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1.THIAZOLE AND OXAZOLE DERIVATIVES AS ACTIVATORS OF HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS 失效
标题翻译: 作为人类过氧化物酶促反应物激活受体的激活剂的噻唑和氧唑衍生物公开(公告)号:US20070225294A1
公开(公告)日:2007-09-27
申请号:US11753848
申请日:2007-05-25
申请人: Pierette Banker , Rodolfo Cadilla , Millard Lambert , Stephen Rafferty , Daniel Sternbach , Marcos Sznaidman
发明人: Pierette Banker , Rodolfo Cadilla , Millard Lambert , Stephen Rafferty , Daniel Sternbach , Marcos Sznaidman
IPC分类号: A61K31/497 , C07D241/04 , C07D401/06 , C07D403/06 , C07D417/06
CPC分类号: C07D417/06 , C07D263/32 , C07D277/24 , C07D277/26 , C07D277/28 , C07D417/10 , C07D417/12
摘要: The present invention provides a compound of formula (I): wherein R1-R5, R25, R26, Y, y, and X2 are as defined herein. The compounds activate human peroxisome proliferater activated receptors (hPPARs) and are useful for the treatment of associated disorders such as dyslipidemia, syndrome X, hypercholesteremia, type II diabetes mellitus, type I diabetes, insulin resistance, hyperlipidemia, and obesity.
摘要翻译: 本发明提供式(I)化合物:其中R 1,R 2,R 2,R 2,R 2, SUP,Y,Y和X 2如本文所定义。 该化合物活化人类过氧化物酶体增殖物激活受体(hPPAR),并且可用于治疗相关疾病如血脂异常,X综合症,高胆固醇血症,II型糖尿病,I型糖尿病,胰岛素抵抗,高脂血症和肥胖。
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2.THIAZOLE AND OXAZOLE DERIVATIVES AS ACTIVATORS OF HUMAN PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS 失效
标题翻译: 作为人类过氧化物酶促反应物激活受体的激活剂的噻唑和氧唑衍生物公开(公告)号:US20070072871A1
公开(公告)日:2007-03-29
申请号:US11550060
申请日:2006-10-17
申请人: Pierette Banker , Rodolfo Cadilla , Millard Lambert , Stephen Rafferty , Daniel Sternbach , Marcos Sznaidman
发明人: Pierette Banker , Rodolfo Cadilla , Millard Lambert , Stephen Rafferty , Daniel Sternbach , Marcos Sznaidman
IPC分类号: A61K31/496 , C07D417/02
CPC分类号: C07D417/06 , C07D263/32 , C07D277/24 , C07D277/26 , C07D277/28 , C07D417/10 , C07D417/12
摘要: The present invention provides a compound of formula (I):
摘要翻译: 本发明提供了式(I)的化合物:
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