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公开(公告)号:US09079859B2
公开(公告)日:2015-07-14
申请号:US13980565
申请日:2012-01-20
申请人: John Irwin , Patrick Sutphin , Denise Chan , Sandra Turcotte , Amato Giaccia , Edwin Lai , Olga Razorenova , Michael Patrick Hay , Muriel Bonnet , Connie Sun , Raymond Tabibiazar
发明人: John Irwin , Patrick Sutphin , Denise Chan , Sandra Turcotte , Amato Giaccia , Edwin Lai , Olga Razorenova , Michael Patrick Hay , Muriel Bonnet , Connie Sun , Raymond Tabibiazar
IPC分类号: A61K31/47 , A61K31/44 , C07D401/12 , C07D413/04 , C07D277/46 , C07D231/18 , C07D213/75 , A61K31/415 , A61K31/422 , A61K31/4245 , A61K31/426 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4412 , A61K31/443 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4545 , A61K31/496 , A61K31/4965 , A61K31/505 , A61K31/506 , A61K31/5377 , A61K31/55 , C07D215/58 , C07D231/42 , C07D277/54 , C07D413/12 , G01N33/50
CPC分类号: C07D213/75 , A61K31/415 , A61K31/422 , A61K31/4245 , A61K31/426 , A61K31/44 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4412 , A61K31/443 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4545 , A61K31/47 , A61K31/496 , A61K31/4965 , A61K31/505 , A61K31/506 , A61K31/5377 , A61K31/55 , C07D215/58 , C07D231/42 , C07D277/54 , C07D401/12 , C07D413/12 , G01N33/5008
摘要: The present invention provides methods for inhibiting growth and proliferation of HIF pathway proficient cells by administering GLUT1 inhibitors of the invention to HIF pathway proficient cells.
摘要翻译: 本发明提供了通过将本发明的GLUT1抑制剂给予HIF途径精通细胞来抑制HIF通路细胞的生长和增殖的方法。
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公开(公告)号:US20140128397A1
公开(公告)日:2014-05-08
申请号:US13980565
申请日:2012-01-20
申请人: John Irwin , Patrick Sutphin , Denise Chan , Sandra Turcotte , Amato Giaccia , Edwin Lai , Olga Razorenova , Michael Patrick Hay , Muriel Bonnet , Connie Sun , Raymond Tabibiazar
发明人: John Irwin , Patrick Sutphin , Denise Chan , Sandra Turcotte , Amato Giaccia , Edwin Lai , Olga Razorenova , Michael Patrick Hay , Muriel Bonnet , Connie Sun , Raymond Tabibiazar
IPC分类号: C07D213/75 , C07D215/58 , C07D231/42 , C07D413/12 , C07D277/54 , G01N33/50 , C07D401/12
CPC分类号: C07D213/75 , A61K31/415 , A61K31/422 , A61K31/4245 , A61K31/426 , A61K31/44 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4412 , A61K31/443 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4545 , A61K31/47 , A61K31/496 , A61K31/4965 , A61K31/505 , A61K31/506 , A61K31/5377 , A61K31/55 , C07D215/58 , C07D231/42 , C07D277/54 , C07D401/12 , C07D413/12 , G01N33/5008
摘要: The present invention provides methods for inhibiting growth and proliferation of HIF pathway proficient cells by administering GLUT1 inhibitors of the invention to HIF pathway proficient cells.
摘要翻译: 本发明提供了通过将本发明的GLUT1抑制剂施用于HIF途径精通细胞来抑制HIF途径精通细胞生长和增殖的方法。
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