Invention Application
- Patent Title: Carbapenem compound crystals and injection preparations
- Patent Title (中): 碳青霉烯复合晶体和注射剂
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Application No.: US11259509Application Date: 2005-10-26
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Publication No.: US20060040916A1Publication Date: 2006-02-23
- Inventor: Hiroyuki Chiba , Masahiko Tsujii , Astsushi Koiwa , Shin Sakurai , Akio Kayano , Hiroyuki Ishizuka , Hiroyuki Saito , Taiju Nakamura , Ikuo Kushida , Yasuyuki Suzuki , Takako Yoshiba , Kazuhide Ashizawa , Masahiro Sakurai , Eiichi Yamamoto
- Applicant: Hiroyuki Chiba , Masahiko Tsujii , Astsushi Koiwa , Shin Sakurai , Akio Kayano , Hiroyuki Ishizuka , Hiroyuki Saito , Taiju Nakamura , Ikuo Kushida , Yasuyuki Suzuki , Takako Yoshiba , Kazuhide Ashizawa , Masahiro Sakurai , Eiichi Yamamoto
- Assignee: EISAI CO., LTD.
- Current Assignee: EISAI CO., LTD.
- Priority: JP11-156810 19990603; JP2000-153891 20000525
- Main IPC: C07D487/04
- IPC: C07D487/04 ; A61K31/407

Abstract:
The present invention provides carbapenem hydrochloride trihydrate crystals, which are chemically stable, easily purified and useful as antimicrobial agents, a process for producing them, and a powdery charged preparation for injection containing them. That is, it provides carbapenem hydrochloride trihydrate crystals having a powdery X-ray diffraction pattern containing lattice distances (d) of 9.0, 4.1 and 2.8 Å, a process for producing them, and a powdery charged preparation for injection containing them.
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