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公开(公告)号:US20170216263A1
公开(公告)日:2017-08-03
申请号:US15488642
申请日:2017-04-17
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Huji Turdi , Jon J. Hangeland , R. Michael Lawrence , Dong Cheng , Saleem Ahmad , Wei Meng , Robert Paul Brigance , Pratik Devasthale , Guohua Zhao
IPC: A61K31/438 , A61K31/5377 , A61K31/4439 , A61K31/4418 , A61K45/06 , C07D401/14 , C07D417/14 , C07D407/14 , C07D417/04 , C07D413/12 , C07D405/14 , C07D401/12 , C07D211/86 , C07D211/90 , C07D401/10 , A61K31/675
CPC classification number: A61K31/438 , A61K31/4418 , A61K31/4439 , A61K31/5377 , A61K31/675 , A61K45/06 , C07D211/86 , C07D211/90 , C07D221/20 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/14 , C07F9/4006 , C07F9/5352 , C07F9/59
Abstract: The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.
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2.
公开(公告)号:US09187424B1
公开(公告)日:2015-11-17
申请号:US14305098
申请日:2014-06-16
Applicant: Bristol-Myers Squibb Company
Inventor: Huji Turdi , Jon J. Hangeland , R. Michael Lawrence , Dong Cheng , Saleem Ahmad , Wei Meng , Robert Paul Brigance , Pratik Devasthale , Guohua Zhao
IPC: C07D211/90 , C07D401/04 , A61K31/4418 , A61K31/5377 , C07D401/10 , C07D413/04 , C07D401/14 , C07D221/20 , C07D413/14 , A61K45/06 , A61K31/4439 , A61K31/438
CPC classification number: A61K31/438 , A61K31/4418 , A61K31/4439 , A61K31/5377 , A61K31/675 , A61K45/06 , C07D211/86 , C07D211/90 , C07D221/20 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/14 , C07F9/4006 , C07F9/5352 , C07F9/59
Abstract: The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.
Abstract translation: 本发明提供式(I)化合物或其立体异构体或其药学上可接受的盐,其中所有变量如本文所定义。 这些化合物是可用作药物的单酰基甘油酰基转移酶2型(MGAT2)抑制剂。
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3.ARYL DIHYDROPYRIDINONES AND PIPERIDINONE MGAT2 INHIBITORS 有权
Title translation: ARYL DIHYDROPYRIDINONES和PIPERIDINONE MGAT2抑制剂公开(公告)号:US20150315144A1
公开(公告)日:2015-11-05
申请号:US14305098
申请日:2014-06-16
Applicant: Bristol-Myers Squibb Company
Inventor: Huji Turdi , Jon J. Hangeland , R. Michael Lawrence , Dong Cheng , Saleem Ahmad , Wei Meng , Robert Paul Brigance , Pratik Devasthale , Guohua Zhao
IPC: C07D211/90 , C07D401/10 , C07D413/04 , C07D401/14 , A61K31/5377 , C07D413/14 , A61K45/06 , A61K31/4418 , A61K31/4439 , A61K31/438 , C07D401/04 , C07D221/20
CPC classification number: A61K31/438 , A61K31/4418 , A61K31/4439 , A61K31/5377 , A61K31/675 , A61K45/06 , C07D211/86 , C07D211/90 , C07D221/20 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/14 , C07F9/4006 , C07F9/5352 , C07F9/59
Abstract: The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.
Abstract translation: 本发明提供式(I)化合物或其立体异构体或其药学上可接受的盐,其中所有变量如本文所定义。 这些化合物是可用作药物的单酰基甘油酰基转移酶2型(MGAT2)抑制剂。
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公开(公告)号:US20160031816A1
公开(公告)日:2016-02-04
申请号:US14883067
申请日:2015-10-14
Applicant: Bristol-Myers Squibb Company
Inventor: Huji Turdi , Jon J. Hangeland , R. Michael Lawrence , Dong Cheng , Saleem Ahmad , Wei Meng , Robert Paul Brigance , Pratik Devasthale , Guohua Zhao
IPC: C07D211/90 , C07D221/20 , C07D401/10 , C07D401/04 , C07D405/14 , C07D401/14 , C07D211/86 , C07D417/04 , C07D413/12 , C07D401/12 , C07D413/04
CPC classification number: A61K31/438 , A61K31/4418 , A61K31/4439 , A61K31/5377 , A61K31/675 , A61K45/06 , C07D211/86 , C07D211/90 , C07D221/20 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/14 , C07F9/4006 , C07F9/5352 , C07F9/59
Abstract: The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.
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5.ARYL DIHYDROPYRIDINONE AND PIPERIDINONE MGAT2 INHIBITORS 有权
Title translation: ARYL DIHYDROPRIDINONE和PIPERIDINONE MGAT2 INHIBITORS公开(公告)号:US20130143843A1
公开(公告)日:2013-06-06
申请号:US13688584
申请日:2012-11-29
Applicant: Bristol-Myers Squibb Company
Inventor: Huji Turdi , Jon J. Hangeland , R. Michael Lawrence , Dong Cheng , Saleem Ahmad , Wei Meng , Robert Paul Brigance , Pratik Devasthale
IPC: A61K31/675 , A61K31/4418 , C07D401/04 , A61K31/4439 , C07D413/04 , A61K45/06 , A61K31/438 , C07D413/14 , A61K31/5377 , C07F9/59 , C07D401/14 , C07D211/90 , C07D221/20
CPC classification number: A61K31/438 , A61K31/4418 , A61K31/4439 , A61K31/5377 , A61K31/675 , A61K45/06 , C07D211/86 , C07D211/90 , C07D221/20 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/14 , C07D407/14 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/14 , C07F9/4006 , C07F9/5352 , C07F9/59
Abstract: The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.
Abstract translation: 本发明提供式(I)化合物或其立体异构体或其药学上可接受的盐,其中所有变量如本文所定义。 这些化合物是可用作药物的单酰基甘油酰基转移酶2型(MGAT2)抑制剂。
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