公开(公告)号：US07056941B1

公开(公告)日：2006-06-06

申请号：US09462647

申请日：1998-07-02

申请人： Bernd Müller ,  Hubert Sauter ,  Herbert Bayer ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Arne Ptock ,  Reinhard Kirstgen ,  Norbert Götz ,  Roland Götz ,  Franz Röhl ,  Eberhard Ammermann ,  Volker Harries ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Bernd Müller ,  Hubert Sauter ,  Herbert Bayer ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Arne Ptock ,  Reinhard Kirstgen ,  Norbert Götz ,  Roland Götz ,  Franz Röhl ,  Eberhard Ammermann ,  Volker Harries ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： A01N43/653 ,  C07D249/12

CPC分类号： A01N43/80 ,  A01N43/653 ,  C07D249/12

摘要： 2-[Pyrazolyl- and triazolyl-3′-oxymethylene]phenylisoxazolones, -triazolones and -tetrazolones of formula I where: X is a group A, B or C,  where # denotes the bond with the phenyl ring, Ra is hydrogen, halogen, alkyl or alkoxy, Rb is alkyl; Y is N or CRc, where Rc is hydrogen, halogen or alkyl; n is 0, 1, 2, 3 or 4, where the substituents R1 may be different if n is greater than 1; R1 is nitro, cyano, halogen, alkyl with or without substitution or alkoxy with or without substitution or is additionally, if n is 2, an optionally substituted 3 or 4 membered bridge which forms together with the ring to which it is attached a bicyclic partially unsaturated or aromatic radical; R2 is hydrogen, nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, alkylthio or alkoxycarbonyl; R3 is optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aryl or optionally substituted hetaryl, their preparation and their use for controlling unwanted animal pests or harmful fungi.

摘要翻译： 2- [吡唑基 - 和三唑基-3'-甲醛]苯基异恶唑酮，式I的三唑酮和四唑酮其中：X是A，B或C基团，其中＃表示与苯环的键，R a 氢，卤素，烷基或烷氧基，R b是烷基; Y是N或CR，其中R c是氢，卤素或烷基; n为0,1,2,3或4，其中如果n大于1，则取代基R 1可以不同; R 1是硝基，氰基，卤素，具有或不具有取代的烷基或具有或不具有取代的烷氧基，或者另外，如果n是2，则与环一起形成的任选取代的3或4元桥 其连接有双环部分不饱和或芳族基团; R 2是氢，硝基，氰基，卤素，烷基，卤代烷基，烷氧基，烷硫基或烷氧基羰基; R 3是任选取代的烷基，任选取代的环烷基，任选取代的芳基或任选取代的杂芳基，它们的制备及其用于防治有害动物害虫或有害真菌的用途。

公开(公告)号：US06537989B1

公开(公告)日：2003-03-25

申请号：US09806608

申请日：2001-04-02

申请人： Markus Gewehr ,  Wassilios Grammenos ,  Hubert Sauter ,  Herbert Bayer ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries

发明人： Markus Gewehr ,  Wassilios Grammenos ,  Hubert Sauter ,  Herbert Bayer ,  Andreas Gypser ,  Bernd Müller ,  Arne Ptock ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  Volker Harries

IPC分类号： A61K3155

CPC分类号： C07D273/00 ,  A01N43/88

摘要： The present invention relates to azadioxacycloalkenes of the formula I in which the substituents R1 to R5 and X, the index n and the bridge member W have the following meanings: R1 is C1-C4-alkyl, halogen, C1-C4-haloalkyl, C3-C6-cycloalkyl; R2 is C1-C4-alkyl, C1-C4-haloalkyl, C3-C4-alkenyl, C3-C4-haloalkenyl, C3-C4-alkynyl or C3-C4-haloalkynyl; R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl or unsubstituted or substituted phenyl; R4 is ═CRaRb, —CRd═CRaRb or ═N—ORc, where Ra, Rb, Rc and Rd are each as defined in claim 1; R5 is nitro, cyano, halogen, C1-C6-alkyl or, in the case that n is 2, additionally a bridge which is attached to two adjacent ring atoms; n is 0, 1, 2, 3 or 4, where the substituents R1 may be different if n is greater than 1; X is C1-C4-alkoxy-N═, C1-C4-alkoxy-CH═ or R6—CH═, where R6 is as defined in claim 1 W is unsubstituted or substituted C1-C3-alkylene.

