Invention Application
- Patent Title: Substituted n-phenyl sulfonamide bradykinin antagonists
- Patent Title (中): 取代的n-苯基磺酰胺缓激肽拮抗剂
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Application No.: US10527384Application Date: 2003-12-18
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Publication No.: US20070093485A1Publication Date: 2007-04-26
- Inventor: Francine Farouz , Michael Dappen , Ying-Zi Xu , Sarah Bartulis , Ryan Holcomb , Ramesh Kasar , Michael Pleiss , Eugene Thorsett , Xiaocong Ye , Andrei Konradi
- Applicant: Francine Farouz , Michael Dappen , Ying-Zi Xu , Sarah Bartulis , Ryan Holcomb , Ramesh Kasar , Michael Pleiss , Eugene Thorsett , Xiaocong Ye , Andrei Konradi
- Assignee: ELAN PHARMACEUTICALS, INC.
- Current Assignee: ELAN PHARMACEUTICALS, INC.
- International Application: PCT/US03/40745 WO 20031218
- Main IPC: A61K31/5377
- IPC: A61K31/5377 ; A61K31/497 ; A61K31/4965 ; A61K31/496 ; A61K31/4545 ; A61K31/454 ; A61K31/4439 ; A61K31/427 ; A61K31/22 ; C07D417/02 ; C07D403/02

Abstract:
Disclosed are certain substituted N-phenylsulfonamide derivatives and related compounds. These compounds are useful as bradykinin antagonists to relieve adverse symptoms in mammals mediated, at least in part, by bradykinin including pain, inflammation, bronchoconstriction, cerebral edema, etc.
Information query
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