公开(公告)号：US07683070B2

公开(公告)日：2010-03-23

申请号：US11874015

申请日：2007-10-17

申请人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Stephen Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

发明人： Ping Ding ,  Robert N. Henrie, II ,  Daniel H. Cohen ,  John W. Lyga ,  David S. Rosen ,  George Theodoridis ,  Qun Zhang ,  Walter H. Yeager ,  Stephen F. Donovan ,  Stephen Shunxiang Zhang ,  Inna Shulman ,  Seong Jae Yu ,  Guozhi Wang ,  Y. Larry Zhang ,  Ariamala Gopalsamy ,  Dennis L. Warkentin ,  Paul E. Rensner ,  Ian R. Silverman ,  Thomas G. Cullen

IPC分类号： A61K31/4523 ,  A61K31/4545 ,  C07D211/06 ,  C07D239/02

CPC分类号： C07D405/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/713 ,  C07D211/14 ,  C07D211/18 ,  C07D211/22 ,  C07D211/24 ,  C07D211/26 ,  C07D211/28 ,  C07D211/32 ,  C07D211/94 ,  C07D401/06 ,  C07D401/10 ,  C07D401/12 ,  C07D401/14 ,  C07D413/12 ,  C07D417/12 ,  C07D451/14 ,  C07D513/04

摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

摘要翻译： 现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。 这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 本文完整地描述了B，D，E，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 8。 此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。