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1.DERIVATIVES OF N- [(1H-PYRAZOL-1-YL) ARYL] - 1H - INDOLE OR 1H - INDAZOLE - 3 - CARBOXAMIDE, THEIR PREPARATION AND THEIR USE AS P2Y12 ANTAGONISTS 审中-公开
Title translation: N- [(1H-吡咯烷-1-基)亚甲基] -1H-吲哚或1H-吲唑-3-羧酰胺的衍生物,其制备及其作为P2Y12拮抗剂的用途公开(公告)号:WO2012146318A1
公开(公告)日:2012-11-01
申请号:PCT/EP2011/065885
申请日:2011-09-13
Applicant: SANOFI , BADORC, Alain , BOLDRON, Christophe , DELESQUE, Nathalie , FOSSEY, Valérie , LASSALLE, Gilbert , YVON, Xavier
Inventor: BADORC, Alain , BOLDRON, Christophe , DELESQUE, Nathalie , FOSSEY, Valérie , LASSALLE, Gilbert , YVON, Xavier
IPC: C07D403/12 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D471/04 , C07D471/08 , C07D487/04 , C07D487/08 , A61K31/455 , A61K31/439 , A61K31/497 , A61K31/501 , A61K31/506 , A61P9/00
CPC classification number: C07D403/12 , C07D401/14 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D471/08 , C07D487/04 , C07D487/08
Abstract: The present invention relates to compounds corresponding to formula (I) and their use as P2Y12 antagonists for the treatment of cardiovascular diseases.
Abstract translation: 本发明涉及式(I)化合物及其作为P2Y12拮抗剂治疗心血管疾病的用途。