摘要翻译： 本发明涉及取代基R1至R5和X，指数n和桥连构件W具有以下含义的式Iin的二恶唑环烯烃：R1为C1-C4烷基，卤素，C1-C4卤代烷基，C3- C6-环烷基; R2是C1-C4-烷基，C1-C4卤代烷基，C3-C4-烯基，C3-C4-卤代烯基，C3-C4-炔基或C3-C4-卤代炔基; R3是氢，C1-C4- 烷基，C1-C4卤代烷基或未取代或取代的苯基; R4是= CRaRb，-CRd = CRaRb或= N-ORc，其中Ra，Rb，Rc和Rd分别如权利要求1中所定义; R5是硝基，氰基， 卤素，C 1 -C 6 - 烷基，或在n为2的情况下，另外是连接到两个相邻环原子上的桥; n为0,1,2,3或4，其中如果n 大于1; X为C 1 -C 4 - 烷氧基-N =，C 1 -C 4 - 烷氧基-CH =或R 6 -CH =，其中R 6如权利要求1W中所定义，为未取代或取代的C 1 -C 3 - 亚烷基。

公开(公告)号：US06469195B1

公开(公告)日：2002-10-22

申请号：US09830365

申请日：2001-04-25

申请人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Oliver Cullmann ,  Markus Gewehr ,  Bernd Müller ,  Arne Ptock ,  Norbert Götz ,  Roland Götz ,  Thorsten Volk ,  Eberhard Ammermann ,  Thomas Grote ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Oliver Cullmann ,  Markus Gewehr ,  Bernd Müller ,  Arne Ptock ,  Norbert Götz ,  Roland Götz ,  Thorsten Volk ,  Eberhard Ammermann ,  Thomas Grote ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： C07C22900

CPC分类号： C07C251/48 ,  C07C69/738

摘要： 2-Phenoxyphenylacetic acid derivatives of the formula I where the substituents and the index have the following meanings: A is  where R1 is halogen, C1-C4-alkyl, C1-C4-alkoxy, CF3, C1-C4-haloalkoxy, formyl, C(═O)NRaRb or C(Ra)═NORb; Ra is hydrogen or C1-C4-alkyl; Rb is C1-C4-alkyl; n is 1, 2, 3 or 4, where the groups R1 may be different if n is not 1; R2 is halogen, CH3 or CF3; m is 0 or 1; and X is OCH3 or NHCH3; processes and intermediates for preparing the compounds I and the use of the compounds I for controlling harmful fungi are described.

摘要翻译： 式I的2-苯氧基苯基乙酸衍生物，其中取代基和指数具有以下含义：A是其中R 1是卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，CF 3，C 1 -C 4 - 卤代烷氧基，甲酰基，C（= O）NR a R b或C（R a）= NOR b; R a是氢或C 1 -C 4烷基; R b是C 1 -C 4 - 烷基; n是1,2,3或4，其中如果n不是 1; R2是卤素，CH3或CF3; m是0或1; 和X是OCH 3或NHCH 3;描述了制备化合物I的方法和中间体以及用于控制有害真菌的化合物I的用途。

公开(公告)号：US06451790B1

公开(公告)日：2002-09-17

申请号：US09889164

申请日：2001-07-11

申请人： Markus Gewehr ,  Hubert Sauter ,  Bernd Müller ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Oliver Cullmann ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Volker Harries ,  Roland Götz ,  Thomas Grote

