公开(公告)号：US07473669B2

公开(公告)日：2009-01-06

申请号：US11417327

申请日：2006-05-03

申请人： Steven Howard Shaber ,  Maurice Chee Hoong Yap ,  Kevin Gerald Meyer ,  Noormohamed Mohamed Niyaz ,  Brent Jeffrey Rieder ,  Michael Thomas Sullenberger ,  William Randal Erickson ,  Frisby Davis Smith

发明人： Steven Howard Shaber ,  Maurice Chee Hoong Yap ,  Kevin Gerald Meyer ,  Noormohamed Mohamed Niyaz ,  Brent Jeffrey Rieder ,  Michael Thomas Sullenberger ,  William Randal Erickson ,  Frisby Davis Smith

IPC分类号： C07D253/06 ,  C07D253/065 ,  C07D253/10 ,  A01N43/707 ,  A61K31/53

CPC分类号： C07D253/06 ,  A01N43/707 ,  C07D401/04 ,  C07D401/06 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/04 ,  C07D409/10 ,  C07D409/14 ,  C07D413/06 ,  C07D413/10 ,  C07D417/12 ,  C07F7/0812

摘要： This invention relates to substituted dihydrotriazinones, triazinones and related compounds, compositions comprising such compounds and an agronomically acceptable carrier, and the use thereof as broad spectrum fungicides. This invention also teaches methods of preparing these compounds as well as methods of using the compounds as fungicides.

摘要翻译： 本发明涉及取代的二氢三嗪酮，三嗪酮和相关化合物，包含这些化合物和农艺学上可接受的载体的组合物及其作为广谱杀真菌剂的用途。 本发明还教导了制备这些化合物的方法以及使用该化合物作为杀真菌剂的方法。

公开(公告)号：US07531482B2

公开(公告)日：2009-05-12

申请号：US11255448

申请日：2005-10-21

申请人： William Kirkland Brewster ,  David Anthony Demeter ,  William Randal Erickson ,  Carla Jean Rasmussen Klittich ,  Christian Thomas Lowe ,  Brent Jeffrey Rieder ,  Jaime Susanne Nugent ,  Carla Nanette Yerkes ,  Yuanming Zhu ,  Terry William Balko

发明人： William Kirkland Brewster ,  David Anthony Demeter ,  William Randal Erickson ,  Carla Jean Rasmussen Klittich ,  Christian Thomas Lowe ,  Brent Jeffrey Rieder ,  Jaime Susanne Nugent ,  Carla Nanette Yerkes ,  Yuanming Zhu ,  Terry William Balko

IPC分类号： C07D495/04 ,  A01N43/90

CPC分类号： C07D498/04 ,  A01N43/90 ,  C07D519/00

摘要： The present invention relates to thieno[2,3-d]-pyrimidine compounds having fungicidal activity. Specifically, the present invention relates to compounds having the Formula (I): wherein each R1, R2 and R3 is independently selected from the group consisting of H, halogen, and alkyl; A is selected from the group consisting of H and alkyl; W is selected from the group consisting of NH and O; D is selected from O, NH and S; E is (—C(O)—)p—R′, wherein p is 0 or 1 and R′ is selected from the group consisting of optionally substituted rings selected from phenyl. furanyl, pyridinyl, pyridinyl-N-oxide, pyrimidinyl, pyridazinyl, pyrazinyl, thiazolyl, triazinyl, thiadiazolyl, oxazolyl, isoxazolyl, thienopyrimidinyl, and pyrimidine fused with an aromatic or heteroaromatic ring selected from bejizene, oxazole, isoxazole, furan, thiazole, pyrimidine, pyridine, pyrrole, pyrazine, and thionhene; each ring being ontionally substituted with one or more substituents selected from the group consisting of alkyl, alkenyl, alkynyl, halogen, haloalkyl, alkoxy, haloalkoxy, nitro, cyano, alkylsulfonyl, alkylsulfoxide, alkylthio, alkoxyiminoalkyl, alkylcarbonyl, alkoxycarbonyl, aminocarbonyl, hydroxycarbonyl, phenyicarbonyl, forrnyl, hydrazidocarbonyl, amidoamino, pyrazolyl, triazolonyl, oxadiazolyl, phenyl, nyridinyl, and phenoxyalkyl; B is selected from the group consisting of halogen, alkyl, haloalkyl, and haloalkoxy; n is an integer from 0 to 3; and m is an integer from 0 to 4 with the proviso that when D is O or S and E is phenyl, then E is not further substituted with halogen.

摘要翻译： 本发明涉及具有杀真菌活性的噻吩并[2,3-d]嘧啶化合物。 具体地，本发明涉及具有式（I）的化合物：其中每个R 1，R 2和R 3独立地选自H，卤素和烷基; A选自H和烷基; W选自NH和O; D选自O，NH和S; E是（-C（O） - ）p -R'，其中p是0或1，R'选自任选取代的选自苯基的环。 呋喃基，吡啶基，吡啶基-N-氧化物，嘧啶基，哒嗪基，吡嗪基，噻唑基，三嗪基，噻二唑基，恶唑基，异恶唑基，噻吩并嘧啶基和与选自异丁唑，恶唑，异恶唑，呋喃，噻唑，嘧啶的芳族或杂芳环稠合的嘧啶 ，吡啶，吡咯，吡嗪和噻吩; 每个环被一个或多个选自烷基，烯基，炔基，卤素，卤代烷基，烷氧基，卤代烷氧基，硝基，氰基，烷基磺酰基，烷基亚砜，烷硫基，烷氧基亚氨基烷基，烷基羰基，烷氧基羰基，氨基羰基，羟基羰基， 苯基羰基，芳基，酰肼基，吡唑基，三唑基，恶二唑基，苯基，吡啶基和苯氧基烷基; B选自卤素，烷基，卤代烷基和卤代烷氧基; n为0〜3的整数。 且m为0至4的整数，条件是当D为O或S且E为苯基时，E不再被卤素取代。

公开(公告)号：US08008487B2

公开(公告)日：2011-08-30

申请号：US11256117

申请日：2005-10-21

申请人： William Kirkland Brewster ,  Carla Jean Rasmussen Klittich ,  Terry William Balko ,  Nneka Tuere Breaux ,  William Randal Erickson ,  James Edward Hunter ,  Christian Thomas Lowe ,  Michael John Ricks ,  Thomas Lyman Siddall ,  Carla Nanette Yerkes ,  Yuanming Zhu

发明人： William Kirkland Brewster ,  Carla Jean Rasmussen Klittich ,  Terry William Balko ,  Nneka Tuere Breaux ,  William Randal Erickson ,  James Edward Hunter ,  Christian Thomas Lowe ,  Michael John Ricks ,  Thomas Lyman Siddall ,  Carla Nanette Yerkes ,  Yuanming Zhu

IPC分类号： C07D495/04 ,  C07D519/00 ,  A01N43/90 ,  A01N43/48 ,  A01N43/10

CPC分类号： A01N43/90 ,  C07D495/04

摘要： The present invention provides compounds of formula (I), thieno[2,3-d]pyrimidines, having fungicidal activity.

摘要翻译： 本发明提供具有杀真菌活性的式（I）化合物噻吩并[2,3-d]嘧啶。