公开(公告)号：US20150342188A1

公开(公告)日：2015-12-03

申请号：US14655568

申请日：2013-12-23

Applicant: DOW AGROSCIENCES LLC

Inventor： Beth Lorsbach ,  W. John Owen ,  Lindsay Stelzer ,  Chenglin Yao

IPC: A01N43/54 ,  C07D239/47

CPC classification number: A01N43/54 ,  C07D239/47

Abstract: This present disclosure is related to the field of 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-ones and their derivatives and to the use of these compounds as fungicides. Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less. The present disclosure relates to 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one compounds and their use as fungicides. The compounds of the present disclosure may offer protection against fungi and fungi like organisms including ascomycetes, basidiomycetes, deuteromycetes, and oomycetes.

Abstract translation: 本公开内容涉及1-（取代的 - 苯甲酰基）-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2（1H） - 酮及其衍生物及其用途 化合物作为杀真菌剂。 杀真菌剂是天然或合成来源的化合物，其用于保护和/或治疗植物免受由农业相关真菌引起的损害。 通常，在所有情况下，没有一种杀真菌剂是有用的。 因此，正在进行研究，以生产可能具有更好性能，更易于使用和更低成本的杀真菌剂。 本公开涉及1-（取代的 - 苯甲酰基）-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2（1H） - 酮化合物及其作为杀真菌剂的用途。 本公开的化合物可以提供对真菌和真菌的保护，所述真菌和真菌包括子囊菌纲，担子菌，芋头菌和卵菌。

公开(公告)号：US09271497B2

公开(公告)日：2016-03-01

申请号：US14655568

申请日：2013-12-23

Applicant: DOW AGROSCIENCES LLC

Inventor： Beth Lorsbach ,  W. John Owen ,  Lindsay Stelzer ,  Chenglin Yao

IPC: A01N43/54 ,  C07D239/47

CPC classification number: A01N43/54 ,  C07D239/47

Abstract: This present disclosure is related to the field of 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-ones and their derivatives and to the use of these compounds as fungicides. Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less. The present disclosure relates to 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one compounds and their use as fungicides. The compounds of the present disclosure may offer protection against fungi and fungi like organisms including ascomycetes, basidiomycetes, deuteromycetes, and oomycetes.

Abstract translation: 本公开内容涉及1-（取代的 - 苯甲酰基）-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2（1H） - 酮及其衍生物及其用途 化合物作为杀真菌剂。 杀真菌剂是天然或合成来源的化合物，其用于保护和/或治疗植物免受由农业相关真菌引起的损害。 通常，在所有情况下，没有一种杀真菌剂是有用的。 因此，正在进行研究，以生产可能具有更好性能，更易于使用和更低成本的杀真菌剂。 本公开涉及1-（取代的 - 苯甲酰基）-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2（1H） - 酮化合物及其作为杀真菌剂的用途。 本公开的化合物可以提供对真菌和真菌的保护，所述真菌和真菌包括子囊菌纲，担子菌，芋头菌和卵菌。

公开(公告)号：US20150359225A1

公开(公告)日：2015-12-17

申请号：US14655570

申请日：2013-12-23

Applicant: DOW AGROSCIENCES LLC

Inventor： Beth Lorsbach ,  Ronald Ross ,  W. John Owen ,  Jeffery D. Webster ,  Lindsay Stelzer ,  Chenglin Yao ,  Paul R. LePlae, Jr. ,  Chris V. Galliford

IPC: A01N47/40 ,  A01N43/54 ,  C07D409/12 ,  A01N47/02 ,  A01N47/18 ,  C07D413/12 ,  A01N43/80 ,  C07D417/12 ,  A01N43/78 ,  C07D239/47 ,  A01N43/56

CPC classification number: C07D417/12 ,  A01N43/54 ,  A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  A01N47/02 ,  A01N47/18 ,  A01N47/22 ,  A01N47/40 ,  C07B59/002 ,  C07B2200/05 ,  C07D239/47 ,  C07D403/12 ,  C07D409/12 ,  C07D413/12

Abstract: This present disclosure is related to the field of 3-alkyl-5-fluoro-4-substituted-imino-3,4-5 dihydropyrimidin-2(1H)-ones and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as Septoria tritici, comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil.

