公开(公告)号：WO1998017663A1

公开(公告)日：1998-04-30

申请号：PCT/KR1997000188

申请日：1997-10-08

Applicant: CHOONGWAE PHARMA CORPORATION ,  MOON, Sung, Hwan ,  CHOI, Hea, Jin ,  LEE, Su, Jin ,  CHUNG, Jea, Uk ,  KIM, Jai, Hyun ,  CHUNG, Dong, Hoon ,  PARK, Moon, Soo ,  CHO, In, Koo ,  CHOI, Kun, Hyock

Inventor： CHOONGWAE PHARMA CORPORATION

IPC: C07D311/94

CPC classification number: C07D311/94

Abstract: The present invention relates to a novel genipin derivative represented by formula (I), which has anti hepatitis B virus (HBV) activity, in which R1 represents lower alkyl, benzyl, etc., R2 represents hydroxymethyl, formyl, acetyl, etc., R3 represents methoxycarbonyl, formyl, etc., its pharmaceutically acceptable salt, and stereoisomer.

Abstract translation: 本发明涉及具有抗乙型肝炎病毒（HBV）活性的式（I）表示的新型京尼平衍生物，其中R1表示低级烷基，苄基等，R2表示羟甲基，甲酰基，乙酰基等， R3表示甲氧基羰基，甲酰基等，其药学上可接受的盐和立体异构体。