发明申请
- 专利标题： PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL INTERMEDIATE
- 专利标题（中）： 制备药物中间体的方法
-
申请号： US12096630申请日： 2006-12-08
-
公开(公告)号： US20090018337A1公开(公告)日： 2009-01-15
- 发明人: Peter Trinka , Tibor Mezei , Jozsef Reiter , Ferenc Bartha , Zoltan Katona , Gyorgyi Vereczkeyne Donath , Kalman Nagy , Laszlo Pongo
- 申请人： Peter Trinka , Tibor Mezei , Jozsef Reiter , Ferenc Bartha , Zoltan Katona , Gyorgyi Vereczkeyne Donath , Kalman Nagy , Laszlo Pongo
- 优先权： HUP0501138 20051208
- 国际申请： PCT/HU2006/000108 WO 20061208
- 主分类号： C07D241/04
- IPC分类号： C07D241/04
摘要：
The present invention relates to a process for the preparation of {2-[4-(α-phenyl-p-chlorobenzyl)-piperazin-1-yl]-ethoxy}-acetic acid-N,N-dimethylamide of the Formula (I) and enantiomers thereof. The compound of the Formula (I) or enantiomers thereof are important pharmaceutical intermediates suitable for direct transformation into non-sedating antihistamine type pharmaceutical active ingredients cetirizine and levocetirizine.
信息查询