发明人： Markus Gewehr ,  Hubert Sauter ,  Bernd Müller ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Oliver Cullmann ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Volker Harries ,  Roland Götz ,  Thomas Grote

IPC分类号： C07D41312

CPC分类号： C07D413/12 ,  A01N43/82 ,  A01N43/88 ,  C07D231/20 ,  C07D249/12 ,  C07D413/14

摘要： Compounds of formula I wherein W is optionally substituted alkylene; Y is N or CRa; Ra is hydrogen, halogen or alkyl; R1n represents hydrogen or 1 to 4 substituents; R2 is hydrogen, nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, alkylthio or alkoxycarbonyl; R3 is optionally substituted alkyl, cycloalkyl, aryl or hetaryl; A is N—OR4, CH—OR4, CH—SR4 or CHR5; R4 is alkyl or haloalkyl; R5 is halogen, alkyl or haloalkyl; methods and intermediates for their preparation. The compounds and compositions comprising them are useful for combating animal pests and harmful fungi.

摘要翻译： 式I的化合物，其中W是任选取代的亚烷基; Y是N或CR a; R a是氢，卤素或烷基; R 11代表氢或1-4个取代基; R 2是氢，硝基，氰基，卤素，烷基，卤代烷基，烷氧基，烷硫基或 烷氧基羰基; R3是任选取代的烷基，环烷基，芳基或杂芳基; A是N-OR4，CH-OR4，CH-SR4或CHR5; R4是烷基或卤代烷基; R5是卤素，烷基或卤代烷基;其制备方法和中间体 。 包含它们的化合物和组合物可用于对抗动物害虫和有害真菌。

公开(公告)号：US06372766B1

公开(公告)日：2002-04-16

申请号：US09529806

申请日：2000-04-20

申请人： Wassilios Grammenos ,  Klaus Oberdorf ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Markus Gewehr ,  Thomas Grote ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Gerhard Hamprecht ,  Norbert Götz ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Wassilios Grammenos ,  Klaus Oberdorf ,  Hubert Sauter ,  Andreas Gypser ,  Herbert Bayer ,  Markus Gewehr ,  Thomas Grote ,  Bernd Müller ,  Arne Ptock ,  Franz Röhl ,  Gerhard Hamprecht ,  Norbert Götz ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： A01N4340

CPC分类号： C07D213/64 ,  A01N43/40

摘要： Substituted 2-(2′-pyridyloxy)phenylacetamides I, where R1 is fluorine, chlorine, CH3 or halomethyl; R2 is fluorine, bromine, alkyl or halomethyl; R3 is hydrogen or one of the radicals mentioned under R2; and R2 is 6-chloro if R3 is hydrogen, R3 is 5-chloro if R2 is fluorine and the compound in which R1, R2 and R3 are each chlorine with the proviso that R1 may not be chlorine if R2 is 5-trifluoromethyl and R3 is hydrogen, and processes for their preparation and their use for controlling harmful fungi and animal pests are described.

摘要翻译： 取代的2-（2'-吡啶基氧基）苯基乙酰胺I，其中R 1是氟，氯，CH 3或卤代甲基; R 2是氟，溴，烷基或卤代甲基; R 3是氢或在R 2下提及的一个基团; 如果R 3为氢，R 2为6-氯，如果R 2为氟，则R 3为5-氯，并且其中R 1，R 2和R 3各自为氯的化合物，条件是如果R 2为5-三氟甲基并且R 3为氢，则R 1可不为氯， 并描述了其制备方法及其用于控制​​有害真菌和动物害虫的用途。

公开(公告)号：US06225349B1

公开(公告)日：2001-05-01

申请号：US09355278

申请日：1999-07-28

申请人： Herbert Bayer ,  Hubert Sauter ,  Bernd Müller ,  Wassilios Grammenos ,  Reinhard Kirstgen ,  Andreas Gypser ,  Arne Ptock ,  Thomas Grote ,  Franz Röhl ,  Michael Rack ,  Roland Götz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Volker Harries

