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公开(公告)号:US20080318962A1
公开(公告)日:2008-12-25
申请号:US11570980
申请日:2005-06-21
申请人: Patrick Jelf Crowley , Urs Muller , Markus Dobler , John Williams
发明人: Patrick Jelf Crowley , Urs Muller , Markus Dobler , John Williams
IPC分类号: A01N43/90 , C07D471/04 , A01P3/00
CPC分类号: C07D471/04 , A01N43/90
摘要: The compound of the general formula (I), wherein W, X, Y, Z, R, R1 and R2 are defined as set forth in the specification, useful as fungicide.
摘要翻译: 通式(I)的化合物,其中W,X,Y,Z,R,R 1和R 2定义如说明书中所述,可用作杀真菌剂。
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公开(公告)号:US20080280766A1
公开(公告)日:2008-11-13
申请号:US11570984
申请日:2005-06-21
申请人: Patrick Jelf Crowley , Urs Muller , Markus Dobler , John Williams
发明人: Patrick Jelf Crowley , Urs Muller , Markus Dobler , John Williams
IPC分类号: A01N43/90 , C07D471/04 , A01P3/00
CPC分类号: C07D471/04
摘要: The compounds of the general formula (I) wherein R, R1, R2, R8, and R9 are defined as set forth in the specification.
摘要翻译: 通式(I)的化合物,其中R 1,R 1,R 2,R 8和R 9, SUP>被定义为说明书中阐述的。
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公开(公告)号:US07947679B2
公开(公告)日:2011-05-24
申请号:US10540037
申请日:2003-12-03
IPC分类号: A61K31/44 , A61K31/535 , C07D471/02
CPC分类号: C07D471/04 , A01N43/90
摘要: The naphthyridine derivatives of formula (I) a and method of combating or controlling phytopathogenic fungi which comprises applying the compounds of formula (I) to a plant, to a seed of a plant and to the locus of the plant.
摘要翻译: 式(I)的萘啶衍生物a和防治植物病原真菌的方法,其包括将式(I)化合物施用于植物,植物种子和植物地点。
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公开(公告)号:US20090069333A1
公开(公告)日:2009-03-12
申请号:US12187072
申请日:2008-08-06
IPC分类号: A01N43/58 , C07D471/04 , A01P3/00 , A01N43/60
CPC分类号: C07D471/04
摘要: This invention relates to novel derivatives of pyridopyrazines and pyridopyridazines, to processes for preparing them, to intermediate chemicals used in their manufacture, to compositions containing them and to methods of using them to combat fungi, especially fungal infections of plants. The fungicidal compounds have the general formula (1) wherein R, R1, R2, W, X Y and Z are defined in the specification
摘要翻译: 本发明涉及吡啶并吡嗪和吡啶并哒嗪的新衍生物,其制备方法,制备中使用的中间体化学品,含有它们的组合物以及使用它们来对抗真菌,特别是植物真菌感染的方法。 杀真菌化合物具有通式(1),其中R,R 1,R 2,W,X Y和Z在本说明书中定义
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公开(公告)号:US07410967B2
公开(公告)日:2008-08-12
申请号:US10540035
申请日:2003-12-03
IPC分类号: C07D487/04 , A61K31/519
CPC分类号: C07D471/04
摘要: Fungicidal compounds of general formula (1) wherein R, R1, R2, W, X, Y and Z are as defined in the specification
摘要翻译: 其中R,R 1,R 2,W,X,Y和Z的通式(1)的杀真菌化合物如本说明书中所定义
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公开(公告)号:US06544989B2
公开(公告)日:2003-04-08
申请号:US09767880
申请日:2001-01-23
申请人: Christopher John Mathews , Russell Viner , Susan Patricia Barnett , Christopher John Urch , Stephen Christopher Smith , Patrick Jelf Crowley , William Guy Whittingham , Stephen Paul Heaney , John Williams , Torquil Eoghan Macleod Fraser , Eric Daniel Clarke , David John Hughes , Sarah Armstrong , Nigel John Barnes , Alan John Whittle , Brian Leslie Pilkington
发明人: Christopher John Mathews , Russell Viner , Susan Patricia Barnett , Christopher John Urch , Stephen Christopher Smith , Patrick Jelf Crowley , William Guy Whittingham , Stephen Paul Heaney , John Williams , Torquil Eoghan Macleod Fraser , Eric Daniel Clarke , David John Hughes , Sarah Armstrong , Nigel John Barnes , Alan John Whittle , Brian Leslie Pilkington
IPC分类号: C07D41712
CPC分类号: C07D417/12 , A01N43/80
摘要: The invention provides compounds of formula (I): where the substituents are as defined in the specification. The invention also provides processes for preparing the compounds, compositions comprising the compounds, methods of using the compounds and compositions to combat fungal diseases, and methods of using the compounds and compositions to combat or control insect, acarine, mollusc and nematode pests.
