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公开(公告)号:US20120035214A1
公开(公告)日:2012-02-09
申请号:US13262781
申请日:2010-04-01
申请人: Daniel J. McKay , Melissa Arbour , Renee Aspiotis , Austin Chen , Pierre-Andre Fournier , Michel Gallant , Yongxin Han , Helene Juteau , Patrick Lacombe , Sebastien Laliberte , Sophie Lauzon , Carmela Molinaro , Paul O'Shea , Yeeman Ramtohul , Daniel Simard , Dwight MacDonald , Bruce Mackay , Christophe Mellon , Krista Morley , Chit Tsui , Sarah Jennifer Dolman , Greg Hughes , Jacob Janey
发明人: Daniel J. McKay , Melissa Arbour , Renee Aspiotis , Austin Chen , Pierre-Andre Fournier , Michel Gallant , Yongxin Han , Helene Juteau , Patrick Lacombe , Sebastien Laliberte , Sophie Lauzon , Carmela Molinaro , Paul O'Shea , Yeeman Ramtohul , Daniel Simard , Dwight MacDonald , Bruce Mackay , Christophe Mellon , Krista Morley , Chit Tsui , Sarah Jennifer Dolman , Greg Hughes , Jacob Janey
IPC分类号: A61K31/451 , C07D401/04 , C07D401/10 , C07D211/26 , C07D211/28 , C07D401/12 , A61K31/4545 , A61K31/454 , A61P9/12 , A61P9/04 , A61P9/10 , A61P27/06 , A61P25/22 , A61P25/00 , A61P13/12 , C07D211/22
CPC分类号: C07D211/26 , C07D211/22 , C07D211/28 , C07D211/52 , C07D401/04 , C07D401/12 , C07D413/04 , C07D413/14
摘要: The present invention relates to biaryl piperidine-based renin inhibitor compounds, and their use in treating cardiovascular events and renal insufficiency.
摘要翻译: 本发明涉及联芳基哌啶基肾素抑制剂化合物及其在治疗心血管事件和肾功能不全中的用途。