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公开(公告)号:US20080103129A1
公开(公告)日:2008-05-01
申请号:US11858972
申请日:2007-09-21
申请人: Yue-Mei Zhang , Bangping Xiang , Shyh-Ming Yang , Kenneth Rhodes , Robert Scannevin , Paul Jackson , Davraj Chakravarty , Xiaodong Fan , Lawrence Wilson , Prabha Karnachi
发明人: Yue-Mei Zhang , Bangping Xiang , Shyh-Ming Yang , Kenneth Rhodes , Robert Scannevin , Paul Jackson , Davraj Chakravarty , Xiaodong Fan , Lawrence Wilson , Prabha Karnachi
IPC分类号: A61K31/55 , A61P35/00 , A61P25/00 , C07D403/02 , C07D223/02
CPC分类号: C07D413/06 , C07D211/94 , C07D213/69 , C07D213/89 , C07D223/12 , C07D225/02 , C07D243/08 , C07D401/12 , C07D403/12 , C07D409/12
摘要: This invention provides novel heterocyclic derived matrix metalloprotease inhibitors of the formula: and pharmaceutical compositions comprising same, useful for treating disorders ameliorated by antagonizing matrix metalloproteases. This invention also provides therapeutic and prophylactic methods using the instant pharmaceutical compositions.
摘要翻译: 本发明提供下式的新型杂环衍生基质金属蛋白酶抑制剂:包含其的药物组合物,可用于治疗通过拮抗基质金属蛋白酶而改善的病症。 本发明还提供了使用本发明的药物组合物的治疗和预防方法。
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公开(公告)号:US20100279986A1
公开(公告)日:2010-11-04
申请号:US12834283
申请日:2010-07-12
申请人: Yue-Mei ZHANG , Bangping Xiang , Shyh-Ming Yang , Kenneth Rhodes , Robert Scannevin , Paul Jackson , Davraj Chakravarty , Xiaodong Fan , Lawrence J. Wilson , Prabha Karnachi
发明人: Yue-Mei ZHANG , Bangping Xiang , Shyh-Ming Yang , Kenneth Rhodes , Robert Scannevin , Paul Jackson , Davraj Chakravarty , Xiaodong Fan , Lawrence J. Wilson , Prabha Karnachi
IPC分类号: A61K31/55 , A61K31/635 , A61K31/4412 , A61K31/5377 , A61K31/45 , A61K31/4436 , A61K31/551 , A61K31/541 , A61P9/00 , A61P9/14 , A61P35/00 , A61P29/00 , A61P25/00 , A61P25/28 , A61P25/14 , A61P19/02 , A61P1/04
CPC分类号: C07D413/06 , C07D211/94 , C07D213/69 , C07D213/89 , C07D223/12 , C07D225/02 , C07D243/08 , C07D401/12 , C07D403/12 , C07D409/12
摘要: This invention provides novel heterocyclic derived matrix metalloprotease inhibitors of the formula: and pharmaceutical compositions comprising same, useful for treating disorders ameliorated by antagonizing matrix metalloproteases. This invention also provides therapeutic and prophylactic methods using the instant pharmaceutical compositions.
摘要翻译: 本发明提供下式的新型杂环衍生基质金属蛋白酶抑制剂:包含其的药物组合物,可用于治疗通过拮抗基质金属蛋白酶而改善的病症。 本发明还提供了使用本发明的药物组合物的治疗和预防方法。
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公开(公告)号:US07803793B2
公开(公告)日:2010-09-28
申请号:US11858972
申请日:2007-09-21
申请人: Yue-Mei Zhang , Bangping Xiang , Shyh-Ming Yang , Kenneth Rhodes , Robert Scannevin , Paul Jackson , Davraj Chakravarty , Xiaodong Fan , Lawrence J. Wilson , Prabha Karnachi
发明人: Yue-Mei Zhang , Bangping Xiang , Shyh-Ming Yang , Kenneth Rhodes , Robert Scannevin , Paul Jackson , Davraj Chakravarty , Xiaodong Fan , Lawrence J. Wilson , Prabha Karnachi
IPC分类号: C07D225/02 , C07D401/06 , C07D401/12 , C07D409/12 , A61K31/55
CPC分类号: C07D413/06 , C07D211/94 , C07D213/69 , C07D213/89 , C07D223/12 , C07D225/02 , C07D243/08 , C07D401/12 , C07D403/12 , C07D409/12
摘要: This invention provides novel heterocyclic derived matrix metalloprotease inhibitors of the formula: and pharmaceutical compositions comprising same, useful for treating disorders ameliorated by antagonizing matrix metalloproteases. This invention also provides therapeutic and prophylactic methods using the instant pharmaceutical compositions.
摘要翻译: 本发明提供下式的新型杂环衍生基质金属蛋白酶抑制剂:包含其的药物组合物,可用于治疗通过拮抗基质金属蛋白酶而改善的病症。 本发明还提供了使用本发明的药物组合物的治疗和预防方法。
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