摘要翻译: 本发明提供式(I)化合物:其中取代基如说明书中所定义。 本发明还提供了制备化合物的方法,包含化合物的组合物,使用化合物和组合物来对抗真菌疾病的方法,以及使用化合物和组合物来对抗或控制昆虫,螨虫,软体动物和线虫的害虫的方法。
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公开(公告)号:US06703347B2
公开(公告)日:2004-03-09
申请号:US10182425
申请日:2002-11-07
申请人: Sarah Armstrong , Nigel John Barnes , Susan Patricia Barnett , Eric Daniel Clarke , Patrick Jelf Crowley , Torquil Eoghan Macleod Fraser , David John Hughes , Christopher John Mathews , Roger Salmon , Stephen Christopher Smith , Russell Viner , William Guy Whittingham , John Williams , Alan John Whittle , William Roderick Mound , Christopher John Urch , Brian Leslie Pilkington
发明人: Sarah Armstrong , Nigel John Barnes , Susan Patricia Barnett , Eric Daniel Clarke , Patrick Jelf Crowley , Torquil Eoghan Macleod Fraser , David John Hughes , Christopher John Mathews , Roger Salmon , Stephen Christopher Smith , Russell Viner , William Guy Whittingham , John Williams , Alan John Whittle , William Roderick Mound , Christopher John Urch , Brian Leslie Pilkington
IPC分类号: C07D41712
CPC分类号: C07D417/12 , A01N43/80
摘要: A compound of formula (I), where A is optionally substituted alkylene, alkenylene, alkynylene, cycloalkylene, alkylenoxy, oxy(C1-6)alkylene, alkylenthio, thio(C1-6)alkylene, C1-6alkylenamino, amino(C1-6)alkylene, [C1-6alkyleneoxy(C1-6)alkylene], [C1-6alkylenethio(C1-6)alkylene], [1-6alkylenesulfinyl(C1-6)alkylene], [C1-6alkylenesulfonyl(C1-6)alkylene] or [C1-6alkyleneamino(C1-6)alkylene]; provided that A is not CH2 or CH2O; B is N,N-oxide or CR8; Y is O, S or NR9; Z is O, S or NR10; and R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 are specified radicals; compositions containing them; process for making them; and their use as insecticides or fungicides.
摘要翻译: 式(I)化合物,其中A为任选取代的亚烷基,亚烯基,亚炔基,亚环烷基,亚烷氧基,氧(C 1-6)亚烷基,烷基硫基,硫代(C 1-6)亚烷基,C 1-6亚烷基氨基,氨基(C 1-6) )亚烷基,[C 1-6亚烷基氧基(C 1-6)亚烷基],[C 1-6亚烷基硫醚(C 1-6)亚烷基],[1-6亚烷基亚烷基(C 1-6)亚烷基] 或[C 1-6亚烷基氨基(C 1-6)亚烷基]; A不是CH2或CH2O; B是N,N-氧化物或CR 8; Y是O,S或NR 9; Z是O,S或NR 10; R 1,R 2,R 3,R 4,R 5,R 6,R 7,R 8,R 9,R 10, 被指定为自由基; 含有它们的组合物; 制作过程; 并将其用作杀虫剂或杀真菌剂。
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公开(公告)号:US5830890A
公开(公告)日:1998-11-03
申请号:US723795
申请日:1996-09-30
IPC分类号: C07D215/22 , A01N43/36 , A01N43/40 , A01N43/42 , A01N43/72 , A01N43/76 , A01N43/84 , C07D211/74 , C07D211/86 , C07D211/88 , C07D215/227 , C07D265/30 , C07D265/32 , C07D265/36 , C07D267/10 , C07D267/14 , C07D279/12 , C07D279/16 , C07D265/34
CPC分类号: C07D215/227 , A01N43/36 , A01N43/42 , A01N43/72 , A01N43/76 , A01N43/84 , C07D211/74 , C07D211/86 , C07D265/32 , C07D265/36 , C07D267/14 , C07D279/16
摘要: Compounds, useful as plant fungicides, having the formula (I): ##STR1## or a stereoisomer thereof, wherein A is CH or N, B is OCH.sub.3 or NHCH.sub.3, X is CH.sub.2, CH.sub.2 O, O or S, Y is R.sup.1 --C.dbd.C--R.sup.2 or R.sup.1 --CH--CH--R.sup.2 wherein R.sup.1 and R.sup.2 are independently H, halo, hydroxy, alkyl, haloalkyl, alkoxy, haloalkoxy, cyano, nitro, amino, mono- or dialkylamino, alkanoylamino, carboxy, alkoxycarbonyl, aminocarbonyl, mono- or di-alkylaminocarbonyl, alkylcarbonyloxy, optionally substituted aryl, optionally substituted aralkyl or optionally substituted aryloxy or R.sup.1 and R.sup.2 join to form with the carbon atoms to which they are attached an optionally substituted benzene ring, and Z is CH.sub.2, CHCH.sub.3, C(CH.sub.3).sub.2 or C.dbd.O.
