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公开(公告)号:US10189812B2
公开(公告)日:2019-01-29
申请号:US15504245
申请日:2015-06-29
申请人: THE KEY LABORATORY OF CHEMISTRY FOR NATURAL PRODUCTS OF GUIZHOU PROVINCE AND CHINESE ACADEMY OF SCIENCES , VERSITECH LTD.
发明人: Weidong Pan , Yibin Feng , Yazhou Liu , Ning Wang , Lan Huang , Guangyi Liang , Maosheng Zhang , Tianlei Li , Huayong Lou , Zhanxing Hu , Sheng Liu , Peixue Cao , Jinghua Ruan , Junjie Lan , Chao Chen
IPC分类号: C07D491/18 , A61K31/4748 , C07D401/12 , C07D405/14 , C07D409/14 , C07D491/16
摘要: The invention disclosed a compound of general formula (I), a single stereoisomer thereof, a mixture of stereoisomers thereof, and a prodrug, pharmaceutically acceptable salt and metabolite thereof, X1, X2, X3, X4, R1, R2, x, y and z being as defined in the present invention.
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2.
公开(公告)号:US20170260161A1
公开(公告)日:2017-09-14
申请号:US15504245
申请日:2015-06-29
申请人: THE KEY LABORATORY OF CHEMISTRY FOR NATURAL PRODUCTS OF GUIZHOU PROVINCE AND CHINESE ACADEMY , VERSITECH LTD.
发明人: Weidong Pan , Yibin Feng , Yazhou Liu , Ning Wang , Lan Huang , Guangyi Liang , Maosheng Zhang , Tianlei Li , Huayong Lou , Zhanxing Hu , Sheng Liu , Peixue Cao , Jinghua Ruan , Junjie Lan , Chao Chen
IPC分类号: C07D401/12 , C07D409/14 , C07D405/14
CPC分类号: C07D401/12 , C07D405/14 , C07D409/14 , C07D491/16 , C07D491/18
摘要: The invention disclosed a compound of general formula (I), a single stereoisomer thereof, a mixture of stereoisomers thereof, and a prodrug, pharmaceutically acceptable salt and metabolite thereof, X1, X2, X3, X4, R1, R2, x, y and z being as defined in the present invention.
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