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公开(公告)号:US07943629B2
公开(公告)日:2011-05-17
申请号:US11759479
申请日:2007-06-07
申请人: Ulrich Luecking , Duy Nguyen , Arne von Bonin , Oliver von Ahsen , Gerhard Siemeister , Rolf Jautelat , Wolf-Dietrich Doecke
发明人: Ulrich Luecking , Duy Nguyen , Arne von Bonin , Oliver von Ahsen , Gerhard Siemeister , Rolf Jautelat , Wolf-Dietrich Doecke
IPC分类号: C07D239/48 , A61K31/506
CPC分类号: C07D401/12 , C07D239/48
摘要: The invention relates to sulphimides as protein kinase inhibitors of the general formula I
摘要翻译: 本发明涉及作为通式I的蛋白激酶抑制剂的硫酰亚胺
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公开(公告)号:US20080058358A1
公开(公告)日:2008-03-06
申请号:US11759479
申请日:2007-06-07
申请人: Ulrich Luecking , Duy Nguyen , Arne von Bonin , Oliver von Ahsen , Gerhard Siemeister , Rolf Jautelat , Wolf-Dietrich Doecke
发明人: Ulrich Luecking , Duy Nguyen , Arne von Bonin , Oliver von Ahsen , Gerhard Siemeister , Rolf Jautelat , Wolf-Dietrich Doecke
IPC分类号: A61K31/505 , A61K31/506 , A61P35/00 , C07D239/30 , C07D239/48 , C07D401/12
CPC分类号: C07D401/12 , C07D239/48
摘要: The invention relates to sulphimides as protein kinase inhibitors of the general formula I
摘要翻译: 本发明涉及作为通式I的蛋白激酶抑制剂的硫酰亚胺
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3.SULPHOXIMINE-SUBSTITUTED QUINAZOLINE DERIVATIVES AS IMMUNO-MODULATORS, THEIR PREPARATION AND USE AS MEDICAMENTS 有权
标题翻译: 作为免疫调节剂的磺酰嘧啶取代的喹唑啉衍生物,其制备和用作药物公开(公告)号:US20090186911A1
公开(公告)日:2009-07-23
申请号:US12138879
申请日:2008-06-13
申请人: Duy NGUYEN , Arne von Bonin , Michael Haerter , Hartmut Schirok , Anne Mengel , Martina Schaefer , Oliver von Ahsen
发明人: Duy NGUYEN , Arne von Bonin , Michael Haerter , Hartmut Schirok , Anne Mengel , Martina Schaefer , Oliver von Ahsen
IPC分类号: A61K31/517 , C07D239/94 , C07D403/12 , C07D417/12 , C07D401/12 , C07D413/12 , A61P29/00 , A61P37/00
CPC分类号: C07D239/94 , C07C381/10 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12
摘要: The present invention relates to sulphoximine-substituted quinazoline derivatives of the formula (I), processes for their preparation and their use as a medicament for the treatment of various diseases.
摘要翻译: 本发明涉及式(I)的磺酰亚胺取代的喹唑啉衍生物,其制备方法及其作为治疗各种疾病的药物的用途。
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4.Sulphoximine-substituted quinazoline derivatives as immuno-modulators, their preparation and use as medicaments 有权
标题翻译: 磺酰亚胺取代的喹唑啉衍生物作为免疫调节剂,其制备和用作药物公开(公告)号:US07863283B2
公开(公告)日:2011-01-04
申请号:US12138879
申请日:2008-06-13
申请人: Duy Nguyen , Arne von Bonin , Michael Haerter , Hartmut Schirok , Anne Mengel , Martina Schaefer , Oliver von Ahsen
发明人: Duy Nguyen , Arne von Bonin , Michael Haerter , Hartmut Schirok , Anne Mengel , Martina Schaefer , Oliver von Ahsen
IPC分类号: A61K31/517
CPC分类号: C07D239/94 , C07C381/10 , C07D401/12 , C07D403/12 , C07D413/12 , C07D417/12
摘要: The present invention relates to sulphoximine-substituted quinazoline derivatives of the formula (I), processes for their preparation and their use as a medicament for the treatment of various diseases.
摘要翻译: 本发明涉及式(I)的磺酰亚胺取代的喹唑啉衍生物,其制备方法及其作为治疗各种疾病的药物的用途。
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