摘要翻译: 可用作植物杀真菌剂的化合物,其具有式(I):其中A是CH或N,B是OCH 3或NHCH 3,X是CH 2,CH 2 O,O或S,Y是 R1-C = C-R2或R1-CH-CH-R2其中R1和R2独立地为H,卤素,羟基,烷基,卤代烷基,烷氧基,卤代烷氧基,氰基,硝基,氨基,单或二烷基氨基,烷酰氨基,羧基, 烷氧基羰基,氨基羰基,单 - 或二 - 烷基氨基羰基,烷基羰基氧基,任选取代的芳基,任选取代的芳烷基或任选取代的芳氧基或R 1和R 2与它们所连接的碳原子形成任选取代的苯环,Z是CH 2 CHCH 3,C(CH 3)2或C = O。
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公开(公告)号:US20070066605A1
公开(公告)日:2007-03-22
申请号:US10540040
申请日:2003-12-04
申请人: Patrick Crowley , Markus Dobler , Urs Mueller , John Williams
发明人: Patrick Crowley , Markus Dobler , Urs Mueller , John Williams
IPC分类号: C07D487/02 , A01N43/90
CPC分类号: C07D239/42 , A01N43/90 , C07D471/04
摘要: Fungicidal compositions having the general formula (1): formula (1) wherein W and Y are both N and X and Z are both CR8 or X and Z are both N and W and Y are both C6, R8 is H, halo, C1-4 alkyl, C1-4alkoxy or halo(C1-4)alkyl; R and R2 are independently H, halo, C1-8alkyl, C1-8alkoxy, C1-8alkylthio, C2-8alkenyl, C2-8 alkynyl, cyano or NR3R4, provided that at least one of R and R2 is NR3R4; R1 is halo, C1-8alkyl, C2-8alkenyl, C2-8alkynyl, C3-8cycloalkyl, C3-8cycloalkyl(C1-6)-alkyl, C1-8alkoxy, C1-8 alkylthio, aryl, aryloxy, arylthio, heteroaryl, heteroaryloxy, heteroarylthio, aryl(C1-4)alkyl, aryl(CI4,)alkoxy, heteroaryl(C1-4)alkyl, heteroaryl(C1-4)alkoxy, aryl(C1-4)alkylthio, heteroaryl(C1-4)alkylthiio, morpholiiio, piperidino or pynrolidino.
