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公开(公告)号:WO2004039410A2
公开(公告)日:2004-05-13
申请号:PCT/IB0304698
申请日:2003-10-24
Applicant: PFIZER PROD INC , SHALABY SHALABY WAHBA , SHAH JAYMIN CHANDRAKANT , POLY MED INC
Inventor: SHALABY SHALABY WAHBA , SHAH JAYMIN CHANDRAKANT
IPC: A61K47/48
CPC classification number: A61K47/593 , A61K47/59 , A61K47/60
Abstract: A liquid phase conjugate formed of a bioactive agent such as a drug compound, e.g. ziprasidone, and a liquid polymer of requisite functionally is disclosed.
Abstract translation: 由生物活性剂如药物化合物形成的液相共轭体, 齐拉西酮和功能性必需的液体聚合物。
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公开(公告)号:WO0009166A2
公开(公告)日:2000-02-24
申请号:PCT/US9918146
申请日:1999-08-10
Applicant: POLY MED INC , SHALABY SHALABY WAHBA , CORBETT JOEL THOMAS
Inventor: SHALABY SHALABY WAHBA , CORBETT JOEL THOMAS
CPC classification number: A61K47/593
Abstract: The present invention is directed to absorbable polyesters comprising one or more monophosphate functionality; a conjugate comprising the foregoing polyester and a peptide and/or a bioactive agent; microparticles comprising an absorbable polyester; a conjugate comprising the microparticles and a peptide and/or a bioactive agent; an acylated or alkylated polysaccharide having one or more monophosphate functionality; a conjugate comprising the acylated or alkylated polysaccharide and a peptide and/or a bioactive agent; and pharmaceutical compositions thereof.
Abstract translation: 本发明涉及包含一种或多种单磷酸官能团的可吸收聚酯; 包含上述聚酯和肽和/或生物活性剂的共轭物; 包含可吸收聚酯的微粒; 包含微粒和肽和/或生物活性剂的缀合物; 具有一个或多个单磷酸官能团的酰化或烷基化多糖; 包含酰化或烷基化多糖和肽和/或生物活性剂的缀合物; 及其药物组合物。
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公开(公告)号:WO2004039411A3
公开(公告)日:2004-05-13
申请号:PCT/IB2003/004699
申请日:2003-10-24
Applicant: PFIZER PRODUCTS INC. , POLY-MED INC. , SHALABY, Shalaby, Wahba , SHAH, Jaymin, Chandrakant , CORBETT, Joel, Thomas
IPC: A61K47/48
Abstract: Aqueous solubility of drugs suich as ziproasidone is improved using a functional polymer to form an ionic conjugate with said drug.
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公开(公告)号:WO2004039411A2
公开(公告)日:2004-05-13
申请号:PCT/IB0304699
申请日:2003-10-24
Applicant: PFIZER PROD INC , SHALABY SHALABY WAHBA , SHAH JAYMIN CHANDRAKANT , CORBETT JOEL THOMAS , POLY MED INC
Inventor: SHALABY SHALABY WAHBA , SHAH JAYMIN CHANDRAKANT , CORBETT JOEL THOMAS
IPC: A61K47/48
CPC classification number: A61K47/593 , A61K47/59 , A61K47/60
Abstract: Aqueous solubility of drugs suich as ziproasidone is improved using a functional polymer to form an ionic conjugate with said drug.
Abstract translation: 使用功能性聚合物与所述药物形成离子结合物,改善了作为拉伐西坦的药物的水溶性。
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公开(公告)号:WO2004039410A3
公开(公告)日:2004-05-13
申请号:PCT/IB2003/004698
申请日:2003-10-24
Applicant: PFIZER PRODUCTS INC. , POLY-MED INC. , SHALABY, Shalaby, Wahba , SHAH, Jaymin, Chandrakant
Inventor: SHALABY, Shalaby, Wahba , SHAH, Jaymin, Chandrakant
IPC: A61K47/48
Abstract: A liquid phase conjugate formed of a bioactive agent such as a drug compound, e.g. ziprasidone, and a liquid polymer of requisite functionally is disclosed.
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