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公开(公告)号:US20090170913A1
公开(公告)日:2009-07-02
申请号:US11719576
申请日:2005-12-16
申请人: James Peter Beck , Brian David Wakefield , Frederic Laurent Cordier , Esteban Dominguez-Manzanares , Kevin Matthew Gardinier , Peter Michael Greenen , Kenneth Allen Savin
发明人: James Peter Beck , Brian David Wakefield , Frederic Laurent Cordier , Esteban Dominguez-Manzanares , Kevin Matthew Gardinier , Peter Michael Greenen , Kenneth Allen Savin
IPC分类号: A61K31/428 , C07D417/04 , A61P3/04
CPC分类号: C07D263/58 , C07D277/68 , C07D277/82 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/12 , C07D417/14
摘要: The present invention relates to a melanin concentrating hormone antagonist compound of formula (I); wherein Ar1, L1, R1, q, X, R2, R3, R4, and R5 are as defined, or a pharmaceutically acceptable salt, solvate, or enantiomer thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.
摘要翻译: 本发明涉及式(I)的黑色素浓缩激素拮抗剂化合物; 其中Ar 1,L 1,R 1,q,X,R 2,R 3,R 4和R 5如所定义,或其药学上可接受的盐,溶剂合物或对映异构体可用于治疗,预防或改善与肥胖症和相关疾病相关的症状 。
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公开(公告)号:US07838543B2
公开(公告)日:2010-11-23
申请号:US11719576
申请日:2005-12-16
申请人: James Peter Beck , Brian David Wakefield , Frederic Laurent Cordier , Esteban Dominguez-Manzanares , Kevin Matthew Gardinier , Peter Michael Greenen , Kenneth Allen Savin
发明人: James Peter Beck , Brian David Wakefield , Frederic Laurent Cordier , Esteban Dominguez-Manzanares , Kevin Matthew Gardinier , Peter Michael Greenen , Kenneth Allen Savin
IPC分类号: A01N43/78 , A61K31/425 , C07D417/00 , C07D277/60
CPC分类号: C07D263/58 , C07D277/68 , C07D277/82 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/12 , C07D417/14
摘要: The present invention relates to a melanin concentrating hormone antagonist compound of formula (I); wherein Ar1, L1, R1, q, X, R2, R3, R4, and R5 are as defined, or a pharmaceutically acceptable salt, solvate, or enantiomer thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.
摘要翻译: 本发明涉及式(I)的黑色素浓缩激素拮抗剂化合物; 其中Ar 1,L 1,R 1,q,X,R 2,R 3,R 4和R 5如所定义,或其药学上可接受的盐,溶剂合物或对映异构体可用于治疗,预防或改善与肥胖症和相关疾病相关的症状 。
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公开(公告)号:US07393868B2
公开(公告)日:2008-07-01
申请号:US11446840
申请日:2006-06-05
申请人: Ana Maria Castano Mansanet , Frederic Laurent Cordier , Esteban Dominguez-Manzanares , Jian Eric Hong , William Joseph Hornback , Delu Jiang
发明人: Ana Maria Castano Mansanet , Frederic Laurent Cordier , Esteban Dominguez-Manzanares , Jian Eric Hong , William Joseph Hornback , Delu Jiang
IPC分类号: A61K31/381 , A61K31/4155 , A61K31/4418 , C07D213/61 , C07D231/16
CPC分类号: C07D257/04 , C07C311/08 , C07C323/63 , C07D213/75 , C07D213/76 , C07D231/38 , C07D333/36 , C07D409/10
摘要: The present invention relates to AMPA receptor potentiators of Formula I: formulations comprising them, methods for their use, and intermediates useful for their preparation.
摘要翻译: 本发明涉及式I的AMPA受体增强剂:包含它们的制剂,它们的使用方法和可用于其制备的中间体。
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