发明人： Herbert Bayer ,  Hubert Sauter ,  Bernd Müller ,  Wassilios Grammenos ,  Reinhard Kirstgen ,  Andreas Gypser ,  Arne Ptock ,  Thomas Grote ,  Franz Röhl ,  Michael Rack ,  Roland Götz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Volker Harries

IPC分类号： A01N3750

CPC分类号： C07C259/02

摘要： Hydroximic acid halides of the formula I where the substituents have the following meanings: X is NOCH3, CHOCH3 or CHCH3; Y is O or NH; R1 is halogen; R2 is unsubstituted or substituted alkyl, alkenyl, alkynyl, cycloalkyl or aryl; R3 is unsubstituted or substituted alkyl, alkoxyalkyl, cycloalkyl-alkyl, alkenyl and alkynyl, their salts, processes for their preparation, and their use.

摘要翻译： 式I的氢酰亚胺卤化物，其中取代基具有以下含义：X为NOCH 3，CHOCH 3或CHCH 3; Y为O或NH; R 1为卤素; R 2为未取代或取代的烷基，烯基，炔基，环烷基或芳基; 或取代的烷基，烷氧基烷基，环烷基 - 烷基，烯基和炔基，它们的盐，它们的制备方法及其用途。

公开(公告)号：US07300908B2

公开(公告)日：2007-11-27

申请号：US10482216

申请日：2002-07-03

申请人： Bernd Müller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

发明人： Bernd Müller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/48

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n=0 or a whole number of 1-5; R=halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R1=alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R1 being able to be substituted according to the description; R2=alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi

摘要翻译： 式（I）的三唑并嘧啶，其中指数和取代基具有以下含义：n = 0或整数1-5; 环烷氧基，烷氧基羰基，链烯氧基羰基，烷氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰基，肟基烷基，链烯基肟基羰基，烷氧基羰基，烷氧基羰基， 烷基羰基，链烯基羰基，炔基羰基，环烷基羰基或五至十元饱和，部分不饱和或芳族杂环，含有一至四个O，N或S基团的杂原子; R 1 =烷基，烯基，炔基，环烷基，环烯基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环，其含有一至四个O，N或S ，R和/或R 1能够根据描述进行取代; 可以被卤素，氰基，硝基，烷氧基或烷氧基羰基取代的烷基，烯基或炔基。 本发明还涉及生产所述化合物的方法，含有该化合物的试剂及其在控制有害真菌中的用途

公开(公告)号：US07071334B2

公开(公告)日：2006-07-04

申请号：US10474461

申请日：2002-04-06

申请人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 6-(2-Chloro-6-fluoro-phenyl)-triazolopyrimidines of formula (I), in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or partially or fully halogenated or may be substituted as defined in the description. R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; X is cyano, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi

摘要翻译： 式（I）的6-（2-氯-6-氟 - 苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基， 炔基，链烯基或卤代烷基，环烷基，二环烷基，苯基，萘基或含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环基，或5-或6-元 含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的杂芳基，或其中R 1和R 2基团可以是未取代的或部分或完全的 卤化的或可以如说明书中所定义的取代。 R 1和R 2与中间的氮原子一起表示含有1-4个氮原子或一至三个氮原子的一个5-或6-元杂环，一个 硫或氧原子，其可以被取代; X是氰基，烷氧基，卤代烷氧基或烯氧基; 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途

公开(公告)号：US06562833B1

公开(公告)日：2003-05-13

申请号：US09701859

申请日：2000-12-05

申请人： Bernd Müller ,  Hubert Sauter ,  Herbert Bayer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Norbert Götz ,  Thomas Grote ,  Michael Rack ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  John-Bryan Speakman

