公开(公告)号：US4878939A

公开(公告)日：1989-11-07

申请号：US258108

申请日：1988-10-13

申请人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

发明人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

IPC分类号： C07C43/225 ,  A01N43/50 ,  A01N43/653 ,  C07C41/00 ,  C07C45/00 ,  C07C49/167 ,  C07C49/175 ,  C07C67/00 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulphur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.

摘要翻译： 其中R 1和R 2各自独立地表示具有多于一个碳原子的烷基，或者R 1表示二氯甲基，三氯甲基，氯乙烯基或二氯乙烯基，并且R 2表示烷基，R 3表示烷基， 酮基或CH（OH）基，Z表示氮原子或CH基，X表示氧或硫，Ar表示任选取代的苯基，或其与酸和金属盐的加成产物对真菌有活性， 植物生长。 还显示了其新的中间体。

公开(公告)号：US4917720A

公开(公告)日：1990-04-17

申请号：US256808

申请日：1988-10-12

申请人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

发明人： Gerhard Jager ,  Manfred Jautelat ,  Wolfgang Kramer ,  Karl H. Buchel ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

IPC分类号： C07C43/225 ,  A01N43/50 ,  A01N43/653 ,  C07C41/00 ,  C07C45/00 ,  C07C49/167 ,  C07C49/175 ,  C07C67/00 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulfur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.

公开(公告)号：US4647302A

公开(公告)日：1987-03-03

申请号：US619949

申请日：1984-06-12

申请人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

发明人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

IPC分类号： A01N43/653 ,  C07D249/08 ,  C07D521/00 ,  A01N43/64 ,  C07F1/08

CPC分类号： C07D231/12 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： 1-Vinyltriazole compounds of the formula ##STR1## wherein R.sup.1 is alkyl, substituted alkyl, cycloalkyl, aryl or substituted aryl;R.sup.2 is alkyl;R.sup.3 is alkyl, cycloalkyl, cycloalkenyl, substituted cycloalkenyl, alkenyl, aryl or substituted aryl; orR.sup.2 and R.sup.3, together with the carbon to which they are bonded, represent cycloalkenyl, substituted cycloalkenyl, cycloalkyl or substituted cycloalkyl;X is the group ##STR2## or, alternatively, X may represent a keto group provided that when X is a keto group R.sup.1 is alkyl, substituted alkyl, cycloalkyl, or substituted cycloalkyl;R.sup.4 is hydrogen, alkyl, aralkyl, substituted aralkyl, acyl, carbamoyl or substituted carbamoyl;R.sup.5 is hydrogen, alkyl, aralkyl or substituted aralkyl;and acid addition salts and metal salt complexes thereof; are outstandingly effective plant growth regulants and as fungicides.

摘要翻译： 式（I）的1-乙烯基三唑化合物，其中R 1是烷基，取代的烷基，环烷基，芳基或取代的芳基; R2是烷基; R3是烷基，环烷基，环烯基，取代的环烯基，烯基，芳基或取代的芳基; 或R 2和R 3与它们所键合的碳一起代表环烯基，取代的环烯基，环烷基或取代的环烷基; 或者X可以表示酮基，条件是当X是酮基时，R 1是烷基，取代的烷基，环烷基或取代的环烷基; R4是氢，烷基，芳烷基，取代的芳烷基，酰基，氨基甲酰基或取代的氨基甲酰基; R5是氢，烷基，芳烷基或取代的芳烷基; 及其酸加成盐和金属盐络合物; 是非常有效的植物生长调节剂和杀真菌剂。