摘要翻译: 具有通式(1):式(1)的杀真菌组合物,其中W和Y都是N,X和Z都是CR 8或X和Z都是N,W和Y都是C R 8是H,卤素,C 1-4烷基,C 1-4烷氧基或卤代 (C 1-4烷基)烷基; R和R 2独立地为H,卤素,C 1-8烷基,C 1-8烷氧基,C 1-8 C 2〜C 8烷基,C 2-8链烯基,C 2-8炔基,氰基或NR 3 R 4, SUP>,条件是R和R 2中的至少一个是NR 3 R 4; R 1是卤素,C 1-8烷基,C 2-8链烯基,C 2-8炔基 C 3-8环烷基,C 3-8环烷基(C 1-6 - ) - 烷基,C 1-8 - C 1-4烷基,芳基,芳氧基,芳硫基,杂芳基,杂芳氧基,杂芳硫基,芳基(C 1-4 - )烷基,芳基(C 1-4, )烷氧基,杂芳基(C 1-4 - )烷基,杂芳基(C 1-4 - )烷氧基,芳基(C 1-4 - )烷硫基 ,杂芳基(C 1-4烷基)硫代,吗啉代,哌啶子基或鸟嘌呤基。
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公开(公告)号:US20060100203A1
公开(公告)日:2006-05-11
申请号:US10540039
申请日:2003-12-03
申请人: Patrick Crowley , Markus Dobler , Urs Mueller , John Williams
发明人: Patrick Crowley , Markus Dobler , Urs Mueller , John Williams
CPC分类号: C07D471/04
摘要: Fungicidal compounds having the general formula (1): formula (1) wherein W, Z and one of X and Y are N and the other one of X and Y is CR8; R8 is H, halo, C1-4alkyl, C1-4alkoxy, C1-4alkylthio or halo(C1-4)alkyl; R and R2 are independently H, halo, C1-8 alkyl, C1-8 alkoxy, C1-8 alkylthio, C2-8alkenyl, C2-8 alkynyl, cyano or NR3R4, provided that at least one of R and R2 is NR3R4; R1 is halo, C1-8 alkyl, C2-8 alkenyl, C2-8alkynyl, C3-8 cycloalkyl, C3-8 cycloalkyl(C1-6)-alkyl, C1-8 alkoxy, C1-8 alkylthio, aryl, aryloxy, arylthio, heteroaryl, heteroaryloxy, heteroarylthio, aryl(C1-4)alkyl, aryl(C1-4)alkoxy, heteroaryl(C1-4)alkyl, heteroaryl(C1-4)alkoxy, aryl(C1-4)alkylthio, heteroaryl(C1-4)alkylthio, morpholino, piperidino or pyrrolidino; R3 and R4 are independently H, C1-8 alkyl, C2-8 alkenyl, C2-8 alkynyl, aryl, aryl(C1-8)-alkyl, C3-8cycloalkyl, C3-8 cycloalkyl(C1-6)alkyl, heteroaryl, heteroaryl(C1-8)alkyl, NR5R6, provided that not both R3 and R4 are H or NR5R6, or R3 and R4 together form a C3-7 alkylene or C3-7 alkenylene chain optionally substituted with one or more C1-4 alkyl or C1-4 alkoxy groups, or, together with the nitrogen atom to which they are attached, R3 and R4 form a morpholine, thiomorpholine, thiomorpholine S-oxide or thiomorpholine S-dioxide ring or a piperazine or piperazine N-(C1-4)alkyl (especially N-methyl) ring; and R5 and R6 are independently H, C1-8 alkyl, C2-8 alkenyl, C2-8-alkynyl, aryl, aryl(C1-8)alkyl, C3-8 cycloalkyl, C3-8 cycloalkyl(C1-6)alkyl, heteroaryl or heteroaryl(C1-8)alkyl; any of the foregoing alkyl, alkenyl, alkynyl or cycloalkyl groups or moieties (other than for R8) being optionally substituted with halogen, cyano, C1-6 alkoxy, C1-6alkylcarbonyl, C1-6 alkoxycarbonyl, C1-6 haloalkoxy, C1-6 alkylthio, tri(C1-4)alkylsilyl, C1-6 alkylamino or C1-6 dialkylamino, any of the foregoing morpholine, thiomopholine, piperidine, piperazine and pyrrolidine rings being optionally substituted with C1-4 alkyl (especially methyl), and any of the foregoing aryl or heteroaryl groups or moieties being optionally substituted with one or more substituents selected from halo, hydroxy, mercapto, C1-6alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-6 alkoxy, C2-6 alkenyloxy, C2-6 alkynyloxy, halo(C1-6)alkyl, halo(C1-6)alkoxy, C1-6 alkylthio, halo(C1-6)alkylthio, hydroxy(C1-6)alkyl, C1-4 alkoxy(C1-6)alkyl, C3-6 cycloalkyl, C3-6cycloalkyl(C1-4)alkyl, phenoxy, benzyloxy, benzoyloxy, cyano, isocyano, thiocyanato, isothiocyanato, nitro, —NR″′R″″, NHCOR″′, —NHCONR″′R″″, —CONR″′R″″, —SO2R″′, —OSO2R″′, —COR″′, —CR″′═NR″″ or —N═CR ″′R″″, in which R″′ and R″″ are independently hydrogen, C1-4 alkyl, halo(C1-4)alkyl, C1-4 alkoxy, halo(C1-4)alkoxy, C1-4 alkylthio, C3-6 cycloalkyl, C3-6 cycloalkyl(C1-4)alkyl, phenyl or benzyl, the phenyl and benzyl groups being optionally substituted with halogen, C1-4 alkyl or C1-4 alkoxy.
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