公开(公告)号：US4005217A

公开(公告)日：1977-01-25

申请号：US153407

申请日：1971-06-15

申请人： Samuel Sidney Berg ,  David Conwil Jenkins ,  George Christopher James Martin ,  Ronald Frederick Phillipson ,  Garth Molesdale Thompson

发明人： Samuel Sidney Berg ,  David Conwil Jenkins ,  George Christopher James Martin ,  Ronald Frederick Phillipson ,  Garth Molesdale Thompson

IPC分类号： C07C335/28 ,  C07D295/14 ,  A61K31/27

CPC分类号： C07D295/14 ,  C07C335/28

摘要： Benzene derivatives of the formula:- ##STR1## wherein R is an aliphatic hydrocarbon group of 1 to 4 carbon atoms optionally substituted by halogen or alkoxy, R.sup.1 is hydrogen or methyl, R.sup.2 is hydrogen, halogen, alkyl, alkanoylamino optionally substituted by cycloalkyl of 3 to 6 carbon atoms, alkoxycarbonylamino, alkanoyl, benzoyl or N-methylmethanesulphonylamino, and Y is primary amino or substituted amino, possess anthelmintic and anti-viral activity. New compounds within that formula possess fungicidal properties.

摘要翻译： 下式的苯衍生物：其中R是任选被卤素或烷氧基取代的1至4个碳原子的脂族烃基，R 1是氢或甲基，R 2是氢，卤素，烷基，烷酰基氨基，任选地被 3至6个碳原子，烷氧基羰基氨基，烷酰基，苯甲酰基或N-甲基甲磺酰氨基，Y是伯氨基或取代氨基，具有驱虫和抗病毒活性。 该配方中的新化合物具有杀菌性。

公开(公告)号：US4048326A

公开(公告)日：1977-09-13

申请号：US153409

申请日：1971-06-15

申请人： Samuel Sidney Berg ,  David Conwil Jenkins ,  Ronald Frederick Phillipson

发明人： Samuel Sidney Berg ,  David Conwil Jenkins ,  Ronald Frederick Phillipson

IPC分类号： C07C335/28 ,  C07D295/14 ,  A61K31/27

CPC分类号： C07D295/14 ,  C07C335/28

摘要： Benzene derivative of the formula: ##STR1## wherein R and R.sup.1 each represent an aliphatic hydrocarbon group optionally substituted by halogen or alkoxy, R.sup.2 and R.sup.3 each represent hydrogen or methyl, and R.sup.4 represents hydrogen, halogen, alkyl, alkanoylamino optionally substituted by cycloalkyl of 3 to 6 carbon atoms, alkoxycarbonylamino, alkanoyl, benzyl or N-methylmethanesulphonylamino, possess anthelmintic and anti-viral activity. New compounds within that formula also possess fungicidal properties.

摘要翻译： 下式的苯衍生物：其中R和R 1各自表示任选被卤素或烷氧基取代的脂族烃基，R 2和R 3各自表示氢或甲基，R 4表示氢，卤素，烷基，烷酰基氨基， 3至6个碳原子，烷氧基羰基氨基，烷酰基，苄基或N-甲基甲磺酰氨基具有驱虫和抗病毒活性。 该配方中的新化合物也具有杀菌性。