发明人： Bernd Müller ,  Hubert Sauter ,  Herbert Bayer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Norbert Götz ,  Thomas Grote ,  Michael Rack ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  John-Bryan Speakman

IPC分类号： C07D23942

CPC分类号： C07D239/42 ,  A01N43/54

摘要： 2-(N-phenylamino)pyrimidines of the formula I, where: R1, R3 independently of one another are cyano, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or are C3-C8-cycloalkyl or a group C(═NORx)Ry R2 is halogen, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or R1 and R2 together with the two linking carbon atoms form a fused-on partially unsaturated 4- to 8-membered ring which may be up to trisubstituted by identical or different substituents selected from the group consisting of C1-C4-alkyl, halogen and C1-C4-alkoxy-carbonyl, which may contain a carbonyl group and/or, in addition to the multiple bond of the pyrimidine ring, a double bond and/or which may be interrupted by O, S or N—(C1-C4-alkyl); the substituents R4 to R8, Rx, Ry, Ra and Rb are as defined in the description; are used as fungicides.

摘要翻译： 式I的2-（N-苯基氨基）嘧啶，其中：R 1，R 3彼此独立地是氰基，C 1 -C 8 - 烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，其中基团烷基，烯基和 炔基可以被氰基，卤素，C 1 -C 4 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代，或者是C 3 -C 8 - 环烷基或C（= NOR x）R 1 R 2是卤素，C 1 -C 8烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，其中基团烷基，烯基和炔基可以被氰基，卤素，C 1 -C 4 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代，或者R 1和R 2与两个连接碳原子一起形成稠合 - 部分不饱和的4-至8-元环，其可以由可以含有羰基的C 1 -C 4 - 烷基，卤素和C 1 -C 4 - 烷氧基 - 羰基的相同或不同取代基取代三取代， /或除了嘧啶环的多重键之外，可以被O，S或N-（C 1 -C 4 - 烷基）中断的双键和/或被中间的取代基取代基R4至R8，Rx，Ry，Ra 和Rb如t所定义 他的描述;被用作杀真菌剂。

公开(公告)号：US06482984B2

公开(公告)日：2002-11-19

申请号：US09760710

申请日：2001-01-17

申请人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Arne Ptock ,  Bernd Müller ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Arne Ptock ,  Bernd Müller ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： C07C23305

CPC分类号： C07C251/48 ,  A01N37/50

摘要： Iminooxy-substituted benzyl phenyl ethers of the formula I in which the substituents and the index are as defined below: Y is H, CH3, F or Cl; Q is C(═CHOCH3)—COOCH3, C(═CHCH3)—COOCH3, C(═NOCH3)—COOCH3, C(═NOCH3)—CONHCH3 or N(—OCH3)—COOCH3; X is hydrogen, halogen, alkyl, alkoxy or CF3; m is 1 or 2, where the radicals X may be different if m=2; R1 is alkyl and R2 is hydrogen or alkyl; or R1 and R2 together are cyclopropyl, cyclopentyl or cyclohexyl; R3 is alkyl or CF3; and R4 is alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl or haloalkynyl; processes and intermediates for their preparation, compositions comprising them, and their use, are described.

摘要翻译： 取代基和指数如下定义的式Iin的亚氨氧基取代的苄基苯基醚：Y是H，CH 3，F或Cl; Q是C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C （= NOCH 3）-COOCH 3，C（= NOCH 3）-CONHCH 3或N（-OCH 3）-COOCH 3; X是氢，卤素，烷基，烷氧基或CF 3; m是1或2，其中基团X可以不同，如果m = 2; R 1是烷基，R 2是氢或烷基; 或者R 1和R 2一起是环丙基，环戊基或环己基; R 3是烷基或CF 3; 和R 4是烷基，烯基，炔基，卤代烷基，卤代烯基或卤代炔基;其制备方法和中间体，包含它们的组合物及其用途。