)号:US20140206606A1
公开(公告)日:2014-07-24
申请号:US14240428
申请日:2012-08-24
CPC分类号: A01N43/20 , A01N43/40 , A01N43/54 , A01N43/80 , C07D331/04 , C07D413/12
摘要: The present invention provides compounds of formula (I), wherein G1 is oxygen; R1 is hydrogen; R2 is group P (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y1 is C—R6, CH or nitrogen; Y2 and Y3 are independently CH or nitrogen; wherein no more than two of Y1, Y2 and Y3 are nitrogen and wherein Y2 and Y3 are not both nitrogen; R5 is hydrogen, halogen, cyano, nitro, NH2, C1-C2alkyl, C1-C2haloalkyl, C3-C5cycloalkyl, C3-C5halocycloalkyl, C1-C2alkoxy, C1-C2haloalkoxy; R6 together with R5 forms a —CH═CH—CH═CH— bridge; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).
摘要翻译: 本发明提供式(I)化合物,其中G1是氧; R1是氢; R2是基团P(P)L是键,亚甲基或亚乙基; A1和A2之一是S,SO或SO2,另一个是-C(R4)R4-R3是氢或甲基; 每个R 4独立地是氢或甲基; Y1是C-R6,CH或氮; Y2和Y3独立地是CH或氮; 其中Y1,Y2和Y3中不超过两个是氮,并且其中Y 2和Y 3不都是氮; R5是氢,卤素,氰基,硝基,NH2,C1-C2烷基,C1-C2卤代烷基,C3-C5环烷基,C3-C5卤代环烷基,C1-C2烷氧基,C1-C2卤代烷氧基; R6与R5一起形成-CH = CH-CH = CH-桥; X2是C-X6或氮; X1,X3和X6独立地为氢,卤素或三卤代甲基,其中X 1,X 3和X 6中的至少两个不是氢; X4是三氟甲基,二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式(I)化合物的中间体,以及使用式(I)化合物控制昆虫,螨虫,线虫或软体动物的方法。
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公开(公告)号:US20130165485A1
公开(公告)日:2013-06-27
申请号:US13771829
申请日:2013-02-20
申请人: Jerome Yves Cassayre , Peter Renold , Vladimir Bobosik , Myriem El Qacemi , Anne Jacqueline Dalencon , Werner Zambach , Christopher Richard Godfrey , Thomas Pitterna , Pierre Joseph Jung , Jagadish Pabba
发明人: Jerome Yves Cassayre , Peter Renold , Vladimir Bobosik , Myriem El Qacemi , Anne Jacqueline Dalencon , Werner Zambach , Christopher Richard Godfrey , Thomas Pitterna , Pierre Joseph Jung , Jagadish Pabba
IPC分类号: C07D413/12 , C07D417/14 , C07D413/14 , A01N43/82 , A01N43/44 , A01N43/76 , A01N43/56 , C07D409/12 , A01N43/80
CPC分类号: C07D413/12 , A01N43/36 , A01N43/44 , A01N43/56 , A01N43/76 , A01N43/80 , A01N43/82 , C07D409/12 , C07D413/14 , C07D417/14
摘要: A compound of formula (I): where A, B, C, G, m, n, o, p, R1, R2, R3, R4, R5, R6, X, R7, R8, R9, R10 and R11 are as defined in claim 1; or a salt or N-oxide thereof.Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
摘要翻译: 式(I)化合物:其中A,B,C,G,m,n,o,p,R1,R2,R3,R4,R5,R6,X,R7,R8,R9,R10和R11为 如权利要求1所述; 或其盐或N-氧化物。 此外,本发明涉及制备式(I)化合物的方法和中间体,其包含式(I)化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物和使用式(I)化合物控制的方法 昆虫,螨虫,线虫和软体动物害虫。
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公开(公告)号:US09867375B2
公开(公告)日:2018-01-16
申请号:US14418213
申请日:2012-07-31
IPC分类号: A01N43/653 , A01N43/56 , A01N43/80 , A01N53/00 , A01N43/08 , A01N43/36 , C07D207/09 , C07D207/20 , C07D261/04 , C07D403/10 , G06Q30/00
CPC分类号: A01N53/00 , A01N43/08 , A01N43/36 , A01N43/56 , A01N43/653 , A01N43/80 , C07D207/09 , C07D207/20 , C07D261/04 , C07D403/10 , G06Q30/018
摘要: The present invention provides methods comprising applying to a crop of soybean plants, the locus thereof, or propagation material thereof, a compound of formula (I) wherein —B1—B2—B3— is —C═N—O—, —C═N—CH2—, —N—CH2—CH2—, or —C═C—O—; R1 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl; R2 is group (X) wherein X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least one of X1, X3 and X6 is not hydrogen; A is selected from group (A1) to (A4) and Y1, Y2, Y3, R5 and R8 are as defined in claim 1. The methods are preferably for the control of stinkbugs, in particular Euschistus.
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公开(公告)号:US09204648B2
公开(公告)日:2015-12-08
申请号:US14240541
申请日:2012-08-24
IPC分类号: C07D331/04 , C07D409/12 , C07D413/12 , A01N43/80 , A01N43/36
CPC分类号: C07D413/12 , A01N43/36 , A01N43/80 , C07D331/04 , C07D409/12
摘要: The present invention relates to processes for the preparation of thietane derivatives of the formula (IA) and thietane derivatives of the formula (IB) wherein R1, R2, A1, A2, A3, A4, B, and n are as defined in the claims. The invention also relates to intermediates useful in the processes, as well as the compounds of formula (IA) and (IB) and their use as pesticides.