公开(公告)号：US4749405A

公开(公告)日：1988-06-07

申请号：US894734

申请日：1986-08-08

申请人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

发明人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

IPC分类号： A01N43/653 ,  A01N47/20 ,  A01N47/24 ,  C07D249/08 ,  C07D521/00 ,  A61K31/41

CPC分类号： C07D231/12 ,  A01N43/653 ,  A01N47/20 ,  A01N47/24 ,  C07D233/56 ,  C07D249/08

摘要： 1-Vinyltriazole compounds of the formula ##STR1## wherein R.sup.1 is alkyl, substituted alkyl, cycloalkyl, aryl or substituted aryl;R.sup.2 is alkyl;R.sup.3 is alkyl, cycloalkyl, cycloalkenyl, substituted cycloalkenyl, alkenyl, aryl or substituted aryl; orR.sup.2 and R.sup.3, together with the carbon to which they are bonded, represent cycloalkenyl, substituted cycloalkenyl, cycloalkyl or substituted cycloalkyl;is the group ##STR2## or, alternatively, X may represent a keto group provided that when X is a keto group, R.sup.1 is alkyl, substituted alkyl, cycloalkyl, or substituted cycloalkyl;R.sup.4 is hydrogen, alkyl, aralkyl, substituted aralkyl, acyl, carbamoyl or substituted carbamoyl;R.sup.5 is hydrogen, alkyl, aralkyl or substituted aralkyl;and acid addition salts and metal salt complexes thereof; are outstandingly effective plant growth regulants and as fungicides.

摘要翻译： 式（I）的1-乙烯基三唑化合物，其中R 1是烷基，取代的烷基，环烷基，芳基或取代的芳基; R2是烷基; R3是烷基，环烷基，环烯基，取代的环烯基，烯基，芳基或取代的芳基; 或R 2和R 3与它们所键合的碳一起代表环烯基，取代的环烯基，环烷基或取代的环烷基; 或者X可以表示酮基，条件是当X是酮基时，R 1是烷基，取代的烷基，环烷基或取代的环烷基; R4是氢，烷基，芳烷基，取代的芳烷基，酰基，氨基甲酰基或取代的氨基甲酰基; R5是氢，烷基，芳烷基或取代的芳烷基; 及其酸加成盐和金属盐络合物; 是非常有效的植物生长调节剂和杀真菌剂。

公开(公告)号：US4743293A

公开(公告)日：1988-05-10

申请号：US894437

申请日：1986-07-30

申请人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

发明人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

IPC分类号： A01N43/653 ,  C07D249/08 ,  C07D521/00 ,  A61K31/41

CPC分类号： C07D231/12 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： 1-Vinyltriazole compounds of the formula ##STR1## wherein R.sup.1 is alkyl, substituted alkyl, cycloalkyl, aryl or substituted aryl;R.sup.2 is alkyl;R.sup.3 is alkyl, cycloalkyl, cycloalkenyl, substituted cycloalkenyl, alkenyl, aryl or substituted aryl; orR.sup.2 and R.sup.3, together with the carbon to which they are bonded, represent cycloalkenyl, substituted cycloalkenyl, cycloalkyl or substituted cycloalkyl;X is the group ##STR2## or, alternatively, X may represent a keto group provided that when X is a keto group, R.sup.1 is alkyl, substituted alkyl, cycloalkyl, or substituted cycloalkyl;R.sup.4 is hydrogen, alkyl, aralkyl, substituted aralkyl, acyl, carbamoyl or substituted carbamoyl;R.sup.5 is hydrogen, alkyl, aralkyl or substituted aralkyl;and acid addition salts and metal salt complexes thereof;are outstandingly effective plant growth regulants and as fungicides.

摘要翻译： 式（I）的1-乙烯基三唑化合物，其中R 1是烷基，取代的烷基，环烷基，芳基或取代的芳基; R2是烷基; R3是烷基，环烷基，环烯基，取代的环烯基，烯基，芳基或取代的芳基; 或R 2和R 3与它们所键合的碳一起代表环烯基，取代的环烯基，环烷基或取代的环烷基; X是基团，或者可选地，X可以表示酮基，条件是当X是酮基时，R 1是烷基，取代的烷基，环烷基或取代的环烷基; R4是氢，烷基，芳烷基，取代的芳烷基，酰基，氨基甲酰基或取代的氨基甲酰基; R5是氢，烷基，芳烷基或取代的芳烷基; 及其酸加成盐和金属盐络合物; 是非常有效的植物生长调节剂和杀真菌剂。

