Wood preservative compositions containing dimethylfurancarboxyanilide
derivatives
    1.
    发明授权
    Wood preservative compositions containing dimethylfurancarboxyanilide derivatives 失效
    含有二甲基呋喃羧酰苯胺衍生物的木防腐剂组合物

    公开(公告)号:US5977168A

    公开(公告)日:1999-11-02

    申请号:US999547

    申请日:1997-12-29

    IPC分类号: A01N43/08 B27K3/34

    CPC分类号: A01N43/08 B27K3/343

    摘要: A dimethylfurancarboxyanilide compound of the formula (I): ##STR1## wherein R.sup.1 and R.sup.2 are the same or different and each is hydrogen, (C.sub.2 -C.sub.6)-alkyl, (C.sub.3 -C.sub.6)-cycloalkyl, (C.sub.3 -C.sub.6)-alkenyl, (C.sub.2 -C.sub.6) alkynyl, (C.sub.1 -C.sub.3)-halogenoalkyl, (C.sub.2 -C.sub.6)-alkoxy, (C.sub.1 -C.sub.6)-alkoxy- (C.sub.1 -C.sub.6)-alkyl, cyano, substituted amide, (C.sub.1 -C.sub.6)-alkoxy-carbonyl, benzoyl which is unsubstituted or has 1 to 2 substituents, benzoylamino which is unsubstituted or has 1 to 2 substituents; (C.sub.2 -C.sub.6)-alkanoylamino, (C.sub.3 -C.sub.6)-cycloalkylcarbonylamino, benzyl which is unsubstituted or has 1 to 2 substituents, phenyl which is unsubstituted or has 1 to 2 substituents, or (C.sub.1 -C.sub.6)-alkoxycarbonyl-(C.sub.2 -C.sub.5)-alkenylene; and R.sup.1 and R.sup.2 do not both represent hydrogen at the same time. A wood preservative containing the dimethylfurancarboxyanilide compound as an active ingredient. A method of preserving wood by applying the dimethylfurancarboxyanilide compound to wood. A wood preservative composition in which the dimethylfurancarboxyanilide compound is combined with at least one of 3-bromo-2,3-diiodo-2-propenylethylcarbamate, 3-iodo-2-propynylbutylcarbamate and 4-chlorophenyl-3-iodopropargylformal.

    摘要翻译: 式(I)的二甲基呋喃羧酰苯胺化合物:其中R 1和R 2相同或不同,各自为氢,(C 2 -C 6) - 烷基,(C 3 -C 6) - 环烷基,(C 3 -C 6) - 烯基,(C 2 -C 1 -C 6)炔基,(C 1 -C 3) - 卤代烷基,(C 2 -C 6) - 烷氧基,(C 1 -C 6) - 烷氧基 - (C 1 -C 6) - 烷基,氰基,取代酰胺,(C 1 -C 6) 羰基,未取代或具有1至2个取代基的苯甲酰基,未取代或具有1至2个取代基的苯甲酰基氨基; (C 2 -C 6) - 烷酰基氨基,(C 3 -C 6) - 环烷基羰基氨基,未被取代或具有1至2个取代基的苄基,未取代或具有1至2个取代基的苯基,或(C 1 -C 6) - 烷氧基羰基 - (C 2 -C 6) C5) - 亚烯基; 并且R1和R2不同时都表示氢。 含有二甲基呋喃羧酰苯胺化合物作为活性成分的木材防腐剂。 一种通过将二甲基呋喃羧酰苯胺化合物施用于木材来保存木材的方法。 一种木材防腐剂组合物,其中二甲基呋喃羧酰苯胺化合物与3-溴-2,3-二碘-2-丙烯基乙基氨基甲酸酯,3-碘-2-丙炔基丁基氨基甲酸酯和4-氯苯基-3-碘代炔丙基甲酰胺中的至少一种组合。

