发明申请
US20110251207A1 BIARYL-SPIROAMINOOXAZOLINE ANALOGUES AS ALPHA 2C ADRENERGIC RECEPTOR MODULATORS
失效
作为ALPHA 2C ADRENERGIC受体调节剂的BIARYL-SPIROAMINOOXAZOLINE ANALOGUES
- 专利标题： BIARYL-SPIROAMINOOXAZOLINE ANALOGUES AS ALPHA 2C ADRENERGIC RECEPTOR MODULATORS
- 专利标题（中）： 作为ALPHA 2C ADRENERGIC受体调节剂的BIARYL-SPIROAMINOOXAZOLINE ANALOGUES
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申请号： US13122679申请日： 2009-10-06
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公开(公告)号： US20110251207A1公开(公告)日： 2011-10-13
- 发明人: Kevin D. McCormick , Li Dong , Christopher W. Boyce , Manuel de Lera Ruiz , Salem Fevrier , Jie Wu , Junying Zheng , Younong Yu , Jianhua Chao , Walter S. Won , Ashwin U. Rao , Rongze Kuang , Pauline C. Ting , Xianhai Huang , Ning Shao , Adandan Palani , Michael Y. Berlin , Robert G. Aslanian
- 申请人： Kevin D. McCormick , Li Dong , Christopher W. Boyce , Manuel de Lera Ruiz , Salem Fevrier , Jie Wu , Junying Zheng , Younong Yu , Jianhua Chao , Walter S. Won , Ashwin U. Rao , Rongze Kuang , Pauline C. Ting , Xianhai Huang , Ning Shao , Adandan Palani , Michael Y. Berlin , Robert G. Aslanian
- 申请人地址： US NJ Rahway
- 专利权人： Merck Sharp & Dohme Corp.
- 当前专利权人： Merck Sharp & Dohme Corp.
- 当前专利权人地址： US NJ Rahway
- 国际申请： PCT/US2009/059636 WO 20091006
- 主分类号： A61K31/501
- IPC分类号： A61K31/501 ; A61K31/506 ; A61K31/4439 ; A61K31/427 ; A61K31/497 ; C07D263/52 ; A61K31/423 ; C07D235/02 ; A61K31/4184 ; C07D405/10 ; C07D409/10 ; A61K31/422 ; C07D403/10 ; A61P27/06 ; A61P25/22 ; A61P21/02 ; A61P9/00 ; A61P25/18 ; A61P25/06 ; A61P25/28 ; A61P3/10 ; A61P11/02 ; C07D413/10
摘要：
In its many embodiments, the present invention provides a novel class of biaryi spiroaminooxazoline analogues as modulators of α2C adrenergic receptor agonists, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more conditions associated with the α2C adrenergic receptors using such compounds or pharmaceutical compositions.
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