公开(公告)号：WO2005023805A1

公开(公告)日：2005-03-17

申请号：PCT/IN2003/000421

申请日：2003-12-31

Applicant: DESHPANDE, Prasad K ,  DESAI, Vijaya N ,  YEOLE, Ravindra D ,  GUPTE, Shrikant V ,  PATEL, Mahesh V ,  DE SOUZA, Noel J

Inventor： DESHPANDE, Prasad K ,  DESAI, Vijaya N ,  YEOLE, Ravindra D ,  GUPTE, Shrikant V ,  PATEL, Mahesh V ,  DE SOUZA, Noel J

IPC: C07D455/04

CPC classification number: C07D471/06

Abstract: The invention relates to crystalline S-(-)-9-fluoro-6,7-dihydro-8-(4-hydroxypiperidin-1-yl)-5-methyl-1-oxo-1H,5H-benzo[i,j]quinolizine-2-carboxylic acid L-arginine salt tetrahydrate, a process for its preparation and pharmaceutical formulations incorporating it as the active ingredient for use in treating microbial infections.

Abstract translation: 本发明涉及结晶S - （ - ） - 9-氟-6,7-二氢-8-（4-羟基哌啶-1-基）-5-甲基-1-氧代-1H，5H-苯并[i，j ]喹嗪-2羧酸L-精氨酸盐四水合物，其制备方法和将其作为用于治疗微生物感染的活性成分的药物制剂。

公开(公告)号：WO2004108744A2

公开(公告)日：2004-12-16

申请号：PCT/IN2004/000137

申请日：2004-05-18

Applicant: DESHPANDE, Prasad, K ,  SINDKHEDKAR, Milind, D ,  DESAI, Vijaya, N ,  GUPTE, Shrikant, V ,  YEOLE, Ravindra, D ,  PATEL, Mahesh, V ,  DE SOUZA, Noel, J

Inventor： DESHPANDE, Prasad, K ,  SINDKHEDKAR, Milind, D ,  DESAI, Vijaya, N ,  GUPTE, Shrikant, V ,  YEOLE, Ravindra, D ,  PATEL, Mahesh, V ,  DE SOUZA, Noel, J

IPC: C07H17/00

CPC classification number: C07H17/00

Abstract: The present invention relates to novel azalides and azaketolides having antimicrobial activity, methods for their preparation, pharmaceutical compositions containing the compounds and methods of treating microbial infections with the compounds.

Abstract translation: 本发明涉及具有抗微生物活性的新型氮杂ides ides ides and az tol tol tol tol for for。。。。。。。。。。。。。。。。。

公开(公告)号：WO2004108744A3

公开(公告)日：2005-03-24

申请号：PCT/IN2004000137

申请日：2004-05-18

Applicant: DESHPANDE PRASAD K ,  SINDKHEDKAR MILIND D ,  DESAI VIJAYA N ,  GUPTE SHRIKANT V ,  YEOLE RAVINDRA D ,  PATEL MAHESH V ,  DE SOUZA NOEL J

Inventor： DESHPANDE PRASAD K ,  SINDKHEDKAR MILIND D ,  DESAI VIJAYA N ,  GUPTE SHRIKANT V ,  YEOLE RAVINDRA D ,  PATEL MAHESH V ,  DE SOUZA NOEL J

IPC: C07H17/00 ,  C07H17/08 ,  A61K31/7048

CPC classification number: C07H17/00

Abstract: The present invention relates to novel azalides and azaketolides having antimicrobial activity, methods for their preparation, pharmaceutical compositions containing the compounds and methods of treating microbial infections with the compounds.

Abstract translation: 本发明涉及具有抗微生物活性的新型氮杂ides ides ides and az tol tol tol tol for for。。。。。。。。。。。。。。。。。。