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1.SMALL- MOLECULE BINDING SITE ON PRO-APOPTOTIC BAX REGULATES INHIBITION OF BAX ACTIVITY 审中-公开
Title translation: 小分子结合位点对BAX活性的抑制作用公开(公告)号:WO2014110476A2
公开(公告)日:2014-07-17
申请号:PCT/US2014/011213
申请日:2014-01-13
Inventor: GAVATHIOTIS, Evripidis , GARNER, Thomas
IPC: G01N33/53
CPC classification number: A61K31/7028 , A61K31/11 , A61K31/325 , A61K31/47 , A61K31/4709 , A61K31/496 , A61K31/4985 , A61K31/506 , A61K31/53 , A61K31/5377 , A61K31/546 , A61K31/675 , G01N33/5008 , G01N33/53 , G01N2510/00
Abstract: Methods are provided for identifying an agent as a selective inhibitor of a Bcl-2-associated x-protein (BAX).
Abstract translation: 提供了用于鉴定作为Bcl-2相关x-蛋白(BAX)的选择性抑制剂的试剂的方法。