    Dimethylfurancarboxyanilide derivatives

    公开(公告)号:US06506913B2

    公开(公告)日:2003-01-14

    申请号:US10040138

    申请日:2001-10-24

    IPC分类号: C07D30768

    CPC分类号: A01N43/08 B27K3/343

    摘要: A dimethylfurancarboxyanilide compound of the formula (I): wherein R1 and R2 are the same or different and each is hydrogen, (C2-C6)-alkyl, (C3-C6)-cycloalkyl, (C3-C6)-alkenyl, (C2-C6) alkynyl, (C1-C3)-halogenoalkyl, (C2-C6)-alkoxy, (C1-C6)-alkoxy-(C1-C6)-alkyl, cyano, substituted amide, (C1-C6)-alkoxy-carbonyl, benzoyl which is unsubstituted or has 1 to 2 substituents, benzoylamino which is unsubstituted or has 1 to 2 substituents; (C2-C6)-alkanoylamino, (C3-C6)-cycloalkylcarbonylamino, benzyl which is unsubstituted or has 1 to 2 substituents, phenyl which is unsubstituted or has 1 to 2 substituents, or (C1-C6)-alkoxycarbonyl-(C2-C5)-alkenylene; and R1 and R2 do not both represent hydrogen at the same time. A wood preservative containing the dimethylfurancarboxyanilide compound as an active ingredient. A method of preserving wood by applying the dimethylfurancarboxyanilide compound to wood. A wood preservative composition in which the dimethylfurancarboxyanilide compound is combined with at least one of 3-bromo-2,3-diiodo-2-propenylethylcarbamate, 3-iodo-2-propynylbutylcarbamate and 4-chlorophenyl-3-iodopropargylformal.

    Dimethylfurancarboxyanilide derivatives
    3.
    发明授权
    Dimethylfurancarboxyanilide derivatives 失效
    二甲基呋喃羧酰苯胺衍生物

    公开(公告)号:US06380247B2

    公开(公告)日:2002-04-30

    申请号:US09729546

    申请日:2000-12-04

    IPC分类号: A61K3134

    CPC分类号: A01N43/08 B27K3/343

    摘要: A dimethylfurancarboxyanilide compound of the formula (I): wherein R1 and R2 are the same or different and each is hydrogen, (C2-C6)-alkyl, (C3-C6)-cycloalkyl, (C3-C6)-alkenyl, (C2-C6) alkynyl, (C1-C3)-halogenoalkyl, (C2-C6)-alkoxy, (C1-C6)-alkoxy-(C1-C6)-alkyl, cyano, substituted amide, (C1-C6)-alkoxy-carbonyl, benzoyl which is unsubstituted or has 1 to 2 substituents, benzoylamino which is unsubstituted or has 1 to 2 substituents; (C2-C6)-alkanoylamino, (C3-C6)-cycloalkylcarbonylamino, benzyl which is unsubstituted or has 1 to 2 substituents, phenyl which is unsubstituted or has 1 to 2 substituents, or (C1-C6)-alkoxycarbonyl-(C2-C5)-alkenylene; and R1 and R2 do not both represent hydrogen at the same time. A wood preservative containing the dimethylfurancarboxyanilide compound as an active ingredient. A method of preserving wood by applying the dimethylfurancarboxyanilide compound to wood. A wood preservative composition in which the dimethylfurancarboxyanilide compound is combined with at least one of 3-bromo-2,3-diiodo-2-propenylethylcarbamate, 3-iodo-2-propynylbutylcarbamate and 4-chlorophenyl-3-iodopropargylformal.

