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1.发明申请NOVEL CRYSTALLINE FORMS OF 2, 3 DIMETHYL-8- (2, 6-DIMETHYLBENZYLAMINO) -N-HYDROXYETHYL-IMIDAZO [1, 2-A] PYRIDINE-6-CARBOXAMIDE MESYLATE SALT. 审中-公开2,6-二甲基-8-（2,6-二甲基苯甲酰氨基）-N-羟基乙基咪唑并[1,2-A]吡啶-6-羧酰胺盐酸盐的新型结晶形式。
公开(公告)号：WO2005058895A1
公开(公告)日：2005-06-30
申请号：PCT/SE2004/001909
申请日：2004-12-16
Applicant: ASTRAZENECA AB , LILLJEQUIST, Lars , LINDKVIST, Maria , NORDBERG, Peter , PETTERSSON, Ursula , SEBHATU, Tesfai
Inventor： LILLJEQUIST, Lars , LINDKVIST, Maria , NORDBERG, Peter , PETTERSSON, Ursula , SEBHATU, Tesfai
IPC: C07D471/04
CPC classification number: C07D471/04
Abstract: The present invention relates to novel crystalline forms of 2,3-dimethyl-8-(2,6-dimethylbenzylamino)-N-hydroxyethyl-imidazo[1,2-a]pyridine-6-carboxamide mesylate salt and to mixture thereof. Further, the present invention also relates to processes for obtaining them, the use of said compounds for the treatment of gastrointestinal disorders, and pharmaceutical compositions containing them.
Abstract translation: 本发明涉及2,3-二甲基-8-（2,6-二甲基苄基氨基）-N-羟乙基 - 咪唑并[1,2-a]吡啶-6-甲酰胺甲磺酸盐的新结晶形式及其混合物。 此外，本发明还涉及获得它们的方法，所述化合物在治疗胃肠道疾病中的用途，以及含有它们的药物组合物。
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2.发明申请NOVEL PROCESS FOR MAKING (2R)-(3-AMINO-2-FLUOROPROPYL)PHOSPHINIC ACID FORM A 审中-公开制备（2R） - （3-氨基-2-氟代丙烯）磷酸形式A的新方法
公开(公告)号：WO2009082344A1
公开(公告)日：2009-07-02
申请号：PCT/SE2008/051491
申请日：2008-12-18
Applicant: ASTRAZENECA AB , ABBASI, Hassan , FINNHULT, Daniel , KRIG, Ann-Sofie , LILLJEQUIST, Lars , LUNDBLAD, Karin , RECKNAGEL, Mikaela , STENEMYR, Anna , TJERNELD, Erica
Inventor： ABBASI, Hassan , FINNHULT, Daniel , KRIG, Ann-Sofie , LILLJEQUIST, Lars , LUNDBLAD, Karin , RECKNAGEL, Mikaela , STENEMYR, Anna , TJERNELD, Erica
CPC classification number: C07F9/4816
Abstract: The present invention is directed to a novel process for the preparation of the crystalline form A of (2 R )-(3-amino-2-fluoropropyl)phosphinic acid.
Abstract translation: 本发明涉及制备（2R） - （3-氨基-2-氟丙基）次膦酸的结晶形式A的新方法。
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