摘要翻译: 本发明涉及制备式(IA)的硫杂环丁烷衍生物和式(IB)的硫杂环丁烷衍生物的方法,其中R1,R2,A1,A2,A3,A4,B和n如权利要求中所定义 。 本发明还涉及可用于该方法的中间体以及式(IA)和(IB)的化合物及其作为农药的用途。
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公开(公告)号:US20140206633A1
公开(公告)日:2014-07-24
申请号:US13581137
申请日:2011-02-03
申请人: Nicholas Phillip Mulholland , Edouard Godineau , Jérôme Yves Cassayre , Peter Renold , Myriem El Qacemi , Guillaume Revol
发明人: Nicholas Phillip Mulholland , Edouard Godineau , Jérôme Yves Cassayre , Peter Renold , Myriem El Qacemi , Guillaume Revol
CPC分类号: A01N43/80 , B01J31/0271 , C07D413/12 , C07D413/14 , C07D453/04
摘要: The present invention relates to processes for the preparation of compounds of formula IB wherein A1, A2, A3, A4, L, Y1, Y2, R1, R2, R3, R4 and R5 are as defined in the claims, comprising reacting a compound of formula (II) wherein Y1, Y2, L, A1, A2, R1, R2, R3, R4 and R5 are as defined for the compound of formula (I); with hydroxylamine in the presence of water, a base and a chiral phase transfer catalyst, which chiral phase transfer catalyst is a quinine derivative. The invention also relates to compounds of formula IB and enantiomerically enriched mixtures comprising compounds of formula IB.
摘要翻译: 本发明涉及制备式IB化合物的方法,其中A1,A2,A3,A4,L,Y1,Y2,R1,R2,R3,R4和R5如权利要求中所定义,包括使 式(II)其中Y1,Y2,L,A1,A2,R1,R2,R3,R4和R5如式(I)化合物所定义; 在水存在下用羟胺,碱和手性相转移催化剂,该手性相转移催化剂是奎宁衍生物。 本发明还涉及式IB化合物和包含式IB化合物的对映体富集的混合物。
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公开(公告)号:US20140194480A1
公开(公告)日:2014-07-10
申请号:US14240140
申请日:2012-08-27
CPC分类号: A01N43/36 , A01N43/713 , A01N43/80 , A01N25/006 , A01N2300/00
摘要: The present invention provides a method for controlling termites comprising applying a liquid formulation comprising a compound of formula I to a location where termite control is needed or is expected to be needed, wherein the compound of formula (I) is wherein X is optionally substituted aryl, optionally substituted heterocyclyl, or a group selected from X1 to X5 cycle A is aryl or heteroaryl; cycle B is a saturated or partially unsaturated heterocyclyl; cycle C is aryl or heteroaryl; R1, R2, R3, R4, R5, R6 and R8 are independently hydrogen or an organic radical; R7 is haloalkyl; G is oxygen or sulfur; L is O, NH, NR1, CR3R4; n is 0, 1, 2, 3, 4 or 5; o is 0, 1, 2, 3, 4 or 5; p is 1, 2, 3, 4 or 5. The invention also relates to methods for protecting man-made structures from termites using the compounds of formula I as well as termite baits comprising the compound of formula I. The invention also provides a method for controlling ants comprising applying a liquid formulation comprising a compound of formula I to a location where ant control is needed or is expected to be needed.
摘要翻译: 本发明提供了一种控制白蚁的方法,包括将包含式I化合物的液体制剂施用于需要或预期需要白蚁控制的位置,其中式(I)化合物是其中X是任选取代的芳基 ,任选取代的杂环基,或选自X 1至X 5的基团A是芳基或杂芳基; 循环B是饱和或部分不饱和的杂环基; 环C是芳基或杂芳基; R1,R2,R3,R4,R5,R6和R8独立地是氢或有机基团; R7是卤代烷基; G是氧或硫; L是O,NH,NR1,CR3R4; n为0,1,2,3,4或5; o是0,1,2,3,4或5; p是1,2,3,4或5.本发明还涉及使用式I化合物保护人造结构免于白蚁的方法以及包含式I化合物的白蚁诱饵。本发明还提供了一种方法 用于控制蚂蚁,包括将包含式I化合物的液体制剂施用于需要或预期需要蚂蚁控制的位置。
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公开(公告)号:US20120329769A1
公开(公告)日:2012-12-27
申请号:US13580626
申请日:2011-01-31
申请人: Myriem El Qacemi , Jerome Yves Cassayre , Julie Clementine Toueg , Peter Renold , Thomas Pitterna
发明人: Myriem El Qacemi , Jerome Yves Cassayre , Julie Clementine Toueg , Peter Renold , Thomas Pitterna
IPC分类号: C07D307/28 , A01N55/04 , A01N43/08 , C07D409/12 , C07D307/33 , A01P9/00 , A01N43/653 , C07D405/04 , A01N43/40 , A01P7/04 , A01P7/02 , A01P5/00 , C07F7/22 , C07D405/10
CPC分类号: C07D307/28 , C07D307/52 , C07D307/58 , C07D405/04 , C07D405/10 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D413/12 , C07D413/14 , C07D417/14
摘要: The present invention relates to compounds of formula (I) wherein Q is Q1 or Q2 P is P1, heterocyclylor heterocyclyl substituted by one to five Z; and wherein A1, A2, A3, A4, G1, Y1, Z, R1, R2, R3 and R4 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
摘要翻译: 本发明涉及式(I)的化合物,其中Q是Q 1或Q 2是P 1,被1至5个Z取代的杂环基杂环基; 并且其中A1,A2,A3,A4,G1,Y1,Z,R1,R2,R3和R4如权利要求1中所定义; 或其盐或N-氧化物。 此外,本发明涉及制备式(I)化合物的方法和中间体,其包含式(I)化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物和使用式(I)化合物控制的方法 昆虫,螨虫,线虫和软体动物害虫。
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