公开(公告)号：US4486218A

公开(公告)日：1984-12-04

申请号：US294603

申请日：1981-08-20

申请人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

发明人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

IPC分类号： A01N43/653 ,  C07D249/08 ,  C07D521/00 ,  A01N43/64

CPC分类号： C07D231/12 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： 1-Vinyltriazole compounds of the formula ##STR1## wherein R.sup.1 is alkyl, substituted alkyl, cycloalkyl, aryl or substituted aryl;R.sup.2 is alkyl;R.sup.3 is alkyl, cycloalkyl, cycloalkenyl, substituted cycloalkenyl, alkenyl, aryl or substituted aryl; orR.sup.2 and R.sup.3, together with the carbon to which they are bonded, represent cycloalkenyl, substituted cycloalkenyl, cycloalkyl or substituted cycloalkyl;X is the group ##STR2## or, alternatively, X may represent a keto group provided that when X is a keto group, R.sup.1 is alkyl, substituted alkyl, cycloalkyl, or substituted cycloalkyl;R.sup.4 is hydrogen, alkyl, aralkyl, substituted aralkyl, acyl, carbamoyl or substituted carbamoyl;R.sup.5 is hydrogen, alkyl, aralkyl or substituted aralkyl;and acid addition salts and metal salt complexes thereof; are outstandingly effective plant growth regulants and as fungicides.

摘要翻译： 式（I）的1-乙烯基三唑化合物，其中R 1是烷基，取代的烷基，环烷基，芳基或取代的芳基; R2是烷基; R3是烷基，环烷基，环烯基，取代的环烯基，烯基，芳基或取代的芳基; 或R 2和R 3与它们所键合的碳一起代表环烯基，取代的环烯基，环烷基或取代的环烷基; X是基团，或者可选地，X可以表示酮基，条件是当X是酮基时，R 1是烷基，取代的烷基，环烷基或取代的环烷基; R4是氢，烷基，芳烷基，取代的芳烷基，酰基，氨基甲酰基或取代的氨基甲酰基; R5是氢，烷基，芳烷基或取代的芳烷基; 及其酸加成盐和金属盐络合物; 是非常有效的植物生长调节剂和杀真菌剂。

公开(公告)号：US4315764A

公开(公告)日：1982-02-16

申请号：US118335

申请日：1980-02-04

申请人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

发明人： Wolf Reiser ,  Wilfried Draber ,  Karl H. Buchel ,  Klaus Lurssen ,  Paul-Ernst Frohberger ,  Volker Paul

IPC分类号： A01N43/653 ,  A01N47/12 ,  A01N47/20 ,  C07D249/08 ,  C07D521/00 ,  A01N43/64

CPC分类号： C07D231/12 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

摘要： 1-Allyl-triazole derivatives of the formula ##STR1## in which R represents hydrogen, alkyl or optionally substituted aralkyl,R.sup.1 represents optionally substituted alkyl, cycloalkyl or optionally substituted aryl,R.sup.2 represents alkyl andR.sup.3 represents alkyl, cycloalkyl, optionally substituted cycloalkenyl, alkenyl or optionally substituted aryl, orR.sup.2 and R.sup.3, together with the carbon atom to which they are bonded, represent optionally substituted cycloalkenyl or cycloalkylX represent the group ##STR2## or the keto group, R.sup.4 represents hydrogen, alkyl, optionally substituted aralkyl, acyl or optionally substituted carbamoyl andR.sup.5 represents hydrogen, alkyl or optionally substituted aralkyl,or acid addition salts or metal salt complexes thereof are characterized by fungicidal and plant growth regulatory activity.

摘要翻译： 其中R表示氢，烷基或任选取代的芳烷基，R1表示任选取代的烷基，环烷基或任选取代的芳基，R 2表示烷基，R 3表示烷基，环烷基，任选取代的环烯基， 烯基或任选取代的芳基，或R 2和R 3与它们所键合的碳原子一起代表任选取代的环烯基或环烷基X代表基团或酮基，R 4表示氢，烷基，任选取代的芳烷基， 酰基或任选取代的氨基甲酰基，R 5表示氢，烷基或任选取代的芳烷基，或其酸加成盐或金属盐络合物的特征在于杀真菌和植物生长调节活性。

