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    Fungicides based on nitrogen-containing heterocycles
    1.
    发明申请
    Fungicides based on nitrogen-containing heterocycles 审中-公开

    公开(公告)号：US20060100203A1

    公开(公告)日：2006-05-11

    申请号：US10540039

    申请日：2003-12-03

    申请人： Patrick Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    发明人： Patrick Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    IPC分类号： A01N43/90 ,  A01N43/42

    CPC分类号： C07D471/04

    摘要： Fungicidal compounds having the general formula (1): formula (1) wherein W, Z and one of X and Y are N and the other one of X and Y is CR8; R8 is H, halo, C1-4alkyl, C1-4alkoxy, C1-4alkylthio or halo(C1-4)alkyl; R and R2 are independently H, halo, C1-8 alkyl, C1-8 alkoxy, C1-8 alkylthio, C2-8alkenyl, C2-8 alkynyl, cyano or NR3R4, provided that at least one of R and R2 is NR3R4; R1 is halo, C1-8 alkyl, C2-8 alkenyl, C2-8alkynyl, C3-8 cycloalkyl, C3-8 cycloalkyl(C1-6)-alkyl, C1-8 alkoxy, C1-8 alkylthio, aryl, aryloxy, arylthio, heteroaryl, heteroaryloxy, heteroarylthio, aryl(C1-4)alkyl, aryl(C1-4)alkoxy, heteroaryl(C1-4)alkyl, heteroaryl(C1-4)alkoxy, aryl(C1-4)alkylthio, heteroaryl(C1-4)alkylthio, morpholino, piperidino or pyrrolidino; R3 and R4 are independently H, C1-8 alkyl, C2-8 alkenyl, C2-8 alkynyl, aryl, aryl(C1-8)-alkyl, C3-8cycloalkyl, C3-8 cycloalkyl(C1-6)alkyl, heteroaryl, heteroaryl(C1-8)alkyl, NR5R6, provided that not both R3 and R4 are H or NR5R6, or R3 and R4 together form a C3-7 alkylene or C3-7 alkenylene chain optionally substituted with one or more C1-4 alkyl or C1-4 alkoxy groups, or, together with the nitrogen atom to which they are attached, R3 and R4 form a morpholine, thiomorpholine, thiomorpholine S-oxide or thiomorpholine S-dioxide ring or a piperazine or piperazine N-(C1-4)alkyl (especially N-methyl) ring; and R5 and R6 are independently H, C1-8 alkyl, C2-8 alkenyl, C2-8-alkynyl, aryl, aryl(C1-8)alkyl, C3-8 cycloalkyl, C3-8 cycloalkyl(C1-6)alkyl, heteroaryl or heteroaryl(C1-8)alkyl; any of the foregoing alkyl, alkenyl, alkynyl or cycloalkyl groups or moieties (other than for R8) being optionally substituted with halogen, cyano, C1-6 alkoxy, C1-6alkylcarbonyl, C1-6 alkoxycarbonyl, C1-6 haloalkoxy, C1-6 alkylthio, tri(C1-4)alkylsilyl, C1-6 alkylamino or C1-6 dialkylamino, any of the foregoing morpholine, thiomopholine, piperidine, piperazine and pyrrolidine rings being optionally substituted with C1-4 alkyl (especially methyl), and any of the foregoing aryl or heteroaryl groups or moieties being optionally substituted with one or more substituents selected from halo, hydroxy, mercapto, C1-6alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-6 alkoxy, C2-6 alkenyloxy, C2-6 alkynyloxy, halo(C1-6)alkyl, halo(C1-6)alkoxy, C1-6 alkylthio, halo(C1-6)alkylthio, hydroxy(C1-6)alkyl, C1-4 alkoxy(C1-6)alkyl, C3-6 cycloalkyl, C3-6cycloalkyl(C1-4)alkyl, phenoxy, benzyloxy, benzoyloxy, cyano, isocyano, thiocyanato, isothiocyanato, nitro, —NR″′R″″, NHCOR″′, —NHCONR″′R″″, —CONR″′R″″, —SO2R″′, —OSO2R″′, —COR″′, —CR″′═NR″″ or —N═CR ″′R″″, in which R″′ and R″″ are independently hydrogen, C1-4 alkyl, halo(C1-4)alkyl, C1-4 alkoxy, halo(C1-4)alkoxy, C1-4 alkylthio, C3-6 cycloalkyl, C3-6 cycloalkyl(C1-4)alkyl, phenyl or benzyl, the phenyl and benzyl groups being optionally substituted with halogen, C1-4 alkyl or C1-4 alkoxy.

