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1.
公开(公告)号:WO2013098833A3
公开(公告)日:2013-10-10
申请号:PCT/IN2012000599
申请日:2012-09-10
Applicant: CADILA HEALTHCARE LTD , DWIVEDI SHRIPRAKASH DHAR , PRASAD ASHOK , PAL DAYA RAM , SHARMA MUKUL HARI PRASAD , JAIN KULDEEP NATWARLAL , PATEL NAITIK BHARATBHAI
Inventor: DWIVEDI SHRIPRAKASH DHAR , PRASAD ASHOK , PAL DAYA RAM , SHARMA MUKUL HARI PRASAD , JAIN KULDEEP NATWARLAL , PATEL NAITIK BHARATBHAI
IPC: C07D413/14 , C07D413/10
CPC classification number: C07D413/14 , C07D265/32 , C07D413/10
Abstract: The invention discloses processes for the preparation of rivaroxaban and its pharmaceutically acceptable salts, solvates, and hydrates thereof. The invention also relates to novel intermediates for the preparation of rivaroxaban.
Abstract translation: 本发明公开了制备利伐沙班及其药学上可接受的盐,溶剂化物和水合物的方法。 本发明还涉及用于制备利伐沙班的新型中间体。
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2.
公开(公告)号:WO2013098833A2
公开(公告)日:2013-07-04
申请号:PCT/IN2012/000599
申请日:2012-09-10
Applicant: CADILA HEALTHCARE LIMITED , DWIVEDI, Shriprakash, Dhar , PRASAD, Ashok , PAL, Daya, Ram , SHARMA, Mukul, Hari, Prasad , JAIN, Kuldeep, Natwarlal , PATEL, Naitik, Bharatbhai
Inventor: DWIVEDI, Shriprakash, Dhar , PRASAD, Ashok , PAL, Daya, Ram , SHARMA, Mukul, Hari, Prasad , JAIN, Kuldeep, Natwarlal , PATEL, Naitik, Bharatbhai
IPC: C07D413/14 , C07D413/10
CPC classification number: C07D413/14 , C07D265/32 , C07D413/10
Abstract: The invention discloses processes for the preparation of rivaroxaban and its pharmaceutically acceptable salts, solvates, and hydrates thereof. The invention also relates to novel intermediates for the preparation of rivaroxaban.
Abstract translation: 本发明公开了制备利伐沙班及其药学上可接受的盐,溶剂化物和水合物的方法。 本发明还涉及制备利伐沙班的新型中间体。 p>
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