公开(公告)号：US4515617A

公开(公告)日：1985-05-07

申请号：US519609

申请日：1983-08-02

申请人： Graham Holmwood ,  Klaus Lurssen ,  Paul-Ernst Frohberger

发明人： Graham Holmwood ,  Klaus Lurssen ,  Paul-Ernst Frohberger

IPC分类号： A01N43/54 ,  C07D239/26

CPC分类号： C07D239/26 ,  A01N43/54

摘要： A benzyl-pyrimidinylalkyl-ether of the formula ##STR1## in which R is alkyl, optionally substituted cycloalkyl or optionally substituted phenyl, andX.sup.1, X.sup.2 and X.sup.3 each independently is hydrogen, halogen, alkyl, cycloalkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy, halogenoalkylthio, cyano, optionally substituted phenoxy, optionally substituted phenylalkyl or optionally substituted phenylalkoxy,or an acid addition salt or metal salt complex thereof, which possesses fungicidal and plant growth-regulating properties. The corresponding pyrimidinyl-carbinols are also new.

摘要翻译： 其中R为烷基，任选取代的环烷基或任选取代的苯基，且X 1，X 2和X 3各自独立地为氢，卤素，烷基，环烷基，烷氧基，烷硫基，卤代烷基，卤代烷氧基的苄基 - 嘧啶基烷基 - 醚 ，卤代烷硫基，氰基，任选取代的苯氧基，任选取代的苯基烷基或任选取代的苯基烷氧基，或其酸加成盐或金属盐络合物，其具有杀真菌剂和植物生长调节性质。 相应的嘧啶基 - 甲醇也是新的。

公开(公告)号：USRE32796E

公开(公告)日：1988-12-06

申请号：US636644

申请日：1984-08-01

申请人： Graham Holmwood ,  Klaus Lurssen ,  Paul-Ernst Frohberger

发明人： Graham Holmwood ,  Klaus Lurssen ,  Paul-Ernst Frohberger

IPC分类号： A01N43/54 ,  C07D239/26

CPC分类号： C07D239/26 ,  A01N43/54

摘要： A benzyl-pyrimidinylalkyl-ether of the formula ##STR1## in which R is alkyl, optionally substituted cycloalkyl or optionally substituted phenyl, andX.sup.1, X.sup.2 and X.sup.3 each independently is hydrogen, halogen, alkyl, cycloalkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy, halogenoalkylthio, cyano, optionally substituted phenoxy, optionally substituted phenylalkyl or optionally substituted phenylalkoxy,or an acid addition salt or metal salt complex thereof, which possesses fungicidal and plant growth-regulating properties. The corresponding pyrimidinyl-carbinols are also new.

公开(公告)号：US4436907A

公开(公告)日：1984-03-13

申请号：US344261

申请日：1982-01-28

申请人： Graham Holmwood ,  Klaus Lurssen ,  Paul-Ernst Frohberger

发明人： Graham Holmwood ,  Klaus Lurssen ,  Paul-Ernst Frohberger

IPC分类号： A01N43/54 ,  C07D239/26

CPC分类号： C07D239/26 ,  A01N43/54

摘要： A benzyl-pyrimidinylalkyl-ether of the formula ##STR1## in which R is alkyl, optionally substituted cycloalkyl or optionally substituted phenyl, andX.sup.1, X.sup.2 and X.sup.3 each independently is hydrogen, halogen, alkyl, cycloalkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy, halogenoalkylthio, cyano, optionally substituted phenoxy, optionally substituted phenylalkyl or optionally substituted phenylalkoxy,or an acid addition salt or metal salt complex thereof, which possesses fungicidal and plant growth-regulating properties. The corresponding pyrimidinyl-carbinols are also new.

摘要翻译： 其中R为烷基，任选取代的环烷基或任选取代的苯基，且X 1，X 2和X 3各自独立地为氢，卤素，烷基，环烷基，烷氧基，烷硫基，卤代烷基，卤代烷氧基的苄基 - 嘧啶基烷基 - 醚 ，卤代烷硫基，氰基，任选取代的苯氧基，任选取代的苯基烷基或任选取代的苯基烷氧基，或其酸加成盐或金属盐络合物，其具有杀真菌剂和植物生长调节性质。 相应的嘧啶基 - 甲醇也是新的。