    Fungicides
    2.
    发明申请
    Fungicides 失效

    公开(公告)号：US20060069089A1

    公开(公告)日：2006-03-30

    申请号：US10540037

    申请日：2003-12-03

    申请人： Patrick Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    发明人： Patrick Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    IPC分类号： C07D471/02 ,  A01N43/42

    CPC分类号： C07D471/04 ,  A01N43/90

    摘要： Fungicidal compositions of the general formula (1): wherein one of W, X, Y and Z is N and the others are CR8; R8 is H, halo, C1-4 alkyl, C1-4 alkoxy or halo(C1-4)alkyl, provided that when X is CH, Z is N, R is NHNH2, R1 is phenyl and R2 is Cl, W and Y are not both CCH3; one of R and R2 is NR3R4 and the other is halo, C1-8 alkyl, C1-8 alkoxy, C1-8 alkylthio, C2-8 alkenyl, C2-8 alkynyl or cyano; R1 is aryl, heteroaryl, morpholino, piperidino or pyrrolidino; R3 and R4 are independently H, C1-8 alkyl, C2-8 alkenyl, C2-8 alkynyl, aryl, aryl(C1-8)-alkyl, C3-8 cycloalkyl, C3-8 cycloalkyl(C1-6)alkyl, heteroaryl, heteroaryl(C1-8)alkyl, NR5R6, provided that not v both R3 and R4 are H or NR5R6, or R3 and R4 together form a C3-7 alkylene or C3-7 alkenylene chain optionally substituted with one or more C1-4 alkyl or C1-4 alkoxy groups, or, together with the nitrogen atom to which they are attached, R3 and R4 form a morpholine, thiomorpholine, thiomorpholine S-oxide or thiomorpholine S-dioxide ring or a piperazine or piperazine N—(C1-4)alkyl (especially N-methyl) ring; and R5 and R6 are independently H, C1-8 alkyl, C2-8 alkenyl, C2-8 alkynyl, aryl, aryl(C1-8)-alkyl, C3-8 cycloalkyl, C3-8 cycloalkyl(C1-6)alkyl, heteroaryl or heteroaryl(C1-8)alkyl; any of the foregoing alkyl, alkenyl, alkynyl or cycloalkyl groups or moieties (other than for R8) being optionally substituted with halogen, cyano, C1-8 alkoxy C1-4 alkylcarbonyl, C1-6 alkoxycarbonyl, C1-6 haloalkoxy, C1-6 alkylthio, tri(C1-4)alkylsilyl, C1-6 alkylamino or C1-6 alkylamino, any of the foregoing morpholine, thiomorpholine, piperidine, piperazine and pyrrolidine rings being optionally substituted with C1-4 alkyl (especially methyl), and any of the foregoing aryl or heteroaryl groups or moieties being optionally substituted with one or more substituents selected from halo, hydroxy, mercapto, C1-4 alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-6 alkoxy, C2-6 alkenyloxy, C2-6 alkynyloxy, halo(C1-4)alkyl, halo(C1-6)alkoxy, C1-6 alkylthio, halo(C1-4)alkylthio, hydroxy(C1-6)alkyl, C1-4 alkoxy(C1-6)alkyl, C1-6 cycloalkyl, C3-4 cycloalkyl(C1-4)alkyl, phenoxy, benzyloxy, benzoyloxy, cyano, isocyano, thiocyanato, isothiocyanato, nitro, —NHCOR″′, —NHCONR″′ R″″, —CONK″′R″″, SO2R″′, —OSO2R″′, —COR″′, —CR″′═NR″ or —N═CR″′R″″, in which R″′ and R″″ are independently hydrogen, C1-4 alkyl, halo-(C1-4)alkyl, C1-4 alkoxy, halo(C1-4)alkoxy, C1-4 alkylthio, C3-4 cycloalkyl, C3-6 cycloalkyl(C1-4)alkyl, phenyl or benzyl groups beings optionally substituted with halogen, C1-4 alkyl or C1-4 alkoxy.

