-
公开(公告)号:US06924297B2
公开(公告)日:2005-08-02
申请号:US10450891
申请日:2001-12-20
申请人: Gerard Martin Paul Giblin , Haydn Terence Jones , Andrew McMurtrie Mason , Neil Derek Miller , Susan Roomans , Stephen Edward Shanahan , Ann Louise Walker
发明人: Gerard Martin Paul Giblin , Haydn Terence Jones , Andrew McMurtrie Mason , Neil Derek Miller , Susan Roomans , Stephen Edward Shanahan , Ann Louise Walker
IPC分类号: C07D401/12 , A61K31/403 , A61K31/42 , A61K31/427 , A61K31/4439 , A61P1/00 , A61P1/02 , A61P1/04 , A61P1/12 , A61P1/16 , A61P3/00 , A61P3/02 , A61P3/10 , A61P3/14 , A61P5/10 , A61P5/18 , A61P7/02 , A61P7/06 , A61P7/12 , A61P9/00 , A61P9/10 , A61P11/00 , A61P11/02 , A61P11/06 , A61P13/04 , A61P13/12 , A61P15/10 , A61P17/00 , A61P17/02 , A61P17/04 , A61P17/06 , A61P19/02 , A61P19/04 , A61P19/06 , A61P19/08 , A61P19/10 , A61P21/00 , A61P21/04 , A61P25/02 , A61P25/06 , A61P25/14 , A61P25/16 , A61P25/20 , A61P25/28 , A61P25/30 , A61P25/32 , A61P25/34 , A61P25/36 , A61P27/02 , A61P27/06 , A61P27/14 , A61P29/00 , A61P31/00 , A61P31/12 , A61P31/16 , A61P31/18 , A61P35/00 , A61P37/06 , A61P39/02 , A61P43/00 , C07D209/64 , C07D209/66 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D209/60
CPC分类号: C07D209/64 , C07D209/66
摘要: Compounds of formula (I) and pharmaceutically acceptable derivatives thereof bind with high affinity to the EP4 receptor and are of use in the treatment or prevention of conditions such as a pain, inflammatory, immunological, bone, neurodegenerative or renal disorder.
摘要翻译: 式(I)化合物及其药学上可接受的衍生物以高亲和力结合EP4受体,并且可用于治疗或预防诸如疼痛,炎症,免疫学,骨骼,神经变性或肾脏疾病的病症。