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![Substituted [(5H-pyrrolo[2,1-c][1,4]benzodiazepin-11-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid compounds as dual activity H1 inverse agonists/5-HT2A antagonists](/abs-image/US/2012/11/20/US08314092B2/abs.jpg.150x150.jpg)
1.发明授权Substituted [(5H-pyrrolo[2,1-c][1,4]benzodiazepin-11-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid compounds as dual activity H1 inverse agonists/5-HT2A antagonists 有权取代的[（5H-吡咯并[2,1-c] [1,4]苯并二氮杂-11-基）哌嗪-1-基] -2,2-二甲基丙酸化合物作为双活性H1反向激动剂/ 5-HT2A拮抗剂公开(公告)号：US08314092B2
公开(公告)日：2012-11-20
申请号：US13357627
申请日：2012-01-25
Applicant: Anne Marie Camp , Peter Thaddeus Gallagher , Andrew James Ledgard , Adam Jan Sanderson , David Andrew Coates
Inventor： Anne Marie Camp , Peter Thaddeus Gallagher , Andrew James Ledgard , Adam Jan Sanderson , David Andrew Coates
IPC: A61P25/20 , A61K31/5517 , C07D487/04
CPC classification number: C07D487/04
Abstract: A dual H1/5-HT2A receptor antagonist of the formula: its uses, and methods for its preparation are described.
Abstract translation: 描述了下式的双重H1 / 5-HT2A受体拮抗剂：其用途及其制备方法。
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Patent Agency Ranking
![(Thieno[2,3-b][1,5]benzoxazepin-4-yl)piperazin-1-yl compounds as dual activity H1 inverse agonists/5-HT2A antagonists](/abs-image/US/2016/12/06/US09512140B2/abs.jpg.150x150.jpg)
2.发明授权(Thieno[2,3-b][1,5]benzoxazepin-4-yl)piperazin-1-yl compounds as dual activity H1 inverse agonists/5-HT2A antagonists 有权（噻吩并[2,3-b] [1,5]苯并氧氮杂-4-基）哌嗪-1-基化合物作为双重活性H1反向激动剂/ 5-HT2A拮抗剂公开(公告)号：US09512140B2
公开(公告)日：2016-12-06
申请号：US14131695
申请日：2012-08-22
Applicant: Andrew James Ledgard
Inventor： Andrew James Ledgard
IPC: A61K31/553 , C07D498/04 , A61K45/06
CPC classification number: C07D498/04 , A61K31/553 , A61K45/06
Abstract: A dual H1 inverse agonist/5-HT2A receptor antagonist of the formula: its uses, and methods for its preparation are described.
Abstract translation: 描述其用途及其制备方法。
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![(THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS](/abs-image/US/2014/06/19/US20140171411A1/abs.jpg.150x150.jpg)
3.发明申请(THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS 有权（THIENO [2,3-b] [1,5]苯并恶唑-4-基）哌嗪-1-基化合物作为双活性H1反相激动剂/ 5-HT2A拮抗剂公开(公告)号：US20140171411A1
公开(公告)日：2014-06-19
申请号：US14131695
申请日：2012-08-22
Applicant: Andrew James Ledgard
Inventor： Andrew James Ledgard
IPC: C07D498/04 , A61K45/06 , A61K31/553
CPC classification number: C07D498/04 , A61K31/553 , A61K45/06
Abstract: A dual H1 inverse agonist/5-HT2A receptor antagonist of the formula (I), its uses, and methods for its preparation are described.
Abstract translation: 描述了式（I）的双H1逆激动剂/ 5-HT2A受体拮抗剂，其用途及其制备方法。
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![(Thieno[2,3-b][1,5]benzoxazepin-4-yl)piperazin-1-yl compounds as dual activity H1 inverse agonists/5-HT2A antagonists](/abs-image/US/2016/11/01/US09481688B2/abs.jpg.150x150.jpg)
4.发明授权(Thieno[2,3-b][1,5]benzoxazepin-4-yl)piperazin-1-yl compounds as dual activity H1 inverse agonists/5-HT2A antagonists 有权（噻吩并[2,3-b] [1,5]苯并氧氮杂-4-基）哌嗪-1-基化合物作为双重活性H1反向激动剂/ 5-HT2A拮抗剂公开(公告)号：US09481688B2
公开(公告)日：2016-11-01
申请号：US14125320
申请日：2012-07-02
Applicant: Andrew James Ledgard
Inventor： Andrew James Ledgard
IPC: A61K31/553 , C07D498/04 , A61K45/06
CPC classification number: C07D498/04 , A61K31/553 , A61K45/06
Abstract: A dual H1/5-HT2A receptor antagonist of the formula: its uses, and methods for its preparation are described.
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![(THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS](/abs-image/US/2014/05/01/US20140121199A1/abs.jpg.150x150.jpg)
5.发明申请(THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS 有权（THIENO [2,3-b] [1,5]苯并恶唑-4-基）哌嗪-1-基化合物作为双活性H1反相激动剂/ 5-HT2A拮抗剂公开(公告)号：US20140121199A1
公开(公告)日：2014-05-01
申请号：US14125320
申请日：2012-07-02
Applicant: Andrew James Ledgard
Inventor： Andrew James Ledgard
IPC: C07D498/04 , A61K45/06 , A61K31/553
CPC classification number: C07D498/04 , A61K31/553 , A61K45/06
Abstract: A dual H1/5-HT2A receptor antagonist of the formula:, its uses, and methods for its preparation are described.
Abstract translation: 描述了下式的双重H1 / 5-HT2A受体拮抗剂：其用途及其制备方法。
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![SUBSTITUTED [(5H-PYRROLO[2,1-c][1,4]BENZODIAZEPIN-11-YL)PIPERAZIN-1-YL]-2,2-DIMETHYLPROPANOIC ACID COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS](/abs-image/US/2012/08/09/US20120202797A1/abs.jpg.150x150.jpg)
6.发明申请SUBSTITUTED [(5H-PYRROLO[2,1-c][1,4]BENZODIAZEPIN-11-YL)PIPERAZIN-1-YL]-2,2-DIMETHYLPROPANOIC ACID COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS 有权取代[（5H-吡咯并[2,1-c] [1,4]苯并咪唑-1-基]哌嗪-1-基] -2,2-二甲基丙酸化合物作为双活性H1反相激动剂/ 5-HT2A拮抗剂公开(公告)号：US20120202797A1
公开(公告)日：2012-08-09
申请号：US13357627
申请日：2012-01-25
Applicant: Anne Marie CAMP , Peter Thaddeus GALLAGHER , Andrew James LEDGARD , Adam Jan SANDERSON , David Andrew COATES
Inventor： Anne Marie CAMP , Peter Thaddeus GALLAGHER , Andrew James LEDGARD , Adam Jan SANDERSON , David Andrew COATES
IPC: A61K31/5517 , A61P25/20 , C07D487/04
CPC classification number: C07D487/04
Abstract: A dual H1/5-HT2A receptor antagonist of the formula: its uses, and methods for its preparation are described.
Abstract translation: 描述了下式的双重H1 / 5-HT2A受体拮抗剂：其用途及其制备方法。
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