Isoxazoline derivatives as insecticidal compounds
    2.
    发明授权
    Isoxazoline derivatives as insecticidal compounds 有权
    异恶唑啉衍生物作为杀虫剂

    公开(公告)号:US09247740B2

    公开(公告)日:2016-02-02

    申请号:US14240428

    申请日:2012-08-24

    摘要: The present invention provides compounds of formula (I), wherein G1 is oxygen; R1 is hydrogen; R2 is group P (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y1 is C—R6, CH or nitrogen; Y2 and Y3 are independently CH or nitrogen; wherein no more than two of Y1, Y2 and Y3 are nitrogen and wherein Y2 and Y3 are not both nitrogen; R5 is hydrogen, halogen, cyano, nitro, NH2, C1-C2alkyl, C1-C2haloalkyl, C3-C5cycloalkyl, C3-C5halocycloalkyl, C1-C2alkoxy, C1-C2haloalkoxy; R6 together with R5 forms a —CH═CH—CH═CH— bridge; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).

    摘要翻译: 本发明提供式(I)化合物,其中G1是氧; R1是氢; R2是基团P(P)L是键,亚甲基或亚乙基; A1和A2之一是S,SO或SO2,另一个是-C(R4)R4-R3是氢或甲基; 每个R 4独立地是氢或甲基; Y1是C-R6,CH或氮; Y2和Y3独立地是CH或氮; 其中Y1,Y2和Y3中不超过两个是氮,并且其中Y 2和Y 3不都是氮; R5是氢,卤素,氰基,硝基,NH2,C1-C2烷基,C1-C2卤代烷基,C3-C5环烷基,C3-C5卤代环烷基,C1-C2烷氧基,C1-C2卤代烷氧基; R6与R5一起形成-CH = CH-CH = CH-桥; X2是C-X6或氮; X1,X3和X6独立地为氢,卤素或三卤代甲基,其中X 1,X 3和X 6中的至少两个不是氢; X4是三氟甲基,二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式(I)化合物的中间体,以及使用式(I)化合物控制昆虫,螨虫,线虫或软体动物的方法。

    ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS
    4.
    发明申请
    ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS 有权
    异辛唑衍生物作为杀虫剂化合物

    公开(公告)号:US20140206606A1

    公开(公告)日:2014-07-24

    申请号:US14240428

    申请日:2012-08-24

    摘要: The present invention provides compounds of formula (I), wherein G1 is oxygen; R1 is hydrogen; R2 is group P (P) L is a bond, methylene or ethylene; one of A1 and A2 is S, SO or SO2 and the other is —C(R4)R4—R3 is hydrogen or methyl; each R4 is independently hydrogen or methyl; Y1 is C—R6, CH or nitrogen; Y2 and Y3 are independently CH or nitrogen; wherein no more than two of Y1, Y2 and Y3 are nitrogen and wherein Y2 and Y3 are not both nitrogen; R5 is hydrogen, halogen, cyano, nitro, NH2, C1-C2alkyl, C1-C2haloalkyl, C3-C5cycloalkyl, C3-C5halocycloalkyl, C1-C2alkoxy, C1-C2haloalkoxy; R6 together with R5 forms a —CH═CH—CH═CH— bridge; X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X1, X3 and X6 are not hydrogen; X4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).

    摘要翻译: 本发明提供式(I)化合物,其中G1是氧; R1是氢; R2是基团P(P)L是键,亚甲基或亚乙基; A1和A2之一是S,SO或SO2,另一个是-C(R4)R4-R3是氢或甲基; 每个R 4独立地是氢或甲基; Y1是C-R6,CH或氮; Y2和Y3独立地是CH或氮; 其中Y1,Y2和Y3中不超过两个是氮,并且其中Y 2和Y 3不都是氮; R5是氢,卤素,氰基,硝基,NH2,C1-C2烷基,C1-C2卤代烷基,C3-C5环烷基,C3-C5卤代环烷基,C1-C2烷氧基,C1-C2卤代烷氧基; R6与R5一起形成-CH = CH-CH = CH-桥; X2是C-X6或氮; X1,X3和X6独立地为氢,卤素或三卤代甲基,其中X 1,X 3和X 6中的至少两个不是氢; X4是三氟甲基,二氟甲基或氯二氟甲基。 本发明还提供了可用于制备式(I)化合物的中间体,以及使用式(I)化合物控制昆虫,螨虫,线虫或软体动物的方法。

    METHODS FOR THE CONTROL OF TERMITES AND ANTS
    9.
    发明申请
    METHODS FOR THE CONTROL OF TERMITES AND ANTS 审中-公开
    控制ERM S和蚂蚁的方法

    公开(公告)号:US20140194480A1

    公开(公告)日:2014-07-10

    申请号:US14240140

    申请日:2012-08-27

    IPC分类号: A01N43/36 A01N43/80

    摘要: The present invention provides a method for controlling termites comprising applying a liquid formulation comprising a compound of formula I to a location where termite control is needed or is expected to be needed, wherein the compound of formula (I) is wherein X is optionally substituted aryl, optionally substituted heterocyclyl, or a group selected from X1 to X5 cycle A is aryl or heteroaryl; cycle B is a saturated or partially unsaturated heterocyclyl; cycle C is aryl or heteroaryl; R1, R2, R3, R4, R5, R6 and R8 are independently hydrogen or an organic radical; R7 is haloalkyl; G is oxygen or sulfur; L is O, NH, NR1, CR3R4; n is 0, 1, 2, 3, 4 or 5; o is 0, 1, 2, 3, 4 or 5; p is 1, 2, 3, 4 or 5. The invention also relates to methods for protecting man-made structures from termites using the compounds of formula I as well as termite baits comprising the compound of formula I. The invention also provides a method for controlling ants comprising applying a liquid formulation comprising a compound of formula I to a location where ant control is needed or is expected to be needed.

    摘要翻译: 本发明提供了一种控制白蚁的方法,包括将包含式I化合物的液体制剂施用于需要或预期需要白蚁控制的位置,其中式(I)化合物是其中X是任选取代的芳基 ,任选取代的杂环基,或选自X 1至X 5的基团A是芳基或杂芳基; 循环B是饱和或部分不饱和的杂环基; 环C是芳基或杂芳基; R1,R2,R3,R4,R5,R6和R8独立地是氢或有机基团; R7是卤代烷基; G是氧或硫; L是O,NH,NR1,CR3R4; n为0,1,2,3,4或5; o是0,1,2,3,4或5; p是1,2,3,4或5.本发明还涉及使用式I化合物保护人造结构免于白蚁的方法以及包含式I化合物的白蚁诱饵。本发明还提供了一种方法 用于控制蚂蚁,包括将包含式I化合物的液体制剂施用于需要或预期需要蚂蚁控制的位置。