公开(公告)号：US20100009956A1

公开(公告)日：2010-01-14

申请号：US12444699

申请日：2007-10-26

Applicant: Jose-Miguel Coteron Lopez ,  Jose Maria Fiandor Roman ,  Senthil Kumar Kusalakumari Sukumar

Inventor： Jose-Miguel Coteron Lopez ,  Jose Maria Fiandor Roman ,  Senthil Kumar Kusalakumari Sukumar

IPC: A61K31/5377 ,  C07D239/02 ,  A61K31/505 ,  C07D401/14 ,  A61K31/497 ,  C07D413/14

CPC classification number: C07D239/42 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D417/12

Abstract: Substituted heteroaryl nitrile salts of Formula I, processes for their preparation, pharmaceutical compositions comprising such compounds and use of the compounds as cysteine protease inhibitors are provided.

Abstract translation: 提供式I的取代的杂芳基腈盐，其制备方法，包含这些化合物的药物组合物和该化合物作为半胱氨酸蛋白酶抑制剂的用途。

公开(公告)号：US20080221110A1

公开(公告)日：2008-09-11

申请号：US11550005

申请日：2006-10-17

Applicant: Nathalie Cailleau ,  David Thomas Davies ,  Joel Michael Esken ,  Alan Joseph Hennessy ,  Senthil Kumar Kusalakumari Sukumar ,  Roger Edward Markwell ,  Timothy James Miles ,  Neil David Pearson

Inventor： Nathalie Cailleau ,  David Thomas Davies ,  Joel Michael Esken ,  Alan Joseph Hennessy ,  Senthil Kumar Kusalakumari Sukumar ,  Roger Edward Markwell ,  Timothy James Miles ,  Neil David Pearson

IPC: A61K31/5025 ,  C07D237/26 ,  A61P31/04

CPC classification number: C07D471/06 ,  C07D519/00

Abstract: Tricyclic nitrogen containing compounds and their use as antibacterials

Abstract translation: 三环含氮化合物及其作为抗菌剂的用途

公开(公告)号：US20080280892A1

公开(公告)日：2008-11-13

申请号：US12090947

申请日：2006-10-17

Applicant: Nathalie Cailleau ,  David Thomas Davies ,  Joel Michael Esken ,  Alan Joseph Hennessy ,  Senthil Kumar Kusalakumari Sukumar ,  Roger Edward Markwell ,  Timothy James Miles ,  Neil David Pearson

Inventor： Nathalie Cailleau ,  David Thomas Davies ,  Joel Michael Esken ,  Alan Joseph Hennessy ,  Senthil Kumar Kusalakumari Sukumar ,  Roger Edward Markwell ,  Timothy James Miles ,  Neil David Pearson

IPC: A61K31/542 ,  C07D471/06 ,  A61K31/436 ,  C07D491/056 ,  A61K31/5025 ,  A61P31/04 ,  C07D498/04 ,  A61K31/5365 ,  C07D513/04

CPC classification number: C07D471/06 ,  C07D519/00

Abstract: Tricyclic nitrogen containing compounds and their use as antibacterials.

Abstract translation: 三环含氮化合物及其作为抗菌剂的用途。