    摘要翻译: 式(I)的二甲基呋喃羧酰苯胺化合物:其中R 1和R 2相同或不同,各自为氢,(C 2 -C 6) - 烷基,(C 3 -C 6) - 环烷基,(C 3 -C 6) - 烯基,(C 2 -C 1 -C 6)炔基,(C 1 -C 3) - 卤代烷基,(C 2 -C 6) - 烷氧基,(C 1 -C 6) - 烷氧基 - (C 1 -C 6) - 烷基,氰基,取代酰胺,(C 1 -C 6) 羰基,未取代或具有1至2个取代基的苯甲酰基,未取代或具有1至2个取代基的苯甲酰基氨基; (C 2 -C 6) - 烷酰基氨基,(C 3 -C 6) - 环烷基羰基氨基,未被取代或具有1至2个取代基的苄基,未取代或具有1至2个取代基的苯基或(C 1 -C 6) - 烷氧基羰基 - (C 2 -C 6) C5) - 亚烯基; 并且R1和R2不同时都表示氢。 含有二甲基呋喃羧酰苯胺化合物作为活性成分的木材防腐剂。 一种通过将二甲基呋喃羧酰苯胺化合物施用于木材来保存木材的方法。 一种木材防腐剂组合物,其中二甲基呋喃羧酰苯胺化合物与3-溴-2,3-二碘-2-丙烯基乙基氨基甲酸酯,3-碘-2-丙炔基丁基氨基甲酸酯和4-氯苯基-3-碘代炔丙基甲酰胺中的至少一种组合。

    Macrolide compounds, their preparation and their use
    7.
    发明授权
    Macrolide compounds, their preparation and their use 失效
    大环内酯类化合物,其制备及其用途

    公开(公告)号:US5212322A

    公开(公告)日:1993-05-18

    申请号:US644100

    申请日:1991-01-22

    IPC分类号: A01N49/00 C07H19/01 C12P17/18

    摘要: Compounds with acaricidal, insecticidal and anthelmintic activities have the formula: ##STR1## wherein: --X--Y-- is selected from the group consisting of --CH.sub.2 --CH.sub.2 --, --CH.sub.2 --CHOH--, --CH.dbd.CH--, and --CH.sub.2 --C(.dbd.O)--;R.sup.1 is selected from the group consisting of a methyl group, an ethyl group, an isopropyl group, a sec-butyl group and groups of formula --C(CH.sub.3).dbd.CHR.sup.5 in which R.sup.5 is selected from the group consisting of a methyl group, an ethyl group and an isopropyl group;R.sup.2 represents a group of formula --(CH.sub.2).sub.n --C(R.sup.6).dbd.C(R.sup.7)(R.sup.8) in which n is 0, 1 or 2, R.sup.6 and R.sup.7 each is selected from the group consisting of a hydrogen atom and a methyl group and R.sup.8 is selected from the group consisting of a hydrogen atom, a C.sub.1-4 alkyl group, a phenyl group and a phenyl group substituted with at least one substituent selected from the group consisting of halogen, methyl and nitro substituents;R.sup.3 is selected from the group consisting of a hydrogen atom, a methyl group, a hydroxy-protecting group, an ester-forming carboxylic acid residue, and an ester-forming carbonic acid residue; andR.sup.4 is selected from the group consisting of a hydrogen atom and an .alpha.-L-oleandrosyl-.alpha.-L-oleandrosyloxy group, with the proviso that R.sup.4 represents a hydrogen atom when the group R.sup.1 is selected from the group consisting of a methyl group, an ethyl group, and groups of formula --C(CH.sub.3).dbd.CHR.sup.5 in which R.sup.5 is selected from the group consisting of a methyl group, an ethyl group and an isopropyl group.

    摘要翻译: 具有杀螨,杀虫和驱虫活性的化合物具有下式:其中:-XY-选自-CH 2 -CH 2 - , - CH 2 -CHOH - , - CH = CH-和 - CH2-C(= O) - ; R 1选自甲基,乙基,异丙基,仲丁基和式-C(CH 3)= CHR 5的基团,其中R 5选自甲基, 乙基和异丙基; R 2表示式 - (CH 2)n C(R 6)= C(R 7)(R 8)的基团,其中n为0,1或2,R 6和R 7各自为氢原子和甲基 并且R 8选自氢原子,C 1-4烷基,苯基和被至少一个选自卤素,甲基和硝基取代基的取代基取代的苯基; R3选自氢原子,甲基,羟基保护基,成酯羧酸残基和形成酯的碳酸残基; 并且R 4选自氢原子和α-L-甘氨酰基-α-L-胆碱基氧基,条件是当R 1选自甲基时,R 4表示氢原子 ,乙基和式-C(CH 3)= CHR 5基团,其中R 5选自甲基,乙基和异丙基。