公开(公告)号：US07875606B2

公开(公告)日：2011-01-25

申请号：US10480376

申请日：2002-06-20

申请人： Masao Nakatani ,  Minoru Ito ,  Kyoko Kimijima ,  Masahiro Miyazaki ,  Makoto Fujinami ,  Ryohei Ueno ,  Satoru Takahashi

发明人： Masao Nakatani ,  Minoru Ito ,  Kyoko Kimijima ,  Masahiro Miyazaki ,  Makoto Fujinami ,  Ryohei Ueno ,  Satoru Takahashi

IPC分类号： A61K31/541 ,  A61K31/496 ,  C07D417/02 ,  C07D413/02

CPC分类号： C07D413/12 ,  A01N43/80 ,  A01N43/82 ,  A01N43/90

摘要： The present invention aims at providing an isoxazoline derivative and a pharmaceutically acceptable salt thereof, both having an excellent herbicidal effect and an excellent selectivity between crop and weed.The isoxazoline derivative of the present invention is represented by the following general formula: wherein R1 is a haloalkyl group; R2 is a hydrogen atom, an alkyl group, or the like; R3, R4, R5 and R6 are each a hydrogen atom, or the like; Y is a pyrrolyl group, a pyrazolyl group, an isothiazolyl group, an oxazolyl group, an imidazolyl group, a pyridazinyl group, a pyrimidinyl group, a pyrazinyl group, a triazinyl group, a triazolyl group, an oxadiazolyl group, or the like; and n is an integer of 0 to 2.

摘要翻译： 本发明的目的在于提供一种异恶唑啉衍生物及其药学上可接受的盐，它们具有优异的除草效果和作物和杂草之间优异的选择性。 本发明的异恶唑啉衍生物由以下通式表示：其中R1是卤代烷基; R2是氢原子，烷基等; R3，R4，R5和R6各自为氢原子等; Y是吡咯基，吡唑基，异噻唑基，恶唑基，咪唑基，哒嗪基，嘧啶基，吡嗪基，三嗪基，三唑基，恶二唑基等; n为0〜2的整数。