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    Optically active diazabicyclooctane derivatives and process for preparing the same
    1.
    发明授权
    Optically active diazabicyclooctane derivatives and process for preparing the same 有权
    光活性二氮杂双环辛烷衍生物及其制备方法

    公开(公告)号：US08772490B2

    公开(公告)日：2014-07-08

    申请号：US13173002

    申请日：2011-06-30

    申请人： Takao Abe ,  Masayuki Okue ,  Yoshiaki Sakamaki

    发明人： Takao Abe ,  Masayuki Okue ,  Yoshiaki Sakamaki

    IPC分类号： C07D471/08 ,  C07D211/60

    CPC分类号： C07D471/08 ,  C07B2200/07 ,  C07D211/60

    摘要： Provided are an optically active diazabicyclooctane derivative defined by formula (F) below, which is useful as a pharmaceutical intermediate for β-lactamase inhibitor, and a process for preparing the same. In formula (F) above, R1 represents CO2R, CO2M, or CONH2, wherein R represents a methyl group, a tert-butyl group, an allyl group, a benzyl group, or a 2,5-dioxopyrrolidin-1-yl group, and M represents a hydrogen atom, an inorganic cation, or an organic cation; and R2 represents a benzyl group or an allyl group.

    摘要翻译： 提供由下式（F）定义的光学活性二氮杂双环辛烷衍生物，其可用作β-内酰胺酶抑制剂的药物中间体及其制备方法。 在上述式（F）中，R 1表示CO 2 R，CO 2 M或CONH 2，其中R表示甲基，叔丁基，烯丙基，苄基或2,5-二氧代吡咯烷-1-基， M表示氢原子，无机阳离子或有机阳离子; 并且R 2表示苄基或烯丙基。

    OPTICALLY ACTIVE DIAZABICYCLOOCTANE DERIVATIVES AND PROCESS FOR PREPARING THE SAME
    2.
    发明申请
    OPTICALLY ACTIVE DIAZABICYCLOOCTANE DERIVATIVES AND PROCESS FOR PREPARING THE SAME 有权
    光学活性二氮杂环戊烷衍生物及其制备方法

    公开(公告)号：US20120165533A1

    公开(公告)日：2012-06-28

    申请号：US13173002

    申请日：2011-06-30

    申请人： Takao ABE ,  Masayuki Okue ,  Yoshiaki Sakamaki

    发明人： Takao ABE ,  Masayuki Okue ,  Yoshiaki Sakamaki

    IPC分类号： C07D471/08 ,  C07D211/60

    CPC分类号： C07D471/08 ,  C07B2200/07 ,  C07D211/60

    摘要： Provided are an optically active diazabicyclooctane derivative defined by formula (F) below, which is useful as a pharmaceutical intermediate for β-lactamase inhibitor, and a process for preparing the same. In formula (F) above, R1 represents CO2R, CO2M, or CONH2, wherein R represents a methyl group, a tert-butyl group, an allyl group, a benzyl group, or a 2,5-dioxopyrrolidin-1-yl group, and M represents a hydrogen atom, an inorganic cation, or an organic cation; and R2 represents a benzyl group or an allyl group.

    摘要翻译： 提供由下式（F）定义的光学活性二氮杂双环辛烷衍生物，其可用作β-内酰胺酶抑制剂的药物中间体及其制备方法。 在上述式（F）中，R 1表示CO 2 R，CO 2 M或CONH 2，其中R表示甲基，叔丁基，烯丙基，苄基或2,5-二氧代吡咯烷-1-基， M表示氢原子，无机阳离子或有机阳离子; 并且R 2表示苄基或烯丙基。