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1.N-((6-AMINO-PYRIDIN-3-YL)METHYL)-HETEROARYL-CARBOXAMIDES AS INHIBITORS OF PLASMA KALLIKREIN 审中-公开
Title translation: N - ((6-氨基 - 吡啶-3-基)甲基) - 乙酰胆碱酰胺作为血浆KALLIKREIN的抑制剂公开(公告)号:WO2012017020A1
公开(公告)日:2012-02-09
申请号:PCT/EP2011/063389
申请日:2011-08-03
Applicant: NOVARTIS AG , BRANDL, Trixi , FLOHR, Stefanie , KOPEC, Sebastian , LACHAL, Julie , MARKERT, Christian , NAMOTO, Kenji , NGANGA, Perle , PIRARD, Bernard , RENATUS, Martin , SEDRANI, Richard , ZOLLER, Thomas
Inventor: BRANDL, Trixi , FLOHR, Stefanie , KOPEC, Sebastian , LACHAL, Julie , MARKERT, Christian , NAMOTO, Kenji , NGANGA, Perle , PIRARD, Bernard , RENATUS, Martin , SEDRANI, Richard , ZOLLER, Thomas
IPC: C07D405/14 , C07D403/12 , C07D413/12 , C07D403/14 , C07D417/14 , C07D409/14 , A61K31/4439 , A61P7/02
CPC classification number: C07D409/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D413/12 , C07D417/14
Abstract: The invention relates to compound of the formula (I) in which the substituents are as defined in the specification; in free form or in salt form; to its preparation, to its use as medicament and to medicaments comprising it.
Abstract translation: 本发明涉及式(I)化合物,其中取代基如说明书中所定义; 以游离形式或盐形式; 作为其制备,用作药物和包含它的药物。