    Fungicides
    3.
    发明申请
    Fungicides 审中-公开
    杀菌剂

    公开(公告)号：US20070066605A1

    公开(公告)日：2007-03-22

    申请号：US10540040

    申请日：2003-12-04

    申请人： Patrick Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    发明人： Patrick Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    IPC分类号： C07D487/02 ,  A01N43/90

    CPC分类号： C07D239/42 ,  A01N43/90 ,  C07D471/04

    摘要： Fungicidal compositions having the general formula (1): formula (1) wherein W and Y are both N and X and Z are both CR8 or X and Z are both N and W and Y are both C6, R8 is H, halo, C1-4 alkyl, C1-4alkoxy or halo(C1-4)alkyl; R and R2 are independently H, halo, C1-8alkyl, C1-8alkoxy, C1-8alkylthio, C2-8alkenyl, C2-8 alkynyl, cyano or NR3R4, provided that at least one of R and R2 is NR3R4; R1 is halo, C1-8alkyl, C2-8alkenyl, C2-8alkynyl, C3-8cycloalkyl, C3-8cycloalkyl(C1-6)-alkyl, C1-8alkoxy, C1-8 alkylthio, aryl, aryloxy, arylthio, heteroaryl, heteroaryloxy, heteroarylthio, aryl(C1-4)alkyl, aryl(CI4,)alkoxy, heteroaryl(C1-4)alkyl, heteroaryl(C1-4)alkoxy, aryl(C1-4)alkylthio, heteroaryl(C1-4)alkylthiio, morpholiiio, piperidino or pynrolidino.

    摘要翻译： 具有通式（1）：式（1）的杀真菌组合物，其中W和Y都是N，X和Z都是CR 8或X和Z都是N，W和Y都是C R 8是H，卤素，C 1-4烷基，C 1-4烷氧基或卤代 （C 1-4烷基）烷基; R和R 2独立地为H，卤素，C 1-8烷基，C 1-8烷氧基，C 1-8 C 2〜C 8烷基，C 2-8链烯基，C 2-8炔基，氰基或NR 3 R 4， SUP>，条件是R和R 2中的至少一个是NR 3 R 4; R 1是卤素，C 1-8烷基，C 2-8链烯基，C 2-8炔基 C 3-8环烷基，C 3-8环烷基（C 1-6 - ） - 烷基，C 1-8 - C 1-4烷基，芳基，芳氧基，芳硫基，杂芳基，杂芳氧基，杂芳硫基，芳基（C 1-4 - ）烷基，芳基（C 1-4， ）烷氧基，杂芳基（C 1-4 - ）烷基，杂芳基（C 1-4 - ）烷氧基，芳基（C 1-4 - ）烷硫基 ，杂芳基（C 1-4烷基）硫代，吗啉代，哌啶子基或鸟嘌呤基。

    FUNGICIDES
    6.
    发明申请
    FUNGICIDES 审中-公开
    杀真菌剂

    公开(公告)号：US20090069333A1

    公开(公告)日：2009-03-12

    申请号：US12187072

    申请日：2008-08-06

    申请人： Patrick Jelf Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    发明人： Patrick Jelf Crowley ,  Markus Dobler ,  Urs Mueller ,  John Williams

    IPC分类号： A01N43/58 ,  C07D471/04 ,  A01P3/00 ,  A01N43/60

    CPC分类号： C07D471/04

    摘要： This invention relates to novel derivatives of pyridopyrazines and pyridopyridazines, to processes for preparing them, to intermediate chemicals used in their manufacture, to compositions containing them and to methods of using them to combat fungi, especially fungal infections of plants. The fungicidal compounds have the general formula (1) wherein R, R1, R2, W, X Y and Z are defined in the specification

    摘要翻译： 本发明涉及吡啶并吡嗪和吡啶并哒嗪的新衍生物，其制备方法，制备中使用的中间体化学品，含有它们的组合物以及使用它们来对抗真菌，特别是植物真菌感染的方法。 杀真菌化合物具有通式（1），其中R，R 1，R 2，W，X Y和Z在本说明书中定义