Abstract translation: 本公开内容涉及3-烷基-5-氟-4-取代 - 亚氨基-3,4,5-二氢嘧啶-2（1H） - 酮及其衍生物的领域以及这些化合物作为杀真菌剂的用途。 还提供了控制真菌性疾病例如小曲霉的方法，包括将有效量的杀真菌化合物施用至至少一个与植物，种子或土壤相关的表面。

公开(公告)号：US20150353506A1

公开(公告)日：2015-12-10

申请号：US14655566

申请日：2013-12-23

Applicant: DOW AGROSCIENCES LLC

Inventor： Beth Lorsbach ,  W. John Owen ,  Lindsay Stelzer ,  Chenglin Yao

IPC: C07D239/47 ,  C07D409/12 ,  A01N43/54

CPC classification number: C07D239/47 ,  A01N43/54 ,  A01N47/30 ,  A01N47/38 ,  C07D409/12 ,  A01N25/00

Abstract: This present disclosure is related to the field of to N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidine-1(2H)-carboxamide compounds and their derivatives and to the use of these compounds as fungicides. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/746,837 filed Dec. 28, 2012, which is expressly incorporated by reference herein. Background and Summary of the Invention Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.

Abstract translation: 本发明涉及N-（取代的）-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1（2H） - 甲酰胺化合物及其衍生物的领域 以及这些化合物作为杀真菌剂的使用。 本申请要求美国临时专利申请 2012年12月28日提交的第61 / 746,837号，其明确地通过引用并入本文。 背景技术杀真菌剂是天然或合成来源的化合物，其用于保护和/或治愈植物免受农业相关真菌引起的损害。 通常，在所有情况下，没有一种杀真菌剂是有用的。 因此，正在进行研究，以生产可能具有更好性能，更易于使用和更低成本的杀真菌剂。

公开(公告)号：US20160198711A1

公开(公告)日：2016-07-14

申请号：US15072035

申请日：2016-03-16

Applicant: DOW AGROSCIENCES LLC

Inventor： Beth Lorsbach ,  W. John Owen ,  Lindsay Stelzer ,  Chenglin Yao

IPC: A01N43/54 ,  A01N47/30 ,  C07D409/12 ,  C07D239/47

CPC classification number: C07D239/47 ,  A01N43/54 ,  A01N47/30 ,  A01N47/38 ,  C07D409/12 ,  A01N25/00

Abstract: This present disclosure is related to the field of to N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidme-1(2H)-carboxamide compounds and their derivatives and to the use of these compounds as fungicides. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/1746,837 filed Dec. 28, 2012, which is expressly incorporated by reference herein. Background and Summary of the Invention Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.

Abstract translation: 本发明涉及N-（取代的）-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-2（2H） - 甲酰胺化合物及其衍生物的领域 以及这些化合物作为杀真菌剂的使用。 本申请要求美国临时专利申请 2012年12月28日提交的No.61 / 1746,837，其明确地通过引用并入本文。 背景技术杀真菌剂是天然或合成来源的化合物，其用于保护和/或治愈植物免受农业相关真菌引起的损害。 通常，在所有情况下，没有一种杀真菌剂是有用的。 因此，正在进行研究，以生产可能具有更好性能，更易于使用和更低成本的杀真菌剂。

公开(公告)号：US09321734B2

公开(公告)日：2016-04-26

申请号：US14655566

申请日：2013-12-23

Applicant: DOW AGROSCIENCES LLC

Inventor： Beth Lorsbach ,  W. John Owen ,  Lindsay Stelzer ,  Chenglin Yao

IPC: C07D239/47 ,  A01N43/54 ,  C07D409/12 ,  A01N47/38

CPC classification number: C07D239/47 ,  A01N43/54 ,  A01N47/30 ,  A01N47/38 ,  C07D409/12 ,  A01N25/00

Abstract: This present disclosure is related to the field of to N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide compounds and their derivatives and to the use of these compounds as fungicides. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/746,837 filed Dec. 28, 2012, which is expressly incorporated by reference herein. Background and Summary of the Invention Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.

Abstract translation: 本发明涉及N-（取代的）-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1（2H） - 甲酰胺化合物及其衍生物的领域， 使用这些化合物作为杀菌剂。 本申请要求美国临时专利申请 2012年12月28日提交的第61 / 746,837号，其明确地通过引用并入本文。 背景技术杀真菌剂是天然或合成来源的化合物，其用于保护和/或治愈植物免受农业相关真菌引起的损害。 通常，在所有情况下，没有一种杀真菌剂是有用的。 因此，正在进行研究，以生产可能具有更好性能，更易于使用和更低成本的杀真菌剂。